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5-[7-(3-methoxyphenyl)-4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl]-N-methyl-1,2,4-oxadiazole-3-carboxamide
(3R)-1-{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-ol
4-(3-chlorophenyl)-N-(5-phenyl-1H-1,2,4-triazol-3-yl)piperazine-1-carboxamide
4-(1,3-benzothiazol-2-yl)-N-(pyridin-2-ylmethyl)piperazine-2-carboxamide
5-fluoro-2-[1-(3-methylfuran-2-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
N-[(1S)-1-[1-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,4-triazol-5-yl]-3-(methylsulfanyl)propyl]acetamide
1-{2-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-oxoethyl}-5,5-dimethylimidazolidine-2,4-dione
N-{[1-(2,2-dimethylpropyl)pyrrolidin-3-yl]methyl}-1-methyl-1H-indole-3-carboxamide
N4-(2,1,3-benzoxadiazol-5-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
1-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-3-(pyridin-3-yl)propan-1-one
1-(2,3-dihydro-1,4-benzodioxine-5-carbonyl)-4-[(3-fluorophenyl)methyl]piperazine
2-(3-acetyl-1H-indol-1-yl)-N-[3-(1H-imidazol-1-yl)propyl]butanamide
5-chloro-N-(3-hydroxypropyl)-N-[(5-methylthiophen-2-yl)methyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
2-{4-[(3,4-difluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}-1,3-thiazole-4-carboxamide
3-{[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl](methyl)amino}-N-methylbutanamide
1-(4-methoxyphenyl)-4-[2-(4-methyl-1,4-diazepan-1-yl)acetyl]piperazin-2-one
3-ethyl-5-{1-[(4-phenyl-1,3-thiazol-5-yl)methyl]-1H-imidazol-2-yl}-1,2-oxazole
[3-(2-methoxyethyl)-1-[2-(pyrrolidin-1-yl)benzoyl]piperidin-3-yl]methanol
2-{methyl[2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}ethan-1-ol
N-(2,5-dihydroxy-2-methylpentyl)-2-(1H-imidazol-2-yl)benzamide
5-(8-chloroquinolin-2-yl)pyridin-3-amine
(2S)-1-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxamide
2-({3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}methyl)-5-methoxy-4H-pyran-4-one
3-[(3R,4S)-1-[2-(4-hydroxyphenyl)acetyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
1-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-4,4,4-trifluorobutan-1-one
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-1-(4-methylphenyl)cyclopropane-1-carboxamide
2-({[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(thiophen-2-ylmethyl)amino)ethan-1-ol
N,8-dimethyl-N-(propan-2-yl)-2-[2-(propan-2-yl)pyrimidin-5-yl]quinoline-4-carboxamide
N,N-dimethyl-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxamide
(1S,6R)-9-(2,1,3-benzothiadiazol-4-ylmethyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
(4aR,7aS)-1-(2-methoxyethyl)-4-[3-(pyridin-2-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1S,5R)-3-(2-methyl-5-propylpyrimidin-4-yl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(2R,3R)-3-[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
(1R,5S)-3-[(5-chlorofuran-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(1H-indol-4-ylmethyl)-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
8-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-1-methyl-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[2-(4-fluorophenyl)ethyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(4-methyl-1H-imidazol-5-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-(1-benzylpyrrolidin-3-yl)-5-fluoro-4-(morpholin-4-yl)pyrimidin-2-amine
5-[(2-fluoro-4-methoxyphenyl)methyl]-5-{3-[2-(hydroxymethyl)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-fluoro-5-sulfamoylbenzamide
{3-[4-(morpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]propyl}({[2-(prop-2-en-1-yloxy)phenyl]methyl})amine
(1-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methanol
N-[(1R,2S)-2-phenylcyclohexyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-1-cyclopropyl-N-methyl-5-oxopyrrolidine-3-carboxamide
2-ethoxy-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
4-({5-[1-(5-fluoropyrimidin-2-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
4-{3-[(4-fluorophenyl)methoxy]azetidine-1-carbonyl}-2,8-dimethylquinoline
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
(2S,4S)-4-amino-N-[(4-fluorophenyl)methyl]-N-[(2-methoxyphenyl)methyl]-1-methylpyrrolidine-2-carboxamide