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4,6-dimethyl-N-(3-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methoxy}phenyl)pyrimidin-2-amine
6-methyl-3-[2-(piperazin-1-yl)ethyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-methyl-5-{1-[2-(1H-1,2,4-triazol-5-yl)benzoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
3-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-5-methyl-1,2-oxazole
2-{[ethyl(2-hydroxyethyl)amino]methyl}-6-methylquinolin-4-ol
3-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenol
2-(3-phenylpropyl)-4-(pyridin-4-ylmethyl)morpholine
5-{2-[4-(cyclopropylamino)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-2-oxoethyl}imidazolidine-2,4-dione
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
6-methoxy-N-methyl-N-[2-(oxan-2-yl)ethyl]pyrimidin-4-amine
[(3R,4R)-4-[(4-ethylpiperazin-1-yl)methyl]-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl]methanol
6-[3-(5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]pyridine-2-carbonitrile
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carboxamide
1-{7-methylthieno[3,2-d]pyrimidin-4-yl}-4-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperazine
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(1-propylcyclopropyl)acetamide
ethyl 3-[(3-chlorophenyl)methyl]-1-(2-acetamidoacetyl)piperidine-3-carboxylate
2-methyl-6-(1-{pyrazolo[1,5-a]pyridine-7-carbonyl}piperidin-4-yl)pyrimidin-4-ol
4-(4-chloro-2-hydroxybenzoyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
1,5-dimethyl-N-{[1-(4-methylpiperazin-1-yl)cyclopentyl]methyl}-1H-pyrrole-2-carboxamide
4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[(2-methoxyphenyl)methyl]pyridine-2-carboxamide
9-[(2-methylphenyl)methyl]-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-(1-methyl-1H-pyrrol-2-yl)-N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}-1H-pyrazole-5-carboxamide
(1S,5R)-6-benzyl-3-(4-fluoro-2-methylbenzoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}pyridin-2-amine
1-({5-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-ylmethyl]-2-methoxyphenyl}methyl)-1H-1,2,4-triazole
3-(2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamido)propanamide
ethyl 1-(furan-3-carbonyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
2-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
3-(3-chloro-1H-1,2,4-triazol-5-yl)-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]propanamide
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-2-methyl-1-benzofuran-5-carboxamide
2-[(3,4-difluorophenyl)methyl]-8-(9H-purin-6-yl)-2,8-diazaspiro[4.5]decan-3-one
1-(2,3-dihydro-1H-inden-2-yl)-5-(1H-imidazol-5-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazole
2-methoxy-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]pyridine-3-carboxamide
1-({5-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
(1R,5R)-3-methanesulfonyl-6-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
4-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-1-ethylpiperidine
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-(dimethylamino)-2-(2-methylphenyl)acetamide
2-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propane-1,3-diol
methyl 4-(4-{[benzyl(cyclopropylmethyl)amino]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
6-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-{3-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]piperidin-1-yl}pyridine
2-{4-[4-(4-fluorophenyl)piperazine-1-carbonyl]-5-(propan-2-yl)-1H-pyrazol-1-yl}-4-(furan-2-yl)pyrimidine
N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-{[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl](methyl)amino}propanamide
N-(furan-2-ylmethyl)-N-methyl-2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]acetamide
(3R,4S)-1-[4-(morpholine-4-carbonyl)benzoyl]-4-phenylpyrrolidin-3-amine
(3S,4R)-4-(hydroxymethyl)-1-(7-methyl-1-benzofuran-2-carbonyl)piperidin-3-ol
4-[2-(benzyloxy)benzoyl]-1,4-oxazepan-6-ol
2-methyl-8-(1,2,3,4-tetrahydroisoquinolin-5-yl)quinolin-4-ol