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7-fluoro-4-[4-(2-methoxyethyl)piperazine-1-carbonyl]-2-methylquinoline
7-hydroxy-4-(8-hydroxyquinolin-2-yl)-6-methyl-1,2,3,4-tetrahydroquinolin-2-one
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
4-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-3-propylmorpholine
(3S,4R)-4-(2-methoxyphenyl)-1-(oxan-4-yl)pyrrolidine-3-carboxylic acid
6-(1-methylpiperidin-4-yl)-N-[2-(thiophen-2-yl)ethyl]pyrimidin-4-amine
5-methanesulfonyl-N-(oxan-4-ylmethyl)-4-(piperidin-3-yl)pyrimidin-2-amine
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-2,3-dimethylquinoxaline-6-carboxamide
(1R,5R)-6-{[2-(difluoromethoxy)phenyl]methyl}-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
6-(3-ethoxyphenyl)pyridine-3-carboxamide
2-[(6-amino-2-{[(4-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)amino]-1-(piperazin-1-yl)ethan-1-one
1-(3-fluorophenyl)-3-[1-(1-{spiro[2.3]hexane-1-carbonyl}piperidin-4-yl)-1H-pyrazol-5-yl]urea
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-6-(4-hydroxypiperidine-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
6-methoxy-2-oxo-N-[2-(pyridin-2-ylsulfanyl)ethyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
(3S,4S)-4-(4-methylpiperazin-1-yl)-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-ol
9-[(4-fluoro-3-methoxyphenyl)methyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-4-(1H-pyrazol-3-yl)benzamide
N-{[(2S,4S)-1-(3-chloro-4-fluoro-1-benzothiophene-2-carbonyl)-4-fluoropyrrolidin-2-yl]methyl}acetamide
3-[5-(furan-2-yl)-4-phenyl-1H-imidazol-1-yl]-N-(2-methoxyphenyl)propanamide
4-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-2-(morpholin-4-ylmethyl)-1,4-oxazepane
1-phenyl-N-({1-[2-(pyrazin-2-yl)acetyl]piperidin-3-yl}methyl)methanesulfonamide
5-methyl-N-[1-(thiophen-2-ylmethyl)piperidin-3-yl]-1,3-oxazole-4-carboxamide
6-methyl-1-{3-oxo-3-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]propyl}-1,2-dihydropyridin-2-one
1-(piperidin-1-yl)-2-(4-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazin-1-yl)ethan-1-one
5-(1-butanoylpyrrolidin-2-yl)-N-ethyl-N-(pyridin-3-ylmethyl)thiophene-2-carboxamide
methyl[3-(phenylsulfanyl)propyl]{[6-(trifluoromethyl)pyridin-3-yl]methyl}amine
N-[3-(cyclopentyloxy)propyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-(methylamino)-1-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
4-(4-methyl-4H-1,2,4-triazol-3-yl)-1-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidine
N-(4-chlorophenyl)-2-ethyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
4-(1H-pyrazol-3-yl)-8-(trifluoromethyl)quinoline
N-(2-methylpropyl)-1-[1-(quinoline-8-sulfonyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
1-{5-[2-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1H-1,2,4-triazol-1-yl}butan-2-ol
N,N-dimethyl-5-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}pyridin-2-amine
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
1-{2-[(1-methylpiperidin-4-yl)oxy]phenyl}-3-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]urea
N-{3-[(5-methylpyridin-2-yl)amino]propyl}-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
[2-(2-methoxyphenyl)ethyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
5-(2-chlorophenyl)-N-[2-(1H-imidazol-4-yl)ethyl]-2-methylfuran-3-carboxamide
(4aR,7aS)-1-[2-(quinolin-7-yloxy)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[7-(oxan-4-yl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]oxane-4-carbonitrile
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(1H-indol-3-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(3S)-3-(dimethylamino)-N-[2-(4-fluorophenoxy)phenyl]pyrrolidine-1-carboxamide
3-(1-{1-[(2,5-dimethylthiophen-3-yl)sulfonyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-1-ol
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
1-[2-(cyclohexylmethyl)morpholin-4-yl]-3-(1,2-oxazinan-2-yl)propan-1-one
(4aS,7aR)-1-(2-methoxypyridine-3-carbonyl)-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(2-amino-1,3-thiazol-4-yl)-1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]propan-1-one
(4aR,7aS)-1-cyclobutanecarbonyl-4-(2-phenylethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(methylsulfanyl)ethyl]amine