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2-(5-acetylthiophen-3-yl)-N-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}acetamide
2-[(1R,5S)-3,8-diazabicyclo[3.2.1]octan-3-yl]-7-methanesulfonyl-4-methylquinazoline
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(furan-2-ylmethyl)methylamine
N-methyl-2-oxo-N-[(1-phenylpyrrolidin-3-yl)methyl]-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
5-[(4aS,8aS)-7-cyclobutanecarbonyl-4a-hydroxy-decahydro-2,7-naphthyridine-2-carbonyl]-1-methyl-1H-pyrrole-3-carbonitrile
4-(2-fluorophenyl)-3-(3-methoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
8-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}quinolin-4-amine
1-{1-[(2,3-difluoro-6-methoxyphenyl)methyl]piperidin-4-yl}piperidin-4-ol
4-[3-({1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)-2,5-dimethyl-1H-pyrrol-1-yl]-4H-1,2,4-triazole
N-benzyl-N,1-dimethyl-5-{[3-(pyridin-4-yl)propyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-{1-[(2E)-4-methylpent-2-en-1-yl]piperidin-4-yl}-N-(2-phenylethyl)piperidine-4-carboxamide
3-(propan-2-yl)-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)-1,2-oxazole-5-carboxamide
(3S,4R)-4-(hydroxymethyl)-1-[2-(pyridin-3-yl)-1,3-thiazole-4-carbonyl]piperidin-3-ol
2-{[4-(3-fluoropyridin-4-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
3-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-4-methylpyridine
4-[1-(4-carboxybutanoyl)piperidin-3-yl]benzoic acid
1-{1-[(4-ethylphenyl)methyl]piperidin-3-yl}-N-(3-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide
3-{1-[1-(2-hydroxyacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methoxyphenyl)urea
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-3-ethyl-5-methyl-1,2-oxazole
(3S,7S)-5-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
2-{[4-(4-benzyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}benzonitrile
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-3-propyl-1H-pyrazole-4-carboxamide
2-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyrimidin-4-amine
3-cyclopropyl-5-[2-(2-methoxyphenyl)ethyl]-1H-1,2,4-triazole
5-methyl-N-{4-[2-(1H-pyrazol-1-yl)butanamido]phenyl}furan-2-carboxamide
(1,4-dioxan-2-ylmethyl)({[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl})amine
(4aS,8aR)-6-(3-chloropyridin-2-yl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)-2-(pyridin-3-yl)acetamide
(3S,5S)-1-(2-phenylacetyl)-5-[(pyridin-4-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
3-{2-[(4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]propanamide
4-{3,9-diazaspiro[5.5]undecane-3-carbonyl}-N-propylaniline
N,2-dimethyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]thieno[3,2-d]pyrimidin-4-amine
5-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-1-propyl-1H-pyrazole-4-carboxamide
1-[2-({[3-chloro-5-methoxy-4-(prop-2-en-1-yloxy)phenyl]methyl}amino)ethyl]-4,6-dimethyl-1,2-dihydropyrimidin-2-one
9-[(3-methylpyridin-2-yl)methyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butan-1-one
3-[(3R,4S)-4-(dimethylamino)-1-(2-fluoro-4-methylbenzoyl)piperidin-3-yl]propan-1-ol
2-chloro-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]benzamide
4-{[2-(3-methoxyphenyl)ethyl]amino}-5-methyl-N-[(3-methyloxetan-3-yl)methyl]thieno[2,3-d]pyrimidine-6-carboxamide
[1-(5,6-dimethylpyrimidin-4-yl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
1-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-2-methyl-2-[(4-methylphenyl)amino]propan-1-one
7-[2-(5-methylfuran-2-yl)ethyl]-2-oxa-7-azaspiro[4.5]decan-8-one
ethyl N-{[(2S,4S)-1-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]-4-fluoropyrrolidin-2-yl]methyl}carbamate
4-(4-chlorophenyl)-N-(piperidin-3-ylmethyl)butanamide
1-(1H-1,2,4-triazole-3-carbonyl)-4-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]piperazine
1-(3-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-3-oxopropyl)-6-methyl-1,2-dihydropyridin-2-one
2-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-4-methylphenol
2-[3-(3-ethylphenoxy)azetidine-1-carbonyl]-6-methylpyridine
(1R,5R)-3-methanesulfonyl-6-{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
methyl[(1-methyl-1H-pyrazol-4-yl)methyl][(2-phenyl-1,3-thiazol-5-yl)methyl]amine