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4-({2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}methyl)piperazin-2-one
1-(2-{4-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethyl)piperazine
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-1-(propan-2-yl)piperidine-4-carboxamide
{[5-(cyclohexylsulfanyl)furan-2-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
N-{[8-(3-methylbut-2-en-1-yl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-1H-1,2,3-triazole-5-carboxamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-{thieno[3,2-d]pyrimidin-4-yl}pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
5-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]quinoxaline
6-(3-chlorophenyl)-N,N-dimethyl-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-2-(3,4-dichlorophenyl)morpholine
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-1-methyl-1H-indole-2-carboxamide
N-[2-(dimethylsulfamoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]oxolane-2-carboxamide
4-[(5-{1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}-1,2,4-oxadiazol-3-yl)methyl]-1-methylpiperidine
(3S,4R)-1-[(8-methoxyquinolin-2-yl)methyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(propan-2-yl)acetamide
2-({2-[2-(2-methoxyethyl)-2H-1,2,3,4-tetrazol-5-yl]morpholin-4-yl}methyl)-6-methylquinolin-4-ol
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-3-(1H-imidazol-1-yl)butan-1-one
3-acetamido-N-methyl-N-(oxan-2-ylmethyl)benzamide
(1R,5R)-3-[1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carbonyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonane
N-[2-(ethanesulfonyl)ethyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
3-(hydroxymethyl)-1-[3-(hydroxymethyl)-8-methylquinolin-2-yl]piperidin-3-ol
5-fluoro-N-methyl-4-(morpholin-4-yl)-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}pyrimidin-2-amine
1-ethyl-6-oxo-N-[2-(1H-pyrrol-1-yl)ethyl]piperidine-3-carboxamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2-(3-methyl-1H-pyrazol-1-yl)acetamide
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
5-(hydroxymethyl)-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}furan-2-carboxamide
1-(4-{4-[(2-fluorophenyl)methyl]piperidine-1-carbonyl}-3,5-dimethyl-1H-pyrrol-2-yl)ethan-1-one
N-[(3S,4R)-4-hydroxyoxolan-3-yl]-6-(4-methoxyphenyl)-N-methyl-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-[1-(2,6-dimethoxypyridin-3-yl)-1H-imidazol-2-yl]-1,2-dihydroquinolin-2-one
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[2-(methylsulfanyl)ethyl]acetamide
1-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}pent-4-en-1-one
1-(2-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-2-oxoethyl)pyrrolidin-2-one
10-(1,3-thiazolidine-3-carbonyl)-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraen-9-one
3-{1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]piperidin-3-yl}-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,4R)-1-[3-(3-fluorophenyl)benzoyl]-4-methylpiperidine-3,4-diol
2-amino-7-(2,6-difluoro-3-methylbenzoyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-methyl-6-{5-[5-(propan-2-yl)-1,2-oxazol-3-yl]-1,2,4-oxadiazol-3-yl}pyridazine
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl)(1,3-thiazol-2-ylmethyl)amine
2-[4-(dimethylsulfamoyl)morpholin-3-yl]-N-[2-(5-methylthiophen-2-yl)ethyl]acetamide
2-[(1-ethylpyrrolidin-2-yl)methyl]-5-(1,2,3,4-tetrahydroisoquinolin-2-yl)-2,3-dihydropyridazin-3-one
2-{4-[(2,3-difluorophenyl)methyl]-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
6-(3,3-diphenylpiperidine-1-carbonyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-({1-[1-(6-ethoxy-4-methylquinazolin-2-yl)pyrrolidine-2-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
N-(2-chloro-4,6-dimethylphenyl)-3-(methanesulfonylmethyl)piperidine-1-carboxamide
[2-(2,4-dimethoxyphenyl)phenyl]methanamine
9-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(3,5-dimethoxyphenyl)-3-[1-(3-methylbut-2-en-1-yl)piperidin-3-yl]propanamide
N-(3-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}-3-oxopropyl)acetamide
N-[(2S,4R,6S)-2-(2-methylpropyl)-6-(pyridin-3-yl)oxan-4-yl]benzamide
N-[(2-amino-1,3-thiazol-4-yl)methyl]-1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide