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(3S,4S)-1-{[5-(4-ethoxyphenyl)furan-2-yl]methyl}-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
1-{2-[1-(2,5-dimethoxybenzenesulfonyl)piperidin-2-yl]ethyl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
methyl 5-cyano-6-[(3R,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-2-methylpyridine-3-carboxylate
(3aS,6aS)-2-(1H-indol-4-ylmethyl)-5-[3-(methylsulfanyl)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2,4-dimethyl-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]pyrimidine-5-carboxamide
1-[(1-propyl-1H-imidazol-2-yl)methyl]-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
N-{[4-chloro-2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-1-(pyridin-2-ylmethyl)piperidin-3-amine
1-[5-methoxy-2-({methyl[(3-methylpyridin-4-yl)methyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-2-(2-oxopyrrolidin-1-yl)propanamide
5-methyl-5-(4-methylpent-3-en-1-yl)-1-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}piperidin-2-one
2-(1H-1,3-benzodiazol-2-yl)-N-[(2-methylphenyl)(pyridin-4-yl)methyl]acetamide
(1-{[1-(2-methyl-5-propylpyrimidin-4-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-methyl-1,4-diazepane
2-(3-hydroxypropyl)-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(1H-1,2,3,4-tetrazol-5-yl)-N-[1-(thian-4-yl)piperidin-4-yl]benzamide
1-(3-methylbutyl)-8-(2-methylpropyl)-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperidine-3-carboxylate
2-(furan-2-yl)-7-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-oxo-1-(pyridin-2-ylmethyl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]pyrrolidine-3-carboxamide
(4aS,8aR)-6-(pyrazin-2-yl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-3-[4-(3-methylphenyl)piperazin-1-yl]propanamide
2-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1,2,3,4-tetrahydroisoquinoline
2-(furan-2-yl)-1-[1-(thiophen-3-yl)propan-2-yl]-1H-imidazole
N-benzyl-6-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-[1-(1-cyclopropanecarbonylpiperidin-4-yl)-1H-pyrazol-5-yl]-2-methoxy-2-phenylacetamide
2-[benzyl(methyl)amino]-N-[2-(1H-pyrazol-4-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
(1S,5R)-3-(5-fluoro-2-methylbenzoyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(4-phenylbutan-2-yl)-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
1-(3-{3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}piperidin-1-yl)ethan-1-one
5-methyl-3-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-4,5,6,7-tetrahydro-2H-indazole
3-{1-[1-(1,3-benzothiazol-2-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-1-ol
1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-3-(pyridin-4-yl)propan-1-one
5-{[(3R,4S)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]methyl}-2-methoxybenzoic acid
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonane-7-carbonyl]cyclopropane-1-carboxamide
(2-{[4-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)piperazin-1-yl]methyl}phenyl)methanol
3-{[3-(pyridin-2-yl)azetidin-1-yl]methyl}pyridin-2-amine
4-(4-fluorophenoxy)-1-(6-methylpyridazin-3-yl)piperidine-4-carboxylic acid
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-methyl-N-{[2-(trifluoromethyl)phenyl]methyl}pyrimidin-2-amine
4-chloro-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
N-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
2-methoxy-2-phenyl-1-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
N-[3-(3-ethylphenoxy)propyl]-N-methyl-2-(propan-2-yl)pyrimidine-4-carboxamide
8-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-2-[(4-methoxyphenyl)amino]-2-methylpropanamide
2-amino-N,4-dimethyl-N-[(4-phenoxyphenyl)methyl]-1,3-thiazole-5-carboxamide
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-4-(4-methoxybenzoyl)piperazine
1-{[2-methoxy-5-(propan-2-yl)phenyl]methyl}-N,N-dimethylazepan-4-amine
2-methyl-5-[2-(pyrrolidine-1-carbonyl)piperazine-1-carbonyl]pyrazine
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-2-propyl-1,3-thiazole-4-carboxamide