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1-tert-butyl-3-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1H-pyrrole
3-(1H-imidazol-1-ylmethyl)-1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidine
2-benzyl-8-(piperidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
N-({2-[3-(2-methoxyacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-4-methyl-2-oxopentanamide
1-(2-methoxyacetyl)-N-methyl-N-(quinoxalin-2-ylmethyl)piperidine-3-carboxamide
2-[4-cycloheptyl-1-(3-methylbutyl)piperazin-2-yl]ethan-1-ol
4-[1-ethyl-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]-6-fluoro-1,2,3,4-tetrahydroquinolin-2-one
(2S)-2-({5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}amino)propanamide
{2-[(4-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}piperazin-1-yl)methyl]phenyl}methanol
{5-[1-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1H-imidazol-2-yl]furan-2-yl}methanol
1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
1-(6-chloro-1,3-benzothiazol-2-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[2-(7-chloro-4-oxo-3,4-dihydroquinazolin-3-yl)ethyl]acetamide
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-(2-methylbenzoyl)piperidin-3-ol
methyl 3-[(pyridin-3-ylformamido)methyl]-5-[2-(thiophen-3-yl)acetamido]benzoate
5-({3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-N-propylpyrimidin-2-amine
3-methyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1H-pyrazole-5-carboxamide
methyl[(2-methyl-1,3-thiazol-4-yl)methyl][(2R)-2-phenylbutyl]amine
5-methyl-N-[2-(4-methyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]thiophene-2-carboxamide
(3S,4S)-1-(cyclopentylcarbamoyl)-4-cyclopropylpyrrolidine-3-carboxylic acid
4-[(3-hydroxypiperidin-3-yl)methyl]-1-[(4-methoxyphenyl)methyl]piperazin-2-one
1-[5-(3-chlorophenyl)-1,2,4-triazin-3-yl]-4-[(3-fluorophenyl)methyl]-1,4-diazepane
1-[1-(cyclopent-1-ene-1-carbonyl)piperidin-3-yl]-4-(2-methylphenyl)piperazine
cyclopentyl 4-{[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]amino}benzoate
4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)-N-(2,5-dimethylphenyl)piperidine-1-carboxamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)acetamide
5-{4-[6-(propan-2-yloxy)pyridazin-3-yl]phenyl}imidazolidine-2,4-dione
5-cyclopropyl-N,N-diethyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-{[6,7-dimethoxy-2-(3-methoxyphenyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)-4-(1H-pyrazol-1-yl)benzamide
2-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carbonyl)-2-azabicyclo[2.2.1]heptane
(4S)-3-{2-[3-(2-methoxyphenoxy)azetidin-1-yl]-2-oxoethyl}-4-phenyl-1,3-oxazolidin-2-one
3-(2-{4-[(dimethylamino)methyl]phenyl}piperidine-1-carbonyl)-1,6-dimethyl-1,2-dihydropyridin-2-one
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-(oxan-4-yl)pyrrolidine-2-carboxamide
N-{2-[5-(2-methoxy-4-methylphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}-2-methylpropanamide
N,N-dimethyl-2-[3-(2-phenylethyl)piperidin-1-yl]pyridine-3-carboxamide
3-({[(5,6-dimethylpyridin-3-yl)methyl]amino}methyl)-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
[(1-benzylpyrrolidin-3-yl)methyl](methyl){4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}amine
8-[(2-ethyl-1,3-thiazol-4-yl)methyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
N-ethyl-1-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]pyrrolidine-3-carboxamide
3-{[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]methyl}-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one
4-ethyl-3-{1-[3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(3-phenylpiperazine-1-carbonyl)-5,6,7,8-tetrahydroquinoline
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-(methoxymethyl)thiophene-2-carboxamide
(4aS,7aR)-1-(3-hydroxypyridine-2-carbonyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
2-methyl-6-(7-methyl-1H-1,3-benzodiazol-2-yl)phenol
6-{[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}-1,4-oxazepan-6-ol
1-(diethylamino)-3-(2-methoxy-4-{[(prop-2-en-1-yl)amino]methyl}phenoxy)propan-2-ol
2-(2-phenyl-1,3-thiazol-4-yl)-1-[3-(1H-pyrazol-5-yl)piperidin-1-yl]ethan-1-one
N-[(6-chloropyridin-3-yl)methyl]-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetamide