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2-[2-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)-2-oxoethyl]-2,7-diazaspiro[4.5]decan-6-one
4-[({3-azaspiro[5.5]undecan-9-yl}amino)methyl]benzene-1-sulfonamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-4-methoxy-3-(morpholin-4-yl)benzamide
1-[4-(2-methoxyphenoxy)piperidin-1-yl]-2-(pyrrolidin-1-yl)propan-1-one
methyl (2R,4S)-4-hydroxy-1-{[3-(hydroxymethyl)-4-(propan-2-yloxy)phenyl]methyl}piperidine-2-carboxylate
2-{2-[bis(propan-2-yl)carbamoyl]phenyl}-N-ethylpyridine-4-carboxamide
6-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidine-2,4-diamine
6-methyl-2-[1-(oxan-4-ylmethyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
5-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-2,3-dihydro-1H-pyrazol-3-one
N-(butan-2-yl)-6-(2,5-dimethylfuran-3-yl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-(4-acetyl-6-hydroxy-1,4-diazepan-1-yl)-3-(2-methoxyphenyl)propan-1-one
2-(2-{1-[(4-methylthiophen-2-yl)sulfonyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-1,9-dioxaspiro[5.5]undecan-4-amine
6-[3-methyl-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N,2-dimethyl-1H-pyrrole-3-carboxamide
N-methyl-4-[6-(trifluoromethyl)pyridin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
(4aR,8aS)-1-(cyclohexylmethyl)-6-[(2-hydroxyphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
(2-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}-2-oxoethyl)urea
(4aS,8aR)-1-(2-aminoethyl)-6-[2-(thiophen-3-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
4-(1-{[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3-carbonyl)morpholine
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-3-ethyl-N,5-dimethyl-1,2-oxazole-4-carboxamide
(2-{2-[1-(4,6-dimethylquinolin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
2-{4-[(2,3-dimethoxyphenyl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-2-(3-fluoro-4-hydroxyphenyl)ethan-1-one
[(1-benzyl-1H-imidazol-2-yl)methyl](methyl){[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amine
2-{1-[1-(4-methyl-1H-imidazole-2-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}pyridine
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
N-methyl-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[1-(pyrimidin-4-yl)ethyl]acetamide
2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-1-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]ethan-1-one
6-(thiophen-2-yl)pyridine-3-carboxamide
2-(2-chloro-6-fluoro-3-methylphenyl)-1-[2-(propane-2-sulfonyl)ethyl]-1H-imidazole
2-{[(1S,2S)-2-[(4-fluorophenyl)methyl]cyclopentyl]amino}propane-1,3-diol
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]ethan-1-one
methyl 9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-3-[(6-methylpyridin-2-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-hydroxy-N-({1-[(5-methylnaphthalen-1-yl)methyl]pyrrolidin-3-yl}methyl)acetamide
(3aS,7aR)-5-methyl-2-(2,6,8-trimethylquinoline-4-carbonyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
1-cyclohexyl-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
N-[2-(ethylsulfanyl)ethyl]-1,5-dimethyl-1H-indole-2-carboxamide
[(3R,4R)-1-[1-(4-chlorophenyl)piperidin-4-yl]-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
3-amino-1-[(3-fluoropyridin-4-yl)methyl]pyrrolidine-3-carboxylic acid
1-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
1-[(3,5-dimethylphenyl)methyl]-4-(1-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)piperazin-2-one
1-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}-2-hydroxyethan-1-one
1-[5-(methoxymethyl)furan-2-carbonyl]-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
methyl 1-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidine-2-carboxylate
3-(quinolin-6-ylmethyl)-3H,4H-thieno[3,2-d]pyrimidin-4-one
9-methoxy-7-(4-methoxyphenyl)-4-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[2-(dimethylsulfamoyl)ethyl]-1-(propan-2-yl)-1H-pyrazole-3-carboxamide
({4-[1-(2-methoxypyridine-4-carbonyl)piperidin-2-yl]phenyl}methyl)dimethylamine
2-{[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}benzonitrile