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N-[(4-ethoxyphenyl)methyl]-N-{[3-(3-methoxyphenyl)oxolan-3-yl]methyl}cyclopropanamine
7-(furan-2-carbonyl)-N-(pyrimidin-4-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-({[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}(methyl)amino)-1λ6-thiolane-1,1-dione
N-(4-ethyl-1,3-dimethyl-1H-pyrazol-5-yl)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-carboxamide
1-(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)butan-1-one
2-[(2R,3R)-3-(dimethylamino)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]pyridine-4-carboxamide
(3aR,6aR)-2-cyclopentyl-5-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[2-(pyrrolidin-1-yl)ethyl]-1H-pyrazole-3-carboxamide
N-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]pyrimidin-2-amine
1-methyl-4-({4-[3-(3-methylpiperidin-1-yl)propoxy]phenyl}methyl)piperazine
3-{[(3,3-diphenylpropyl)amino]methyl}-7-fluoro-1-methyl-1,2-dihydroquinolin-2-one
methyl (2S)-2-{[5-(azepane-1-carbonyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridin-3-yl]formamido}-3-methylbutanoate
2-hydroxy-3-methoxy-N-[(3S,4S)-4-methoxy-1,1-dioxo-1λ6-thiolan-3-yl]benzamide
5-butyl-4-[2-(1H-imidazol-1-yl)acetyl]-1-(3-methylphenyl)piperazin-2-one
1-(propan-2-yl)-N-[1-(pyridin-4-yl)propyl]-1H-pyrazole-4-carboxamide
N-(3-chloro-2-methylphenyl)-N'-({2-[(dimethylamino)methyl]phenyl}methyl)-N'-methylpropanediamide
2-(dimethylamino)-2-(3-methylphenyl)-1-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]ethan-1-one
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
N-methyl-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}-N-(thiophen-2-ylmethyl)benzamide
N-({1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)-3-methyl-1H-pyrazole-5-carboxamide
4-(2-fluoro-5-methoxyphenyl)pyridin-2-amine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
1-(1-methyl-1H-pyrazole-3-carbonyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-methoxyethan-1-one
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({[2-(1,3-thiazol-2-yl)ethyl]amino}methyl)piperidin-2-one
{5-[2-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]-2,3-dihydro-1-benzofuran-2-yl}methanamine
4-(3-chlorophenyl)-3-(3-cyclopropyl-1H-pyrazol-5-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-cyclopropyl-1-[2-(4-methoxyphenyl)ethyl]-5-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
7-(2-methoxyphenyl)-2-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-[3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-6-(propan-2-yl)pyridazine
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-4-oxo-4H-chromene-2-carboxamide
2,3-dimethyl-6-[1-(propan-2-yl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]quinoxaline
N,3-dimethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1H-pyrazole-5-carboxamide
9-(4-hydroxy-3-methylbenzoyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-3-(piperidin-3-yl)benzamide
methyl({[1-(3-methylbutyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl})(pyrazin-2-ylmethyl)amine
1-[2-(1H-indol-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]piperidine-3-carboxamide
1-ethoxy-3-[5-(2-methoxy-4-methylphenyl)-4-phenyl-1H-imidazol-1-yl]propan-2-ol
7-(2-methylphenyl)-4-(pyrimidine-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
(4-benzyl-1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-4-yl)methanol
(2S)-2-{[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino}-2-phenylethan-1-ol
(2S,4S)-4-amino-1-[2-(methylsulfanyl)pyrimidine-5-carbonyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-({methyl[1-(pyrimidin-4-yl)ethyl]amino}methyl)-N-(1,2,3-thiadiazol-5-yl)benzamide
N-[(3S)-1-[4-(4-ethoxy-3-methylphenyl)butanoyl]pyrrolidin-3-yl]acetamide
(2S,4R)-N-[2-(4-fluorophenyl)ethyl]-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
2-[(3-methoxyphenyl)methyl]-8-(pyridine-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide