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1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(1H-imidazol-2-ylmethyl)-N-methylpiperidine-3-carboxamide
2-[2-(1-methyl-1H-pyrazol-4-yl)phenoxy]propanamide
1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-[4-(methylsulfanyl)phenyl]ethan-1-one
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
3-({4-[(8-fluoro-4-hydroxyquinolin-2-yl)methyl]piperazin-1-yl}methyl)benzonitrile
2-[4-(6-chloroquinolin-4-yl)-1-cyclopentylpiperazin-2-yl]ethan-1-ol
2-{1-[(6-methylpyridin-2-yl)methyl]-4-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperazin-2-yl}ethan-1-ol
3-(1H-1,2,3-benzotriazol-1-yl)-1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]propan-1-one
2-(4-methylpyridine-3-carbonyl)-N-(oxolan-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
1-({4-methyl-5-[1-(pent-2-yn-1-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-4-amine
2-[1-(hydroxymethyl)-9-(3-methoxypropanoyl)-3,9-diazaspiro[5.5]undecan-3-yl]acetamide
5-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
8-[2-chloro-5-(1H-pyrazol-1-yl)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
4-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
3-{2-azaspiro[4.4]nonan-2-ylmethyl}-7-methyl-1,2-dihydroquinolin-2-one
2-(3-{4-[(3Z)-hex-3-en-1-yl]-1H-1,2,3-triazol-1-yl}piperidin-1-yl)pyrimidine
4-chloro-N-[3-(1H-imidazol-1-yl)propyl]-1-methyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-3-carboxamide
N-(2-hydroxyethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]-2-(1H-pyrazol-1-yl)butanamide
N-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-N-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2-(1H-1,2,4-triazol-3-yl)benzamide
3-(2-hydroxyphenyl)-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1H-pyrazole-5-carboxamide
1-(3-{2-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl]phenoxy}propyl)-1H-imidazole
N-[(3R,4S)-4-cyclopropyl-1-(oxan-4-yl)pyrrolidin-3-yl]-4-(1H-pyrazol-1-yl)butanamide
4-[4-(2-methyloxane-2-carbonyl)piperazin-1-yl]quinazoline
5-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2,4-dimethylpyrimidine
(3aS,6aS)-2-{[4-(methylcarbamoyl)phenyl]methyl}-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(1-ethyl-1H-imidazol-2-yl)-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidine
5-(1-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-3-[(4-fluorophenyl)methyl]-5-methylimidazolidine-2,4-dione
(4aR,7aS)-1-propyl-4-[2-(pyridin-3-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl 4-[3-methyl-1-(2-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]benzoate
(1-{[1-(3-cyclopentylpropyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
N-[(1-cyclopropanecarbonylpiperidin-4-yl)methyl]-6-methylpyridine-3-carboxamide
2-(methylsulfanyl)-5-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)pyrimidine
3-(5-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
(4aS,7aR)-1-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-3-propylpiperidine-3-carboxylic acid
2-[1-(2,2-dimethylpropyl)-4-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperazin-2-yl]ethan-1-ol
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(oxolan-2-ylmethyl)acetamide
4-cyclopentyl-3-(4-hydroxy-3-methoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{2-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]phenyl}morpholine
1-(pyridin-2-ylmethyl)-4-{1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}pyrrolidin-2-one
(1R,7S)-N-benzyl-3-(4-fluoro-2-methylphenyl)-N-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
4-ethyl-3-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-ethyl-4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidine-1-carboxamide
2-(2,6-dimethoxy-4-methylphenyl)-N-methylpyridine-4-carboxamide
8-chloro-2-[({[1-(2-hydroxyethyl)piperidin-4-yl]methyl}(methyl)amino)methyl]quinolin-4-ol
(3aS,6aS)-2-(ethanesulfonyl)-5-[2-(3-fluorophenyl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(9H-carbazol-3-yl)-1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-3-(3-hydroxyquinoxalin-2-yl)propanamide