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N-{[4-(methylsulfanyl)phenyl]methyl}-N-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}cyclopropanamine
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2-(pyrrolidin-3-yl)benzamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1-benzothiophene-5-carboxamide
3-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-1-(3-methylcinnolin-5-yl)urea
2-hydroxy-N-({1-[(4-methoxy-2,3-dimethylphenyl)methyl]pyrrolidin-3-yl}methyl)acetamide
(3S,9aR)-8-[(2,4-dimethylphenyl)methyl]-3-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[(3-fluorophenyl)methyl]-3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
N-(2-oxopyrrolidin-3-yl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]oxane-2-carboxamide
N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
(1S,5R)-6-(2-phenylethyl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-(1-methyl-1H-pyrazol-4-yl)-N-[2-(3-phenylpiperidin-1-yl)ethyl]propanamide
ethyl 3-[(4-fluorophenyl)methyl]-1-[3-(1,2-oxazinan-2-yl)propanoyl]piperidine-3-carboxylate
6-[3-(2-methoxyethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]-1,3-benzothiazole
6-(2-benzyl-1,3-thiazole-4-carbonyl)-1-methyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
8-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-{[(2R)-1-hydroxybutan-2-yl]amino}pyridine-2-carboxamide
5-{2-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(3-chloro-4-methylphenyl)-5-[(S)-methoxy(phenyl)methyl]-1,2,4-oxadiazole
3-(1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-2-yl)propan-1-ol
1-[(3-methylphenyl)methyl]-4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}piperazine
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-(2-hydroxyethyl)-N-methylacetamide
(1S,5R)-3-(2,1,3-benzoxadiazol-4-ylmethyl)-3,9-diazabicyclo[3.3.2]decan-10-one
5-(4-methoxyphenyl)-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]furan-2-carboxamide
4-[2-(4-fluorophenyl)ethyl]-11-[(1,2-oxazol-3-ylmethyl)amino]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-[(2-{3-[cyclohexyl(methyl)amino]-2-hydroxypropoxy}phenyl)methyl]-4-methylpiperidine-4-carbonitrile
1,2,5-trimethyl-N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)-1H-pyrrole-3-carboxamide
2-(4-benzylmorpholin-2-yl)-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
2-{2-methyl-3-[({[2-(trifluoromethyl)phenyl]methyl}amino)methyl]-1H-indol-1-yl}acetamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)acetamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[4-(1H-pyrazol-3-yl)benzoyl]-4-(pyridin-4-yl)piperazine
N-methyl-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
2-(1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-2-yl)pyridine
N-methyl-N-{2-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}methanesulfonamide
N-(4-methoxyphenyl)-2-{4-[2-(3-methyl-6-oxo-1,6-dihydropyridazin-1-yl)acetyl]morpholin-3-yl}acetamide
N4-{[3-(3-fluorophenyl)-1,2-oxazol-5-yl]methyl}-5,6,7,8-tetrahydroquinazoline-2,4-diamine
[1-(5-chloropyridin-2-yl)-3-(2-phenoxyethyl)piperidin-3-yl]methanol
2-(4-chloro-2-methylphenoxy)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]ethan-1-one
1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]-4-(morpholin-4-yl)butan-1-one
N-{[4-(cyclohex-3-en-1-ylmethoxy)phenyl]methyl}-N-cyclopropylthiophene-2-carboxamide
8-[2-(2-methoxy-4-methylphenoxy)ethyl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]acetamide
2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}-1-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
8-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-3-[2-(dimethylamino)ethyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{[2-(benzyloxy)phenyl]methyl}-2-methylpyrimidine-5-carboxamide
1-[(3-chlorophenyl)methyl]-5-(thiomorpholin-4-yl)azepan-2-one