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N-[(3R,4S)-4-cyclopropyl-1-(dimethylcarbamoyl)pyrrolidin-3-yl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-benzylpiperidine-4-carboxamide
(3S,9aR)-3-[(2S)-butan-2-yl]-8-[(4-methylphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3,5-dimethoxy-2-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}benzoic acid
3-[5-(5-chloro-2-fluorobenzoyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl]pyridine
methyl (2S,4S,5R)-4-[(cyclopropylmethyl)carbamoyl]-5-(2,3-difluorophenyl)-1-methylpyrrolidine-2-carboxylate
N-{[5-({cyclopropyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)furan-2-yl]methyl}-N-methylmethanesulfonamide
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-[(3R,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]acetamide
1-[5-(4-ethylphenyl)-4-phenyl-1H-imidazol-1-yl]-3-methoxypropan-2-ol
1-(2-{2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholin-4-yl}-2-oxoethyl)-4,4-dimethylpyrrolidin-2-one
3-[3-(oxolan-3-yl)-1-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]quinoline
2-({[(propan-2-yl)carbamoyl]methyl}sulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
(4aS,7aR)-1-[(2-methoxy-4-methylphenyl)methyl]-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[4-(pyrrolidine-1-carbonyl)phenoxy]-1-[(2,4,5-trimethylphenyl)methyl]piperidine
N-[1-(1-propyl-1H-1,2,4-triazol-5-yl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
4-[(4-methoxy-3-methylphenyl)methyl]-3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]piperazin-2-one
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}acetamide
N-[(3R,4S)-1-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-4-propylpyrrolidin-3-yl]acetamide
1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)-3-[4-(trifluoromethyl)benzoyl]piperidine
2-[(3,4-dihydro-2H-1-benzopyran-3-ylformamido)methyl]-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-3-methyl-1H-pyrazole-5-carboxamide
3-(pyridin-4-yl)-1-[4-(thian-4-yl)piperazin-1-yl]propan-1-one
2-(cyclohex-1-en-1-yl)-N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
4-{1-[(4-methoxyphenyl)methyl]-1H-imidazol-2-yl}quinoline
N-(piperidin-4-ylmethyl)-4-(pyrrolidin-3-yl)benzamide
3-({1-butyl-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl}methyl)-4-ethylpiperazin-2-one
N-(2-methylpropyl)-N-(pyridin-2-ylmethyl)-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
methyl 4-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-4-oxobutanoate
2-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-{[1-(hydroxymethyl)cyclobutyl]methyl}-N-methyl-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
2-[(2-amino-5,6-dimethylpyrimidin-4-yl)amino]-1-(pyrrolidin-1-yl)ethan-1-one
5-methyl-3-{2-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
1-[(4aR,8aR)-6-[(4-fluorophenyl)methyl]-decahydro-1,6-naphthyridin-1-yl]-2-(3-methyl-1H-1,2,4-triazol-5-yl)ethan-1-one
1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(1-methylpiperidin-4-yl)piperidine
2-{2-[2-(5-phenylthiophen-2-yl)-1H-imidazol-1-yl]ethyl}pyrazine
3-methyl-8-[2-(3-oxo-2,3-dihydro-1,2-benzothiazol-2-yl)acetyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-amino-4-[2-(2-hydroxyethoxy)phenyl]-6-(3-methoxyphenyl)pyridine-3-carbonitrile
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-[3-(3-methoxyphenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
9-methyl-3-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]-3,9-diazaspiro[5.6]dodecan-10-one
2-(2-hydroxyethyl)-8-[3-(4-hydroxyphenyl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
2-{5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-[hydroxy(phenyl)methyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
1-cyclohexyl-5-[2-(2-methoxyphenyl)ethyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidine
7-[(3,4-difluorophenyl)methyl]-2-(pyrazine-2-carbonyl)-2,7-diazaspiro[4.5]decane
N-(3-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-oxopropyl)acetamide
1-[3-(benzyloxy)piperidin-1-yl]-3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]propan-1-one
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-6-(4-methoxypiperidin-1-yl)pyridine-3-carboxamide
2-(4-{[2-(5-methylfuran-2-yl)phenyl]methyl}piperazin-1-yl)-1-(pyrrolidin-1-yl)ethan-1-one
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-({[(5-methylfuran-2-yl)methyl]amino}methyl)piperidin-2-one
3-({[(4-chlorophenyl)(phenyl)methyl]amino}methyl)-7-(methylsulfanyl)-1-(pyridin-2-ylmethyl)-1,2-dihydroquinolin-2-one