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6-methyl-4-oxo-N-[1-(piperidine-1-carbonyl)piperidin-4-yl]-4H-pyran-2-carboxamide
1-(4-methyl-1H-imidazole-5-carbonyl)-4-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine
2,3,5,6-tetramethyl-N-[(1-methyl-1H-pyrazol-5-yl)methyl]benzamide
N-[4-(pyridin-3-yloxy)phenyl]-1-(1,3-thiazol-2-yl)piperidine-4-carboxamide
1-[1-(2-phenylethyl)piperidin-4-yl]-N-(1H-1,2,4-triazol-3-ylmethyl)piperidine-3-carboxamide
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
6-(benzyloxy)-1-(2-methylpropyl)-4-(1H-pyrazol-3-ylmethyl)-1,4-diazepan-2-one
N-(2-chloro-5-fluorophenyl)-2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}morpholine-4-carboxamide
3,3-dimethyl-2-[1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-1,2,3,4-tetrahydroisoquinoline
N4-[(3-methyl-1-benzofuran-2-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-1-[(4-methanesulfonylphenyl)methyl]piperidine
1-cyclopentyl-4-[3-(pyridin-2-yl)azetidine-1-carbonyl]pyrrolidin-2-one
2-[4-methyl-2,5-dioxo-4-(piperidin-4-yl)imidazolidin-1-yl]-N-[(2-methylphenyl)methyl]acetamide
3-(3-ethylphenoxy)-1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}azetidine
(3S,4S)-1-[1-(4-methanesulfonylphenyl)cyclobutanecarbonyl]-4-methylpiperidine-3,4-diol
N-[2-(4-methoxyphenyl)phenyl]-1-(pyridine-3-carbonyl)pyrrolidine-2-carboxamide
1-{4-[(3-methoxyphenyl)methyl]piperazin-1-yl}-3-(oxolan-2-yl)propan-1-one
8-(2-hydroxy-3-methylbenzoyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
(1R,3S)-7-(2-ethylpyridine-4-carbonyl)-3-methoxy-7-azaspiro[3.5]nonan-1-ol
[(3R,4R)-1-[(3,4-dimethoxyphenyl)methyl]-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
N3-[3-(dimethylamino)propyl]-N3-methyl-N5-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-benzyl-9-(1,2-dimethyl-1H-pyrrole-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
(1R,5S,6S)-6-[(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]-3-azabicyclo[3.1.0]hexane
5-[(1E)-1-(furan-2-yl)prop-1-en-2-yl]-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-7-one
7-(cyclopropylmethyl)-2-[(4-fluorophenyl)methanesulfonyl]-2,7-diazaspiro[4.5]decan-6-one
4-(2,4-dimethyl-1,4-diazepane-1-carbonyl)-6-fluoro-2-(1-methyl-1H-pyrazol-4-yl)quinoline
3-{1-[(5-chloro-2-hydroxyphenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)propanamide
6-({methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)pyridine-2-carboxylic acid
1-{1-[2-(1H-1,3-benzodiazol-1-yl)propanoyl]piperidin-4-yl}-N-(propan-2-yl)piperidine-4-carboxamide
ethyl 5-{[(2,4-dimethylpyrimidin-5-yl)formamido]methyl}furan-2-carboxylate
2-(4-benzyl-2-oxopyrrolidin-1-yl)-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]acetamide
2-(1,2-benzoxazol-3-yl)-N-{[1-(furan-2-ylmethyl)pyrrolidin-3-yl]methyl}acetamide
N-cyclopropyl-4-(2-oxopyrrolidin-1-yl)-N-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)benzamide
4-{7-[2-(dimethylamino)butanoyl]-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl}benzamide
N'-(3-chloro-4-fluorophenyl)-N-[1-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]butanediamide
N-({1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]piperidin-3-yl}methyl)-1H-indole-2-carboxamide
4-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(2-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]-1,2,3,6-tetrahydropyridin-4-yl}ethyl)-3,3-dimethylurea
1-[(4-fluorophenyl)methyl]-4-(oxolan-3-ylmethyl)-1,4-diazepane
1-methyl-3-({5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1,2-dihydropyridin-2-one
N-[1-(4-methanesulfonylphenyl)ethyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(morpholin-4-yl)ethan-1-one
5-methoxy-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-1H-indole-2-carboxamide
5-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]pyridin-2-amine
N-{[1-(1,4-dithiepan-6-yl)piperidin-3-yl]methyl}-3,5-dimethoxybenzamide
4-(1H-1,3-benzodiazol-1-yl)-1-(3-methylpyrazin-2-yl)piperidine-4-carboxylic acid
1-(2-methoxyethyl)-3-methyl-8-(quinolin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-N-methyl-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
(3E)-2-(4-hydroxy-4-phenylpiperidin-1-yl)hept-3-enoic acid
2-({3-benzyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}methyl)-4-(propan-2-yl)morpholine