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4-{6,7-dimethoxy-2-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1,2,3,4-tetrahydroisoquinolin-1-yl}phenol
3-hydroxy-1-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)propan-1-one
3-(pyridin-2-yl)-3-(pyridin-4-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)propanamide
3-(3-hydroxy-3-methylbutyl)-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]benzamide
11-{methyl[2-(pyridin-2-yl)ethyl]amino}-4-(3-methylbutyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-hydroxy-1-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperidine-4-carboxylic acid
5-benzyl-1-(3-methoxyphenyl)-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-2-one
N-{2-[(3-{[(3-methylphenyl)methyl]amino}-5-[(2-methylphenyl)sulfamoyl]phenyl)formamido]ethyl}acetamide
2-(2-methylpropyl)-8-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-2,8-diazaspiro[4.5]decan-3-one
(3S,4R)-1-(2-hydroxy-4-methoxybenzoyl)-4-methylpiperidine-3,4-diol
2-({2-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]phenyl}amino)acetic acid
N-[2-(1H-imidazol-2-yl)ethyl]-6-methyl-2-(morpholin-4-yl)pyrimidin-4-amine
5-fluoro-1-methyl-3-[2-(morpholin-4-ylmethyl)phenyl]-1H-indazole
2-methyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-4-phenylpyrimidine-5-carboxamide
(1R,5S,8R)-8-methoxy-3-({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)-3-azabicyclo[3.2.1]octane
N-phenyl-1-(4-phenylbenzoyl)piperidin-3-amine
5,8-dimethyl-2-{[(2S)-2-(piperidine-1-carbonyl)pyrrolidin-1-yl]methyl}quinolin-4-ol
3-[(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)methyl]-1H-indole
1-[2-methoxy-4-(1,4-oxazepan-4-ylmethyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
N-(propan-2-yl)-1-[(1s,4s)-4-[2-(1-methyl-1H-pyrrol-3-yl)acetamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-aminothiophene-2-carboxamide
methyl (2S)-2-{[5-(cycloheptylcarbamoyl)-1-cyclopropyl-4-oxo-1,4-dihydropyridin-3-yl]formamido}-2-phenylacetate
1-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]cyclopropane-1-carboxamide
8-fluoro-2-[(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)methyl]quinolin-4-ol
1-(carbamoylmethyl)-N-ethyl-N-[2-(4-fluorophenoxy)ethyl]piperidine-4-carboxamide
6-methyl-2-({2-[(3-methylpyrazin-2-yl)amino]ethyl}amino)-3,4-dihydropyrimidin-4-one
2-methyl-5-(propan-2-yl)-N-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
5-(2,6-difluorophenoxymethyl)-N-(1H-imidazol-2-ylmethyl)-1,2-oxazole-3-carboxamide
3-cyclopropyl-N-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-1H-pyrazole-5-carboxamide
6-(4-chlorophenyl)-N-ethyl-N-(oxolan-2-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
(4aS,8aR)-6-(2-aminoacetyl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
3-(2-methylpropyl)-1-(2-phenylethyl)-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(oxolan-3-yl)-5-[5-(propan-2-yl)-1,2-oxazol-3-yl]-1,2,4-oxadiazole
5-(3-aminopyrrolidine-1-carbonyl)-2-[(2,6-dichlorophenyl)methyl]pyrimidin-4-ol
7-fluoro-2-methyl-4-[4-(9H-purin-6-yl)piperazine-1-carbonyl]quinoline
methyl (1R,3S,3aR,6aS)-1,5-dimethyl-3-(3-methyl-1,2-benzoxazol-5-yl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)pyrimidin-2-amine
N-(2-ethoxyphenyl)-N'-ethyl-N'-(pyridin-4-ylmethyl)propanediamide
N-[(3S,4R)-1-(dimethyl-1,3-oxazole-4-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
3-({[(4,6-dimethylpyridin-3-yl)methyl]amino}methyl)-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
1-[3-(6-hydroxypyrimidin-4-yl)piperidin-1-yl]-3-(3-hydroxyquinoxalin-2-yl)propan-1-one
N'-(2-fluoro-5-methylphenyl)-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)butanediamide
ethyl 3-{[(3S,4S)-3,4-bis(hydroxymethyl)pyrrolidine-1-carbonyl]amino}-1-benzothiophene-2-carboxylate
1-{2-[(1H-indol-7-ylmethyl)(methyl)amino]ethyl}cyclopentan-1-ol
1-ethyl-8-[(3-methoxyphenyl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(pyridin-3-yl)-7-(4,4,4-trifluorobutanoyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(3-fluoro-4-hydroxyphenyl)-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-(furan-2-ylmethyl)-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)piperidine-3-carboxamide
5-cyclobutyl-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1,3,4-oxadiazol-2-amine
2-acetyl-8-(5-fluoropyrimidin-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid