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N-[3-(4-methylpiperazin-1-yl)propyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(pyridine-3-sulfonyl)piperidin-3-yl]piperazine
2-(2-phenylethyl)-N-(prop-2-en-1-yl)morpholine-4-carboxamide
2-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)-1,2-oxazolidin-4-ol
(1S,5R)-3-cyclobutanecarbonyl-N-(4-ethoxyphenyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetamide
1-methyl-9-[1-(phenylamino)cyclopentanecarbonyl]-1,4,9-triazaspiro[5.5]undecan-5-one
5-methyl-N-{[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,3,4-oxadiazol-2-amine
N-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carboxamide
3-ethyl-N-[3-oxo-3-(pyrrolidin-1-yl)propyl]-1H-indole-2-carboxamide
N-(2-hydroxyethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-2-{2-methylimidazo[1,2-a]pyridin-3-yl}acetamide
2-(5-acetylthiophen-3-yl)-N-cycloheptylacetamide
[(3R,4R)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-1-(1-phenylcyclopropanecarbonyl)pyrrolidin-3-yl]methanol
8-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-1-oxa-8-azaspiro[4.5]decane
9-{[3-methoxy-2-(prop-2-yn-1-yloxy)phenyl]methyl}-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
1'-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-1-methyl-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
2-(3-{[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}phenyl)ethan-1-amine
N-[2-(3-carbamoylpiperidin-1-yl)ethyl]-1,3-benzothiazole-6-carboxamide
5-[3-(5-methylfuran-2-yl)-1H-pyrazol-5-yl]-3-[(methylsulfanyl)methyl]-1,2,4-oxadiazole
5-(2-chlorophenyl)-4-[1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidin-3-yl]pyrimidine
N-[5-(4-methylphenoxymethyl)-1,3,4-thiadiazol-2-yl]-1,1-dioxo-1λ6-thiomorpholine-4-carboxamide
4-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
4-[4-(dimethylamino)-5-methylpyrimidin-2-yl]-1-[(4-methylphenyl)methyl]piperazin-2-one
1-butyl-4-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]-1,4-diazepan-6-ol
2-[(1,3-benzothiazol-2-yl)amino]-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]acetamide
4-(2,6-dimethylpyridin-3-yl)-N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]pyrimidin-2-amine
2-(2-methoxy-4-methylphenoxymethyl)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-1,3-oxazole-4-carboxamide
2-amino-4-(3,4-dihydroxyphenyl)-6-(5-methyl-1-propyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
2-(adamantan-1-yl)-N-[1-(1H-imidazol-2-yl)ethyl]acetamide
N-(1,2-oxazol-5-ylmethyl)-3-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzamide
1-(4-chlorophenyl)-N-({1-[(3-methylphenyl)methyl]piperidin-3-yl}methyl)cyclopropane-1-carboxamide
ethyl 1-benzyl-5-(1H-pyrazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
ethyl 2-({3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidine-1-carbonyl}amino)acetate
3-(1,4-oxazepane-4-sulfonyl)-N-(oxolan-2-ylmethyl)benzamide
2-({2-amino-6-[3-(2-methylpropoxy)phenyl]pyrimidin-4-yl}amino)ethan-1-ol
1-(1H-imidazol-4-ylmethyl)-N-[4-(1,3-thiazol-4-yl)phenyl]pyrrolidine-2-carboxamide
2-(pyridin-3-yloxy)-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]acetamide
5-ethyl-N-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-{[4-(2-methanesulfonylethyl)piperazin-1-yl]methyl}-8-methoxyquinoline
5-[methyl(2-phenylethyl)amino]-2-[2-(morpholin-4-yl)-2-oxoethyl]-2,3-dihydropyridazin-3-one
(3R,9aR)-3-[(4-hydroxyphenyl)methyl]-8-[(3-methylphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(4-chloro-2-{[3-(ethylcarbamoyl)pyrrolidin-1-yl]methyl}phenoxy)acetic acid
N-methyl-6-(morpholin-4-yl)-N-(quinolin-8-ylmethyl)pyrimidin-4-amine
N-[phenyl(pyridin-4-yl)methyl]-4-(piperidin-1-yl)butanamide
2-(2-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}ethoxy)ethan-1-ol
(2E)-1-{4-[4-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}-3-phenylprop-2-en-1-one
8-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2,6-dimethyloctan-2-ol
6-fluoro-4-{1-oxa-7-azaspiro[3.5]nonane-7-carbonyl}-1,2,3,4-tetrahydroquinolin-2-one