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2-(2-{[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]methyl}phenoxy)acetic acid
3-(3-chlorophenyl)-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3-phenylpropanamide
2-{5-[(5-ethylpyridin-2-yl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
N-(2,3-dihydro-1H-inden-2-yl)-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N'1-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N'1-methylcyclopropane-1,1-dicarboxamide
N2-ethyl-N2-[2-(piperidin-1-yl)ethyl]pyrrolidine-1,2-dicarboxamide
N-[4-(methylamino)butyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-butyl-2-[(dimethylcarbamoyl)amino]-N-[(2-methylphenyl)methyl]acetamide
1-[4-({3-[3-(diethylamino)pyrrolidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)-3-methoxyphenyl]ethan-1-one
3-{2-[(2-butyl-6-methylpyrimidin-4-yl)amino]ethyl}-1-(4-cyano-2-fluorophenyl)urea
N-methyl-5-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-ylmethyl}furan-2-carboxamide
2-methyl-5-(2-{1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)-1,3,4-oxadiazole
4-phenyl-1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}azepane
N-(prop-2-en-1-yl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-{4-[(3-ethoxy-4-methoxyphenyl)methyl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-({1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}methyl)naphthalene-1-carboxamide
2-{5-[1-(2-phenylacetyl)piperidin-2-yl]-1,2,3,6-tetrahydropyridin-1-yl}acetamide
1-{5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-1,4-diazepane
4-{1-[2-(morpholin-4-yl)acetyl]piperidin-3-yl}benzoic acid
N-[(2R,3R)-2-(pyridin-4-ylmethoxy)-1'-(thiophene-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
4-(3,5-difluorobenzoyl)-1-[(3,5-dimethylphenyl)methyl]piperazin-2-one
5-{2-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-1H-imidazol-1-yl}-4,5,6,7-tetrahydro-1H-indazole
4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
(3R,4R)-3-methyl-1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-4-(oxan-4-yl)piperidin-4-ol
1-[2-(1-{2-[4-(dimethylamino)phenyl]acetyl}piperidin-4-yl)ethyl]pyrrolidin-2-one
N,N,4-trimethyl-5-(3-phenylpiperazine-1-carbonyl)pyrimidin-2-amine
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-hydroxypropanamide
5-methyl-N2-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}pyrimidine-2,4-diamine
3-[1-(adamantan-2-yl)piperidin-3-yl]-N-[(3,4-difluorophenyl)methyl]propanamide
2-(3-cyano-2-methyl-1H-indol-1-yl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}acetamide
1-[3-(azepan-1-yl)propanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-({[(1R,2S)-2-hydroxycyclohexyl](methyl)amino}methyl)-1H-pyrazole-3-carboxylic acid
2-(2-hydroxypropyl)-9-[2-(4-methyl-1H-pyrazol-1-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[(4-fluorophenyl)methyl]-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-(3-methylbut-2-en-1-yl)-1-(2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carbonyl)piperidine-3-carboxylic acid
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]methanesulfonamide
2-methoxy-4-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carbonitrile
7-(3,6-dimethylpyrazin-2-yl)-4-(6-ethylpyrimidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(3S,4R)-3-benzyl-1-{6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}-4-methylpiperidin-4-ol
(4aR,7aS)-1-(2-methoxyacetyl)-4-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(6-hydroxypyrimidin-4-yl)methyl]-N'-(2-methylphenyl)propanediamide
1-(2,3-dihydro-1H-indene-5-carbonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
8-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[(3-methoxyphenyl)amino]-N-methyl-N-[2-(pyridin-2-yl)ethyl]butanamide
N,N-dimethyl-3-{[(4-methyl-1H-imidazol-5-yl)methyl]amino}-5-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)benzene-1-sulfonamide
2-(dimethylamino)-2-(4-fluorophenyl)-N-(1H-indol-6-ylmethyl)acetamide
3,5-dimethoxy-N-{[1-(1,2,3-thiadiazole-4-carbonyl)piperidin-3-yl]methyl}benzamide
2-[4-(6-chloro-2-methylquinoline-4-carbonyl)morpholin-3-yl]acetic acid
2-(dimethylamino)-N-[1-(hydroxymethyl)cyclopentyl]-2-(3-methylphenyl)acetamide
1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane