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1-benzyl-N3-[(5-methylfuran-2-yl)methyl]-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
(4aR,7aS)-1-(2-methoxyacetyl)-4-[(2-methoxyphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S,4S)-4-cyclopropyl-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]pyrrolidine-3-carboxylic acid
6-(methylsulfanyl)-2-[3-(piperidin-3-yl)benzoyl]-1,2,3,4-tetrahydroisoquinoline
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-2-[4-(2-oxoimidazolidin-1-yl)phenyl]acetamide
[(5-cyclopropyl-1H-pyrazol-3-yl)methyl][(5-fluoro-3-methyl-1H-indol-2-yl)methyl]methylamine
ethyl 4-{1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}piperazine-1-carboxylate
2,3-dimethyl-7-{[4-(1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}-1H-indole
3-amino-1-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
3-({3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}sulfonyl)pyridine
6-chloro-4-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methylquinoline
(3S,4R)-1-(2-chloro-5-fluorobenzoyl)-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
4-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1,4-oxazepan-5-one
1-[(2E)-4-methylpent-2-enoyl]-4-(2-methylpropyl)-1,4-diazepan-5-one
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methoxyethyl)-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(2-fluorophenyl)methyl]-4-(5-{[(4-fluorophenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)piperidine
(1S,5R)-1,3,3-trimethyl-6-{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}-6-azabicyclo[3.2.1]octane
2-[(1-acetylpiperidin-4-yl)oxy]-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-5-methoxybenzamide
2-{[2-(1,3-thiazol-4-yl)ethyl]amino}pyridine-3-carboxamide
({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)[1-(thiophen-2-yl)ethyl]amine
7-(5-chloropyridin-2-yl)-4-cyclopentyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(1-{2-methylthieno[3,2-d]pyrimidin-4-yl}piperidine-3-carbonyl)pyridine
N-methyl-2-(oxan-2-ylmethoxy)-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]acetamide
N-methyl-5-[1-(2-phenoxyacetyl)pyrrolidin-2-yl]thiophene-2-carboxamide
3-[5-(2-methylpentyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-1-(pyrrolidin-1-yl)propan-1-one
3-(1H-imidazol-2-yl)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}benzamide
2-cyclopentyl-9-(4,6-dimethylpyrimidin-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]-2-(1,3-thiazol-2-yl)piperidine
2-[(3S,4R)-3-cyclopropyl-4-(dimethylamino)pyrrolidin-1-yl]-5-fluoro-N-methylpyrimidin-4-amine
1-cyclopentyl-4-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}piperazin-2-one
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
4-(1-cyclopropyl-5-oxopyrrolidine-3-carbonyl)-1-[(4-methoxyphenyl)methyl]piperazin-2-one
2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-3-(trifluoromethyl)pyridine
2-[2-(5-methyl-1H-indol-3-yl)phenyl]ethan-1-amine
N-({6-[2-(hydroxymethyl)phenyl]pyridin-3-yl}methyl)acetamide
1-(4-{[(3-cyclopentylpropyl)amino]methyl}-2-methoxyphenoxy)-3-(morpholin-4-yl)propan-2-ol
1-(2-methyl-1,3-thiazole-4-carbonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-benzyl-N-(1,1-dioxo-1λ6-thiolan-3-yl)-1,3-benzoxazole-5-carboxamide
methyl 2-[3-({[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amino}methyl)-1H-indol-1-yl]acetate
2-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-6-methylpyridine
N-ethyl-2,6-dimethyl-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}quinoline-4-carboxamide
4-benzyl-3-ethyl-1-[3-(pyrrolidin-1-yl)propanoyl]-1,4-diazepan-5-one
N3-benzyl-4-oxo-1-(propan-2-yl)-N5-[1-(thiophen-3-yl)propan-2-yl]-1,4-dihydropyridine-3,5-dicarboxamide
6-{[2-(2-oxoimidazolidin-1-yl)ethyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
5-(3-methylbutyl)-5-(piperidin-4-yl)-3-(pyridin-3-ylmethyl)imidazolidine-2,4-dione
2-{1-azabicyclo[3.2.1]octan-5-yloxy}-N-phenylbenzamide
6-amino-2-{2-[(5-ethyl-2-methylpyrimidin-4-yl)amino]ethyl}pyrimidin-4-ol
1-(propan-2-yl)-6-{[1-(pyridin-4-ylmethyl)-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1,2,3,4-tetrahydroquinoline
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
N,N-diethyl-4-[3-(hydroxymethyl)-4-methoxyphenyl]benzamide