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(1R,5R)-N,N-dimethyl-6-[3-(prop-2-en-1-yloxy)benzoyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
1-[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]-3-(1,2-oxazinan-2-yl)propan-1-one
(2S,4R)-4-amino-1-(2-{[(3,5-dimethylphenyl)methyl]sulfanyl}acetyl)-N-methylpyrrolidine-2-carboxamide
N,3-dimethyl-1-propyl-N-(quinoxalin-2-ylmethyl)-1H-pyrazole-4-carboxamide
(1S,5R)-3-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(4aS,8aR)-N-benzyl-1-(4-hydroxybutyl)-2-oxo-decahydro-1,6-naphthyridine-6-carboxamide
3-(2-{3-[2-(2,3-dihydro-1H-isoindol-2-yl)-2-oxoethyl]morpholin-4-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
(2R)-2-cyclohexyl-2-hydroxy-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
N-{[5-methyl-7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1,2,3-thiadiazole-4-carboxamide
6-cyclopropyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)pyrimidin-4-amine
1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
3-{2-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
8-fluoro-3-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3,4-dihydroquinazolin-4-one
2-(1H-1,3-benzodiazol-1-ylmethyl)-N-[3-(methylsulfanyl)propyl]-1,3-oxazole-4-carboxamide
N-cyclopentyl-2,5-dimethoxy-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}benzene-1-sulfonamide
4-(1H-imidazol-1-yl)-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]butanamide
(3S,4S)-3-hydroxy-N-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-4-(4-methylpiperazin-1-yl)pyrrolidine-1-carboxamide
2-[(3S)-3-hydroxypyrrolidin-1-yl]-N,1-dimethyl-N-(1H-pyrazol-3-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
(4-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methanol
N-methyl-3-(3-methylpiperazine-1-carbonyl)-N-[2-(methylsulfanyl)ethyl]benzene-1-sulfonamide
4-(5-methylpyridin-2-yl)-1-(1,3,7-trimethyl-1H-indole-2-carbonyl)piperidin-4-ol
3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]propanamide
2-[(4-acetyl-6-hydroxy-1,4-diazepan-1-yl)methyl]-6-methyl-1,4-dihydroquinolin-4-one
4-(dimethyl-1,2-oxazol-4-yl)-3-(furan-2-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[(4aR,7aS)-6,6-dioxo-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
1-(3-methoxy-5-methylthiophene-2-carbonyl)-4-(piperidine-1-carbonyl)piperidine
2-{4-cyclobutyl-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
(1S,5R)-3-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
[(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)sulfamoyl]dimethylamine
(1-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methanol
(3S)-3-benzyl-4-(1,3-thiazol-4-ylmethyl)piperazin-2-one
2-(2-methoxyethyl)-1-{[2-(2-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
4-chloro-1-methyl-N-[(3R)-pyrrolidin-3-yl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
3-[(dimethylamino)methyl]-1-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]pyrrolidin-3-ol
5-tert-butyl-4-({3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.5]decan-7-yl}methyl)furan-2-carboxamide
3-(4-cyclopentyl-1,4-diazepane-1-carbonyl)-6-phenyl-1,2-dihydropyridin-2-one
3-({1-[(1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-4-yl}methyl)-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(4-{[3-(trifluoromethyl)phenyl]methyl}morpholin-2-yl)ethan-1-ol
6-(pyrrolidin-1-ylmethyl)-4-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-1,4-oxazepan-6-ol
N-(3-hydroxypropyl)-5-{1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
2-[(4-chlorophenyl)methyl]-8-(2-methylpyrimidine-5-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
(3S,4R)-1-[(2,3-dimethoxyphenyl)methyl]-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-(1,2-oxazol-3-ylmethyl)-2-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzamide
2-(2H-1,3-benzodioxol-5-yl)-1-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethan-1-one
2-{[3-(propan-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
(3aS,6aR)-5-[(5-chlorothiophen-2-yl)methyl]-3-cyclopentyl-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-methyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-3-propanamidobenzamide
1-(cyclopropylmethyl)-5-(pyridine-3-sulfonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(6-methylquinolin-4-yl)pyrrolidin-3-yl]methanol