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N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-[2-(methylsulfanyl)acetyl]pyrrolidine-2-carboxamide
1-[(3-chlorophenyl)methyl]-4-[2-(4-methyl-1,4-diazepane-1-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
9-{2-[(cyclopropylmethyl)sulfanyl]acetyl}-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-amino-4-(5-cyano-1,2-dimethyl-1H-pyrrol-3-yl)-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-6-oxo-1,6-dihydropyridazine-3-carboxamide
5-(1H-indol-1-ylmethyl)-N-[2-(4-methyl-1H-pyrazol-1-yl)propyl]-1H-pyrazole-3-carboxamide
1-{1-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]piperidin-3-yl}-4-(2-fluorophenyl)piperazine
1-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidin-1-yl]-2-(2H-1,2,3-benzotriazol-2-yl)ethan-1-one
4-[6-(morpholine-4-carbonyl)pyrazin-2-yl]-2-(trifluoromethyl)morpholine
4-[5-(1-phenoxypropan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl]morpholine
2-(4-fluorophenoxy)-N-(isoquinolin-5-ylmethyl)-N-methylacetamide
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}pyrazolo[1,5-a]pyridine-3-carboxamide
1-[2-(3-fluorophenoxy)acetyl]-3-(3-methoxypropyl)piperidine-3-carboxylic acid
1-methyl-N-[1-(thiophen-3-yl)propan-2-yl]-1H-indole-6-carboxamide
N-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-4-amine
4-(quinolin-8-yl)-1H-pyrazolo[3,4-d]pyrimidin-6-amine
(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-7-{[(3-methoxyphenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
1-[3-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)phenyl]ethan-1-one
N-[3-(1H-imidazol-1-yl)propyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
1-{2-[3-(2-fluorophenoxy)azetidin-1-yl]-2-oxoethyl}piperidin-2-one
1-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(pyrrolidin-1-yl)ethan-1-one
4-[2-(dimethylamino)-2-(3-methylphenyl)acetamido]butanoic acid
2-(4-carbamoylpiperidin-1-yl)-2-(4-chloro-3-fluorophenyl)acetic acid
1-(5-chloropyridin-2-yl)-4-(1H-pyrrole-2-carbonyl)piperazine
3-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}-1,4,6-trimethyl-1,2-dihydropyridin-2-one
8-chloro-2-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-3-ylmethyl]quinoline
(1S,5R)-6-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane
2-(1,4-dimethylpiperazin-2-yl)-N-{2-[2-(trifluoromethoxy)phenyl]ethyl}acetamide
4-(4-methylphenyl)-N-[2-(morpholin-4-yl)ethyl]-5-(pyridin-4-yl)pyrimidin-2-amine
N-cyclopentyl-2-[methyl({[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl})amino]propanamide
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
[(2-methoxyphenyl)methyl](pyridin-3-ylmethyl){[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
N-({1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-3-yl}methyl)acetamide
1-cyclohexanecarbonyl-N-[(3-methyl-1H-pyrazol-5-yl)methyl]pyrrolidine-2-carboxamide
N-(cyclopropylmethyl)-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-[(1S,5R)-3-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
N-[2-(furan-2-ylmethyl)-3-hydroxypropyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
2-(dimethylamino)-2-(2-fluorophenyl)-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]acetamide
(1S,6R)-9-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
2-[2-(methylsulfanyl)acetyl]-N-(1-phenylethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
(3R,4R)-4-amino-1-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}piperidin-3-ol
3-(azocan-1-yl)-N-{1-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]ethyl}propanamide
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-3-(1H-pyrazol-1-yl)benzamide
1-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)-2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]ethan-1-one
1-(1-ethyl-1H-pyrazole-4-carbonyl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
1-methyl-4-({5-[5-(propan-2-yl)-1,3-oxazol-4-yl]-1,2,4-oxadiazol-3-yl}methyl)piperidine
2-(5-acetylthiophen-3-yl)-N-[1-(thiophen-2-ylmethyl)piperidin-3-yl]acetamide
7-(3-phenylpropyl)-2-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
3-(1H-imidazol-2-yl)-1-[5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2-carbonyl]piperidine
2-methoxy-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide