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(3R,5S)-N3-methyl-N5-(6-methylpyridin-3-yl)-N3-(1,3-thiazol-2-ylmethyl)piperidine-3,5-dicarboxamide
(2S,4S)-1-[(4-chlorophenyl)methyl]-4-({[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}amino)-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
3-(4-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propanamide
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2,8-dimethylquinoline-4-carboxamide
N-(3,4-dimethylphenyl)-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
4-methoxy-6-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-2-amine
{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}({2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl})amine
1-({1-[(3,4-dimethylphenyl)methyl]piperidin-3-yl}methyl)-3-(propan-2-yl)urea
[(2S,4R)-4-(dimethylamino)-1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-2-yl]methanol
(4aR,8aR)-2-(5-chloro-6-hydroxy-2-methylpyrimidin-4-yl)-7-cyclopentanecarbonyl-decahydro-2,7-naphthyridin-4a-ol
2-(2-chloro-6-methoxy-4-{[methyl(pyrazin-2-ylmethyl)amino]methyl}phenoxy)acetamide
2-{1-[(2-methylphenyl)methyl]-4-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
N-[1-(1H-imidazol-1-yl)-3-methylbutan-2-yl]-3-propyl-1H-pyrazole-5-carboxamide
4-[({[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)methyl]-2-ethoxyphenol
methyl 4-{4-[(4R)-3-methyl-1,3-thiazolidine-4-carbonyl]piperazin-1-yl}benzoate
N-{[5-(3,6-dimethylpyrazin-2-yl)-7-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methylpiperidine-2-carboxamide
5-methoxy-2-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]phenol
N-methyl-4-({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)butanamide
3-[(5-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-3,4-dihydroquinazolin-4-one
11-{[(2,6-difluoro-3-methylphenyl)methyl]amino}-4-[(1-methyl-1H-pyrazol-4-yl)methyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-methyl-4-({5-[3-(1H-pyrazol-4-yl)phenyl]-1,2,4-oxadiazol-3-yl}methyl)piperidine
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-N'-cyclopentyl-N-methylbutanediamide
3-(3-chloro-1H-1,2,4-triazol-5-yl)-N-[(1S,2R)-2-[(2,3-dihydro-1H-inden-2-yl)amino]cyclobutyl]propanamide
(3aS,7aR)-2-[3-(dimethylamino)benzoyl]-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
2-chloro-4-({1-ethyl-3-[hydroxy(phenyl)methyl]-1H-1,2,4-triazol-5-yl}methyl)phenol
N-methyl-N-{2-[4-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenoxy]ethyl}pyridine-4-carboxamide
3-(3-chlorophenyl)-1-[4-(2-methoxyethyl)piperazin-1-yl]-3-phenylpropan-1-one
1-[3-(2-methylphenyl)phenyl]-N-(thiolan-3-yl)piperidin-4-amine
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N,N-bis(1,3-oxazol-4-ylmethyl)acetamide
6-phenyl-3-[2-(pyridin-3-yl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-phenyl-4-{1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}piperazine
6-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)pyrimidine-2,4-diamine
3-acetyl-N-[(4-fluorophenyl)methyl]-N-(pyridin-4-ylmethyl)-1H-pyrazole-5-carboxamide
4-{3-cyclopropyl-5-[3-(1H-1,2,3,4-tetrazol-1-yl)phenoxymethyl]-1H-1,2,4-triazol-1-yl}-3-methylpyridine
[(2,3-difluoro-6-methoxyphenyl)methyl](1,4-dioxan-2-ylmethyl)methylamine
1-[(1-hydroxycyclohexyl)methyl]-5-oxopyrrolidine-3-carboxylic acid
1-{[3-(difluoromethoxy)phenyl]methyl}-4-[1-(pyrrolidin-1-yl)ethyl]piperidine
3-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-5-propyl-1,2,4-oxadiazole
3-{[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]amino}-N-(thiophen-2-ylmethyl)propanamide
(1S,5R)-6-[(2,4-dimethoxyphenyl)methyl]-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-ethyl-N-[2-(1H-indol-3-yl)ethyl]-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(4-{[(1S,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}thiophen-2-yl)ethan-1-one
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
[(3R,4R)-1-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
3-{methyl[2-(pyridin-2-yl)ethyl]amino}-N-(2-phenylethyl)piperidine-1-carboxamide
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-N-methyl-N-(pyridin-3-ylmethyl)piperidin-4-amine
2-{2-[2-(benzyloxy)ethyl]phenyl}-5-methyl-1,3,4-oxadiazole
6-[2-(5-ethyl-1,2,4-oxadiazol-3-yl)ethyl]-2-methoxy-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-1-[3-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidine
(4aS,7aR)-1-[(3-hydroxyphenyl)methyl]-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione