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{1-[1-(6-methylpyridazin-3-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}(phenyl)methanol
5-[1-(cyclohex-3-en-1-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1,2-dimethyl-1H-imidazole
N-[2-(2,5-dimethylphenoxy)ethyl]-2-[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]-N-methylacetamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-5-fluoro-4-(pyrrolidin-1-yl)pyrimidine
2-{methyl[(3-methylpyridin-2-yl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
1-{1,3-dioxo-2-[2-(1H-pyrazol-1-yl)ethyl]-2,3-dihydro-1H-isoindol-4-yl}-N-[(4-methylphenyl)methyl]piperidine-3-carboxamide
(3aR,6aS)-2-(2-methyl-1-benzofuran-7-carbonyl)-octahydropyrrolo[3,4-c]pyrrole
3-{5-[(2R)-oxolane-2-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-(propan-2-yl)propanamide
N-benzyl-4-[4-(thiomorpholin-4-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
1-[(3-ethoxy-4-methoxyphenyl)methyl]-4-[(4-methylphenyl)methyl]-1,4-diazepan-5-one
N-{1-[(4-fluorophenyl)methyl]piperidin-3-yl}-4-hydroxy-2-methylpyrimidine-5-carboxamide
2-acetamido-N-[4-methoxy-2-(2-methylpropanamido)phenyl]pentanamide
(1S,6R)-3-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-3,9-diazabicyclo[4.2.1]nonane
7-fluoro-1-methyl-2-(5-methyl-1,3-oxazole-4-carbonyl)-1,2,3,4-tetrahydroisoquinoline
4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]-1-(2-methylpentyl)piperidine
1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-N-(pyrimidin-4-ylmethyl)piperidine-3-carboxamide
N,N-dimethyl-5-{methyl[(4-methyl-1,3-thiazol-2-yl)methyl]amino}-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-(1-{5-[(cyclohexylmethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}-2-phenylethyl)-2-(1-methyl-1H-pyrrol-3-yl)acetamide
N-[2-(3-phenylpiperidin-1-yl)ethyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N6-[(2-methyl-1,3-thiazol-4-yl)methyl]-9H-purine-2,6-diamine
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-2-oxo-N-(oxolan-2-ylmethyl)propanamide
N-[3-(2-ethylphenoxy)propyl]-N-methyl-3-(1H-pyrazol-4-yl)propanamide
4-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-1-methylpiperazine-2-carboxylic acid
[(3S,5R)-1-(2,1,3-benzothiadiazol-5-ylmethyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
4-{3-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]propoxy}benzamide
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(thiophene-3-carbonyl)pyrrolidin-3-yl]-2-oxo-2,3-dihydro-1H-imidazole-4-carboxamide
N-(2,3-dihydro-1H-inden-5-yl)-2-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]morpholine-4-carboxamide
5-methyl-1-(5-methylpyridin-2-yl)-1H-pyrazole-3-carboxylic acid
N-{5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-4-methylphenyl]pyridin-2-yl}acetamide
(3R,4R)-1-(5,6-dimethylpyrimidin-4-yl)-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
4-(1-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}piperidin-4-yl)thiomorpholine
{[7-chloro-2-(2,5-dimethoxyphenyl)quinolin-3-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)butanamide
N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-6-(morpholin-4-yl)pyrimidin-4-amine
1-{4-[2-(cyclopropylcarbamoyl)ethyl]phenyl}-5-oxopyrrolidine-3-carboxylic acid
1-[5-chloro-2-(1H-1,2,4-triazol-1-yl)phenyl]-3-ethyl-3-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]urea
(4aS,7aR)-1-[(2-methylpyrimidin-5-yl)methyl]-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-[4-(methylamino)pyrimidin-2-yl]-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
methyl 6-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-1-methyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxylate
2-({[1-(2-fluorophenyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)-5-methyl-1,3,4-oxadiazole
(2E)-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-3-(1-methyl-1H-pyrazol-4-yl)-N-(oxolan-2-ylmethyl)prop-2-enamide
8-(1H-1,3-benzodiazol-2-ylmethyl)-3-[(4-methoxyphenyl)methyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-1-oxopropan-2-yl)-1,2-dihydrophthalazin-1-one
[(3R,4R)-1-[6-(dimethylamino)pyridine-3-carbonyl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
N-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-N-[(1-methyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
N3-(cyclohexylmethyl)-1-cyclopropyl-N5-[3-(dimethylamino)-2,2-dimethylpropyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-(1-benzyl-1H-pyrazol-4-yl)-2-[4-(pyridin-3-yloxy)piperidin-1-yl]acetic acid
3-[1-(5-aminopyridin-3-yl)-1H-pyrazol-4-yl]benzoic acid
N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)-2-methoxypyridine-3-carboxamide