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2-{4-[2-amino-3-cyano-6-(2,2-dimethylcyclopropyl)-5-methylpyridin-4-yl]phenoxy}acetamide
2-(2,3-difluorophenoxymethyl)-N-{[1-(dimethylamino)cyclohexyl]methyl}-1,3-oxazole-4-carboxamide
4-(6-methyl-2-propylpyrimidin-4-yl)-N-(pyridin-3-ylmethyl)piperazine-2-carboxamide
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]acetamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-4-amine
(2S,4S)-4-amino-1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-chloro-5-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
9-(6-methylpyridine-2-carbonyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-7-fluoro-N,2-dimethylquinoline-4-carboxamide
(3aR,6aS)-5-{[5-(2-propoxyethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
4-(1H-pyrazol-3-yl)-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}benzamide
2-methyl-N-[3-(2-phenylacetamido)phenyl]-3-(1H-pyrazol-1-yl)propanamide
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)pyrimidin-2-amine
1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}-3-[3-(2-oxopyrrolidin-1-yl)propyl]urea
1-[3,3-dimethyl-1-(pyridin-3-yl)butyl]-3-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}urea
2-[2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)acetyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
4-phenyl-1-{[3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]methyl}pyrrolidin-2-one
2-{1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]pyrrolidin-2-yl}pyridine
1-{4-[3-(2-hydroxyethyl)-4-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-1-yl]piperidin-1-yl}ethan-1-one
7-[(4-phenyl-1,3-thiazol-2-yl)methyl]-2-oxa-7-azaspiro[4.5]decan-8-one
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2,6-dimethylpyrimidine-4-carboxamide
5-(1H-imidazol-1-ylmethyl)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]pyridin-2-amine
2-(dimethylamino)-4-methyl-N-[(2-propyl-1,3-thiazol-4-yl)methyl]pyrimidine-5-carboxamide
3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-(pyridin-4-ylmethyl)propanamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N,6-dimethyl-4-oxo-4H-pyran-2-carboxamide
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(pyrazin-2-yl)ethan-1-one
8-(2-chloro-6-fluorobenzoyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-[2-hydroxy-4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
1-(cyclopropylmethyl)-5-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
6-[(diethylamino)methyl]-N-[(1R,2S)-2-phenylcyclopropyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
(2S,4S)-4-amino-1-[(2-chlorophenyl)methanesulfonyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-[(1-methylpiperidin-4-yl)oxy]-N-(oxolan-3-ylmethyl)aniline
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-(3-methylpyrazin-2-yl)piperidin-3-amine
2-[(2-methoxyethyl)sulfanyl]-4-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-3-yl)-5-(3-methoxyphenyl)pyrimidine
1-methyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-5-(3-fluorophenyl)-1,2,4-triazin-3-amine
2-{[4-(oxolan-3-yl)-1H-1,2,3-triazol-1-yl]methyl}-1H-indole
4-{[3-(oxan-4-yl)-1-phenyl-1H-1,2,4-triazol-5-yl]methyl}piperidine
5-tert-butyl-3-{[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1,2,4-oxadiazole
3-[1-(propane-1-sulfonyl)piperidin-3-yl]benzoic acid
4-[4-(dimethyl-1,3-oxazole-4-carbonyl)piperazin-1-yl]quinazoline
N-{1-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]piperidin-4-yl}methanesulfonamide
3-(1,2-oxazinan-2-yl)-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}propanamide
1-methanesulfonyl-4-(pyrrolidine-1-carbonyl)-1,4-diazepane-6-carboxylic acid
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-(trifluoromethyl)pyrimidin-4-amine
N-(2-methoxy-2-methylpropyl)-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
2-[7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-N-methyl-N-phenylacetamide
({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]amine
3-(3-phenyl-1,2,4-thiadiazol-5-yl)-1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)urea
1-(azepan-1-yl)-3-{4-chloro-2-[({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}amino)methyl]phenoxy}propan-2-ol