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(1R,5S)-6-methyl-3-[(1-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-cyclopropyl-2-[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]-N-(1,3-thiazol-5-ylmethyl)acetamide
N-methyl-2-(5-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
1-[(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methylpyrrolidine-3-carbonyl]-4-(propan-2-yl)piperazine
N-{1-[(5-methylfuran-2-yl)methyl]-1H-pyrazol-5-yl}-2-[3-(pyridin-2-yl)-1H-pyrazol-1-yl]acetamide
3-(3-fluorophenyl)-N-(furan-2-ylmethyl)-N-propyl-1H-pyrazole-4-carboxamide
3,3,3-trifluoro-1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]propan-1-one
2-(dimethylamino)-2-(3-fluorophenyl)-N-[1-(methoxymethyl)cyclopentyl]acetamide
1-(6-aminopyridine-3-carbonyl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
4-[4-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)piperazin-1-yl]quinazoline
5-[4-(piperidin-4-yloxy)phenyl]furan-2-carboxamide
N-[2-(morpholin-4-yl)ethyl]-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(3S,4S)-1-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-4-(propan-2-yloxy)pyrrolidin-3-ol
N-[2-(ethylsulfanyl)ethyl]-3-(piperidin-3-yl)benzamide
(3R,4S)-4-{[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl](methyl)amino}oxolan-3-ol
4-chloro-2-methoxy-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]benzamide
5-(2,4-difluorophenoxymethyl)-N-[(3R)-4-hydroxy-3-methylbutyl]-1,2-oxazole-3-carboxamide
1-(1-benzoylpiperidin-3-yl)-3-(2-propylphenyl)urea
3-hydroxy-1-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}propan-1-one
3-({4-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-1-yl]phenyl}methyl)-5-methyl-4H-1,2,4-triazole
3-[2,2-bis(prop-2-en-1-yl)pyrrolidine-1-carbonyl]benzonitrile
N-[3-(3,4-diethoxyphenyl)propyl]-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
N-(4-{[methyl(2,2,6,6-tetramethylpiperidin-4-yl)amino]methyl}phenyl)acetamide
(3R,4S)-4-[({3-[(4-ethylpiperazin-1-yl)methyl]-2,5-dimethylphenyl}methyl)(methyl)amino]oxolan-3-ol
N-[2-(dimethyl-1,2-oxazol-4-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[(4-phenyl-1,3-thiazol-2-yl)methyl]-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
3-(2-amino-1,3-thiazol-4-yl)-N-[(4-sulfamoylphenyl)methyl]propanamide
1-(2-amino-6-methylpyrimidin-4-yl)-4-(2-fluorophenoxy)piperidine-4-carboxylic acid
2-(dimethylamino)-N-[2-(1-hydroxycyclopentyl)ethyl]-N-methyl-2-(4-methylphenyl)acetamide
4-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}thiomorpholine
7-(cyclopropylmethyl)-2-(1H-imidazol-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
4-chloro-N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-1H-pyrazole-3-carboxamide
4,5-dimethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]thiophene-2-carboxamide
N5-cyclooctyl-N3,N3-diethyl-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
N-{[5-(methylcarbamoyl)furan-2-yl]methyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
5-[3-methyl-5-(pyrrolidin-1-ylmethyl)phenyl]pyrimidine
[(3S,5R)-1-(3,6-dimethylpyrazin-2-yl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
5-methoxy-2-[4-(2-propoxyethyl)piperazine-1-carbonyl]-1,4-dihydropyridin-4-one
1-[9-(but-3-yn-1-yloxy)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-cyclopentylethan-1-one
2-hydroxy-2-(4-methoxyphenyl)-N-methyl-N-(quinolin-3-ylmethyl)acetamide
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(propan-2-yl)-2-(pyridin-3-yloxy)acetamide
1-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-methoxypiperidine
6-[1-(6-methylpyridazin-3-yl)piperidin-4-yl]-2-(6-methylpyridin-3-yl)-3,4-dihydropyrimidin-4-one
8-({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
(3aR,5S,6S,7aS)-2-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}-octahydro-1H-isoindole-5,6-diol
2,6-dimethoxy-N-{2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}pyridine-3-carboxamide
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(2-methoxypyridine-4-carbonyl)pyrrolidin-3-yl]methanol
(1S,8R)-4-amino-6-[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]-3-azatricyclo[6.2.1.02,7]undeca-2,4,6-triene-5-carbonitrile
3-{1-[(6-fluoroquinolin-2-yl)methyl]piperidin-4-yl}-1-(morpholin-4-yl)propan-1-one
3-(3-methyl-1H-pyrazol-1-yl)-1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one