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4-methoxy-N-(2-{7-[3-(5-methylfuran-2-yl)butyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
4-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}butanamide
3-{5-[(6-chloropyridin-3-yl)carbamoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
1-[(3-fluorophenyl)methyl]-4-[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazin-2-one
4-{4-[1-(1-methoxybutan-2-yl)-4-phenyl-1H-imidazol-5-yl]phenyl}but-3-yn-1-ol
4-(5-hydroxy-1,2-dimethyl-1H-indole-3-carbonyl)-1-methylpiperazine-2-carboxylic acid
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-[2-(phenylsulfanyl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
9-[(3-fluoro-5-methylphenyl)methyl]-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-ethyl-3-(1H-indol-3-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(dimethyl-1,2-oxazol-4-yl)-4-{[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carboxamide
ethyl 4-[(3-fluorophenyl)methyl]-1-methylpiperidine-4-carboxylate
3-chloro-4-[(1-cyclohexylpiperidin-4-yl)oxy]-N-(2-methoxyethyl)benzamide
5-{[2-(2-aminoethyl)morpholin-4-yl]methyl}-N-ethylpyrimidin-2-amine
(4-{[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)pyrrolidin-3-yl]methyl}phenyl)methanol
3-cyclohexyl-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-1H-pyrazole-4-carboxamide
N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-(piperidin-1-ylmethyl)benzamide
2-{[1-(2-fluoro-4-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,3-thiazole
4-methyl-5-[1-(thiophen-3-ylmethyl)-1H-pyrazol-3-yl]-N-[(2,3,4-trimethoxyphenyl)methyl]-1,3-thiazol-2-amine
N-[1-(cyclohexylmethyl)piperidin-3-yl]-3-methoxypropanamide
1-{2-[3-(1H-1,3-benzodiazol-2-yl)azetidin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
7-[(2,3-difluorophenyl)methyl]-2-(4-methyl-1,3-thiazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}ethane-1-sulfonamide
2-[2-(1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperidin-4-yl)-1H-imidazol-1-yl]acetamide
N-(2-ethyl-3-methyl-1-benzofuran-7-yl)-2-(1,3-thiazol-2-yl)pyrrolidine-1-carboxamide
4-(2-phenoxyethyl)-1-{2-[3-(trifluoromethyl)phenyl]acetyl}-1,4-diazepan-5-one
N-({1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)-3-methylbut-2-enamide
4-(4-{4-[2-(oxolan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine-1-carbonyl}phenyl)morpholine
4-methyl-6-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-carbonyl]-1,3-benzothiazol-2-amine
7-(1,3-benzothiazol-2-yl)-4-[1-(2-methoxyphenyl)propan-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
ethyl 1-[1-(pyridin-2-yl)propan-2-yl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
1-(1-ethyl-5-{[2-(furan-2-yl)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl)pyrrolidine
N-(1H-indol-3-yl)quinoline-3-carboxamide
N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
4-(4-{2-[2-(4-methoxyphenyl)ethyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)-N,N-dimethyl-4-oxobutanamide
3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]quinolin-7-ol
4-methyl-5-{4-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidine-1-carbonyl}-1,3-thiazol-2-amine
{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}(4-phenylbutan-2-yl)amine
[1-(1H-pyrazol-1-yl)propan-2-yl](4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)amine
N-methyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
4-({[(5-ethylpyridin-2-yl)methyl](methyl)amino}methyl)-2-fluoro-6-methoxyphenol
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-2-(methylamino)acetamide
1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(2-fluorophenyl)piperazine
(1,3-benzoxazol-2-ylmethyl)({[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl})methylamine
1-(furan-3-ylmethyl)-3-(pyrrolidin-1-yl)piperidine
N-[(3R,4S)-1-(cyclobutylmethyl)-4-propylpyrrolidin-3-yl]-3-(2-oxopyrrolidin-1-yl)propanamide
1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-4-(3-methylpyridin-4-yl)-1,4-diazepane
7-(3-chlorophenyl)-4-(5,6-dimethylpyrimidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-methyl-4-phenyl-5-(2-propyl-2,5-dihydro-1H-pyrrole-1-carbonyl)pyrimidine
4-[3-(2-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,2,3-thiadiazole
1-[3-(1H-imidazol-2-yl)benzoyl]-4-(2-phenoxyethyl)piperazine