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3-methyl-N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)furan-2-carboxamide
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-1-[3-(pyridin-3-yl)azetidin-1-yl]propan-1-one
N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-2,3-dioxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
2-({4-[3-(2-fluorophenoxy)azetidine-1-carbonyl]phenyl}sulfanyl)ethan-1-ol
2-[5-(2-amino-5,6,7,8-tetrahydroquinazolin-4-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-hydroxy-2-[4-(trifluoromethyl)phenyl]acetamide
N-cyclopropyl-5-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
8-(3-methoxy-5-methylthiophene-2-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(3S,9aR)-3-[(2S)-butan-2-yl]-8-(4-phenylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(3aS,6aS)-5-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-2-ethyl-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-ethyl-5-[4-(1-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]piperidin-2-one
2-cyclopentyl-9-(2-fluoro-4-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
5-(1-{2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetyl}pyrrolidin-2-yl)thiophene-2-carboxamide
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-3-(3-hydroxyquinoxalin-2-yl)propanamide
5-[4-(2-methoxyethyl)piperazine-1-carbonyl]-1-(3-methylbutyl)-N-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-[3-(propan-2-yloxy)phenyl]pyridine-3-carboxamide
5-{8-benzyl-2,8-diazaspiro[5.5]undecane-2-carbonyl}-N-ethyl-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]piperidin-3-ol
{4-[(4-methoxyphenyl)methyl]-1-(3-methoxypyrazin-2-yl)piperidin-4-yl}methanol
5-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}-N-propylpyrimidin-2-amine
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-5-phenyl-1,2-oxazole-3-carboxamide
(2S,4R)-4-{[(2,6-difluorophenyl)methyl]amino}-N-(2-methoxyethyl)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
[(3R,4R)-1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
2-[6-amino-2-(dimethylamino)pyrimidin-4-yl]benzamide
3-{[1-(2,1,3-benzoxadiazol-5-ylmethyl)pyrrolidin-3-yl]methyl}-1-cyclopentylurea
1-methyl-N-(3-phenylprop-2-yn-1-yl)-N-propyl-1H-pyrrole-2-carboxamide
1-(2-methylpropyl)-4-[4-(trimethyl-1H-pyrazol-4-yl)-1H-imidazol-2-yl]pyrrolidin-2-one
ethyl 2-{[7-(2-chlorobenzamido)-1,2,3,4-tetrahydroisoquinoline-2-carbonyl]amino}acetate
3-{[ethyl(oxan-2-ylmethyl)amino]methyl}pyridin-2-ol
4-(hydroxymethyl)-1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}azepan-4-ol
{3-[(2,4-difluorophenyl)methyl]-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl}methanol
4-(1-ethyl-1H-pyrazole-4-carbonyl)-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-5-methyl-5-phenylpiperidin-2-one
3-(4-ethyl-1H-pyrazol-5-yl)-1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidine
N-[3-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)-2-methylphenyl]furan-2-carboxamide
2-(4-{[5-(2-chlorophenyl)furan-2-yl]methyl}-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl)ethan-1-ol
2-(2H-1,3-benzodioxol-5-ylmethyl)-4-[4-(2-phenylpropyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
(3S,4S)-4-(dimethylamino)-1-[2-(furan-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]pyrrolidin-3-ol
3-methyl-1-[(3-methylphenyl)methyl]-4-(4,4,4-trifluorobutanoyl)piperazin-2-one
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-(diphenylmethyl)acetamide
4-(5-methoxy-1H-indole-2-carbonyl)-5-methyl-1-(3-methylphenyl)piperazin-2-one
1-benzyl-N,N-dimethyl-5-({[4-(trifluoromethoxy)phenyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-acetyl-N-(1,4-oxazepan-6-ylmethyl)-1,2,3,4-tetrahydroquinoline-6-sulfonamide
6-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-9H-purine
N,N-diethyl-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
N-[(2-methoxyphenyl)methyl]-2-{6-oxo-2,7-diazaspiro[4.5]decan-2-yl}acetamide
ethyl 3-[(3-methoxyphenyl)methyl]-1-[(4-methylthiophen-2-yl)sulfonyl]piperidine-3-carboxylate
6-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(2-methoxyethyl)-8-(6-methylpyridazin-3-yl)-2,8-diazaspiro[5.5]undecan-3-one
(1S,5R)-1,3,3-trimethyl-6-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]-6-azabicyclo[3.2.1]octane