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2-(4-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)ethan-1-ol
N-(adamantan-2-ylmethyl)-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-5-methyl-N-(pyridin-4-ylmethyl)pyrazine-2-carboxamide
3-{[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}pyridin-2-amine
2-[(2-{[2-(3-ethylphenoxy)ethyl](methyl)carbamoyl}phenyl)amino]acetic acid
2,6-difluoro-N-[(3R,4R)-3-hydroxypiperidin-4-yl]-3-methylbenzamide
5-methyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-4-{[3-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
5-{2-[(4-oxopiperidin-1-yl)methyl]phenyl}pyridine-3-carboxamide
(1S,4S)-2-(5-chloro-2-methoxyphenyl)-5-(pyridin-2-ylmethyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
2-cyclopropyl-5-(4-methanesulfonylpiperazine-1-carbonyl)-3,4-dihydropyrimidin-4-one
1-(1H-indol-7-ylmethyl)-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
(3-{2-[1-(dimethyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
N4-[3-(3-chlorophenyl)phenyl]-N1,N1-dimethylpiperidine-1,4-dicarboxamide
7-(3-chlorophenyl)-4-(6-methylpyridazin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-benzyl-N-cyclohexyl-N-(thiophen-3-ylmethyl)-1H-pyrazole-4-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}ethan-1-one
N-[(4-acetylmorpholin-2-yl)methyl]hexanamide
6-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(5-methyl-1H-pyrazol-1-yl)propanamide
N-(2-methoxyethyl)-3-{1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl}propanamide
5-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]pyridin-2-amine
1-[3-(2-methyl-1,3-thiazol-4-yl)-5-[(pyridin-4-ylsulfanyl)methyl]-1H-1,2,4-triazol-1-yl]butan-2-ol
5-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}pyridin-2-amine
3-{[(2-hydroxypyridin-3-yl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-N5-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
5-chloro-N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
9-[(2-methoxyphenyl)methyl]-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
5-{2-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-oxoethyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-[(3S,5R)-5-[4-(pyrimidin-4-yl)piperidine-1-carbonyl]piperidine-3-carbonyl]morpholine
5-{[4-(5,6-dimethylpyrimidin-4-yl)piperazin-1-yl]methyl}-N,N-dimethylpyridin-2-amine
N-cyclohexyl-3-{[(dimethylcarbamoyl)(phenyl)methyl]amino}propanamide
1-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)urea
1-methyl-N-[1-(2-propoxyphenyl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
methyl 2-[3-(hydroxymethyl)-3-(2-phenylethyl)piperidine-1-carbonyl]benzoate
1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-2-(3-methoxyphenyl)piperidine
2-(adamantan-1-yl)-N-(1,4-dioxan-2-ylmethyl)-4-hydroxypyrimidine-5-carboxamide
5-methoxy-9-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}-1-oxa-9-azaspiro[5.5]undecane
4-{3-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)formamido]propyl}-1,2,5-oxadiazole-3-carboxylic acid
N-[2-(dimethylamino)-2-(3-methylphenyl)ethyl]-4-methyl-1H-imidazole-5-carboxamide
3-methyl-N-(2-{4-[(4-methyl-1H-imidazol-5-yl)methyl]morpholin-2-yl}ethyl)but-2-enamide
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-(oxolan-3-yl)benzamide
5-(propan-2-yl)-N-[1-(pyrimidin-4-yl)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
3-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}-N-(2-methylphenyl)-3-oxopropanamide
2-(2-hydroxyethyl)-6-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
methyl 3-[(2E)-3-(3-fluorophenyl)prop-2-enamido]-6-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)thieno[2,3-b]pyridine-2-carboxylate
[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl](2-methylpropyl)(pyridin-2-ylmethyl)amine
1-[1-(5-chloropyridin-2-yl)piperidin-4-yl]-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
N-[(3,4-difluorophenyl)methyl]-3-[1-(5-ethyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]propanamide
(3S,4R)-1-[(3-hydroxy-4-methoxyphenyl)methyl]-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid