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7-(3-methoxypropyl)-2-{thieno[3,2-d]pyrimidin-4-yl}-2,7-diazaspiro[4.5]decan-6-one
(3R,9aR)-8-(4-methoxybenzoyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
7-chloro-4-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-methyl-N-[(1R,2S)-2-phenylcyclopropyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[(3S,4R)-1-[3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanoyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
N,N-dimethyl-2-[5-(6-methylpyridin-2-yl)-4-phenyl-1H-imidazol-1-yl]-2-phenylacetamide
2-methoxy-1-[1'-(9H-purin-6-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
2-methyl-N-[2-(2-methylpropanesulfonyl)ethyl]-1,3-benzothiazole-6-carboxamide
3-(2-{[(5-tert-butyl-1H-pyrazol-3-yl)methyl](ethyl)amino}-1-hydroxyethyl)phenol
1-[3-oxo-3-(pyrrolidin-1-yl)propyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-methyl-2-(methylamino)-N-{[2-(trifluoromethyl)phenyl]methyl}acetamide
dimethyl(2-{[6-(4-methylpiperazine-1-carbonyl)pyrazin-2-yl]oxy}hex-5-en-1-yl)amine
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]ethan-1-one
9-[5-(propan-2-yl)pyrimidin-4-yl]-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 2-{1-[(naphthalen-1-yl)carbamoyl]pyrrolidin-3-yl}acetate
[(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl){[5-(oxolan-2-yl)thiophen-2-yl]methyl}amine
8-(5,6-dimethylpyrazin-2-yl)-5-fluoroquinoline
2-[(3-methoxyphenyl)methyl]-4-(4,4,4-trifluorobutyl)morpholine
ethyl 3-benzyl-1-[(2-fluorophenyl)carbamoyl]piperidine-3-carboxylate
1-[6-(2,5-dimethylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
1-(2-fluorophenyl)-N-[1-(1-methyl-1H-imidazol-2-yl)butyl]cyclopropane-1-carboxamide
N-(3-methylphenyl)-3-(1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)propanamide
4-(3-methylphenoxy)-1-(1,3-thiazol-2-yl)piperidine-4-carboxylic acid
4-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-5-[1-(thiophen-3-ylmethyl)-1H-pyrazol-3-yl]-1,3-thiazol-2-amine
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-1-[2-(morpholin-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-cyclopentyl-1-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
3-{1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]piperidin-3-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[(4-phenyloxan-4-yl)methyl]acetamide
1-(1-{1-[(3,4-dimethylphenyl)methyl]piperidin-4-yl}ethyl)-4-methylpiperazine
4-[1-(1-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-4-yl)ethyl]morpholine
5-[1-(2-methoxy-2-methylpropyl)-1H-imidazol-2-yl]-N-(propan-2-yl)pyrimidin-2-amine
2-(2H-1,3-benzodioxol-5-yl)-1-(4-{[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)ethan-1-one
5-[5-(1-ethyl-3-methylpiperidin-3-yl)-1,2,4-oxadiazol-3-yl]-1H-1,3-benzodiazole
2-(2-{[(2-methoxyphenyl)methyl]amino}-4-(morpholin-4-yl)pyrimidin-5-yl)-2-methylpropanoic acid
5-methyl-N-[1-(oxolan-2-ylmethyl)piperidin-4-yl]-1-propyl-1H-pyrazole-4-carboxamide
3-[N-(2-phenylethyl)-1-{2-[(prop-2-en-1-yl)amino]phenyl}formamido]propanamide
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-1-benzoxepine-4-carboxamide
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(pyrrolidine-1-carbonyl)pyrrolidin-3-yl]methanol
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methyl-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-{[2-(1H-imidazol-1-yl)phenyl]methyl}furan-2-carboxamide
1-[(6-methylpyridin-2-yl)methyl]-4-{[1,2,4]triazolo[4,3-a]pyrimidin-5-yl}piperazine
4-[3-(aminomethyl)phenyl]-N-methyl-1H-pyrrolo[2,3-b]pyridin-6-amine
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-[3-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-yl]methanol
2-{1-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-1H-imidazol-2-yl}quinoline
1-[4-(2-methoxyphenoxy)piperidin-1-yl]-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-{[3-(2-aminoethyl)phenyl]methyl}-1-methyl-N-(pyridin-3-ylmethyl)piperidin-4-amine
1-(4-chloro-2-ethylphenyl)-3-cyclopropyl-3-[(1-methyl-1H-pyrazol-4-yl)methyl]urea
[(3R,4R)-1-(3-chloro-4-methylbenzoyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
2-{[1-(3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-6-methylpyridine