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methyl[(2E)-2-methylbut-2-en-1-yl]{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-(2-ethoxyethyl)-N-methyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}benzamide
2-(4-cyclobutyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-1-phenoxypropan-2-ol
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-{7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}acetamide
[(2S,4R)-4-(dimethylamino)-1-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]pyrrolidin-2-yl]methanol
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-{[4-(propan-2-yl)phenyl]methyl}piperidine
3-(2H-1,3-benzodioxol-5-yl)-N-methyl-N-(oxan-4-yl)-3-phenylpropanamide
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-1-[(2R,6S)-2,6-dimethylmorpholin-4-yl]propan-1-one
2-(methylamino)-1-{2-[2-(thiophen-2-yl)ethyl]piperidin-1-yl}ethan-1-one
6-fluoro-2-oxo-N-[2-(pyridin-2-ylsulfanyl)ethyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-ethyl-5-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-4-methyl-1,3-oxazole
3-[3-(3-hydroxypropyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]benzoic acid
N-(5-acetamido-2-fluorophenyl)-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-1-carboxamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-1-ethyl-1H-pyrazole-4-carboxamide
8-[(2-butoxy-3-methoxyphenyl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-1-ethyl-5-oxopyrrolidine-3-carboxamide
1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-N-(2,2,2-trifluoroethyl)piperidine-4-carboxamide
ethyl 3-(2-phenoxyethyl)-1-[2-(1H-pyrazol-1-yl)acetyl]piperidine-3-carboxylate
N-(2-methoxy-2-methylpropyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-[(3-{[(5-chloro-2-methoxyphenyl)methyl](methyl)carbamoyl}phenyl)amino]acetic acid
4-{5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl}-3-methylpyridine
5-(3-phenylpiperazine-1-carbonyl)-1H-pyrrole-3-carbonitrile
6,8-dimethyl-2-{[3-(1H-pyrazol-3-yl)piperidin-1-yl]methyl}quinolin-4-ol
(2E)-1-[4-(3-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxy)piperidin-1-yl]-3-(thiophen-2-yl)prop-2-en-1-one
5-[4-(4-fluorophenyl)-4-hydroxypiperidine-1-carbonyl]-1-(2-methoxyethyl)piperidin-2-one
2-(4-ethylpiperazin-1-yl)-N-(piperidin-4-ylmethyl)-2,3-dihydro-1H-indene-2-carboxamide
5-{[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1-(2-methoxyethyl)-1H-imidazole
1-{5-[({[1-(dimethylamino)cyclohexyl]methyl}amino)methyl]-2-methoxyphenoxy}-3-(4-methylpiperazin-1-yl)propan-2-ol
3-(1H-imidazol-2-yl)-N-[2-(1,3-thiazol-4-yl)ethyl]benzamide
5-{[benzyl(methyl)amino]methyl}-N-(2-methylbutan-2-yl)-1,2-oxazole-3-carboxamide
N-[(2-methylphenyl)methyl]quinoxaline-6-carboxamide
1-[(2R)-1-hydroxy-3-methylbutan-2-yl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylic acid
N-cyclopropyl-N-(2-methylpropyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
3-{2-oxo-2-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole
2-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}azetidin-3-yl)pyridine
7-({[1-(furan-2-yl)ethyl](methyl)amino}methyl)-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
N-{3-[(4-chlorophenyl)sulfanyl]propyl}-2-(2-oxopiperidin-1-yl)acetamide
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-5-propyl-1,3,4-oxadiazol-2-amine
N,N-dimethyl-4-(4-methyl-3,4-dihydro-2H-1,4-benzoxazine-2-carbonyl)piperazine-1-sulfonamide
methyl 6-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]pyrimidine-4-carboxylate
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-3-(1,2-oxazolidin-2-yl)propanamide
3-({[1-(5-chlorothiophene-2-carbonyl)piperidin-3-yl]oxy}methyl)pyridine
1-methyl-3-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}-6-(propan-2-yl)-1,2-dihydropyridin-2-one
6-[(3R,4S)-3-amino-4-phenylpyrrolidine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
6-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]pyridin-2-amine
2-(4-fluoro-2-methoxyphenyl)pyridine-4-carbonitrile
5-ethyl-2-{4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazin-1-yl}pyrimidine
N-benzyl-2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide