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2-(1-{[1-(pyrrolidine-1-sulfonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-ol
(2-methoxyethyl)[(2-propylpyrimidin-5-yl)methyl](thiophen-2-ylmethyl)amine
(1R,5R)-3-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-3,9-diazabicyclo[3.3.2]decan-10-one
3-(3-chloro-1H-1,2,4-triazol-5-yl)-1-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]propan-1-one
2-{5-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
4-methyl-3-({[1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)-4H-1,2,4-triazole
N-(1-{1-[(4-acetamidophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxybenzamide
methyl[1-(pyridin-2-yl)ethyl]{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
N-[3-(dimethylcarbamoyl)phenyl]-3-phenylpiperazine-1-carboxamide
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
1-[1-(2-methylfuran-3-carbonyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
8-(1-benzothiophene-2-sulfonyl)-2-methyl-2,8-diazaspiro[4.5]decan-3-one
3-[(3,3-dimethylcyclohexyl)amino]-N-[3-(1H-imidazol-1-yl)propyl]-5-(pyrrolidine-1-sulfonyl)benzamide
2-fluoro-5-[2-(morpholin-4-ylmethyl)phenyl]benzamide
2-{4-[(8-methoxyquinolin-2-yl)methyl]-1-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
1-(1-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}pyrrolidin-3-yl)piperidine
ethyl 3-{[3-(6-methoxynaphthalene-2-carbonyl)piperidine-1-carbonyl]amino}propanoate
(3aS,6aS)-2-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{[(cyclopropylmethyl)(2-methoxyethyl)amino]methyl}-6,8-dimethylquinolin-4-ol
(3R,4R)-3-cyclopropyl-4-methyl-1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)pyrrolidin-3-ol
8-({4-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)-2-methyl-2,8-diazaspiro[4.5]decan-3-one
(2S)-1-acetyl-N-butyl-N-[(3-methylthiophen-2-yl)methyl]pyrrolidine-2-carboxamide
1-[1-(2-amino-6-methylpyrimidin-4-yl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
2-ethyl-4-methyl-N-{5-[2-(3-methylphenoxy)ethyl]-1,3,4-thiadiazol-2-yl}-1,3-oxazole-5-carboxamide
2-{[5-(3-acetylphenoxymethyl)-1H-pyrazol-3-yl]formamido}-N,2-dimethylpropanamide
1-{4-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]thiophen-2-yl}ethan-1-one
(4aR,7aS)-1-[(5-methylfuran-2-yl)methyl]-4-[2-(1H-1,2,4-triazol-1-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(dimethyl-1,3-thiazole-5-carbonyl)-4-(4-ethyl-1H-pyrazol-5-yl)piperidine
1-cyclopentyl-4-{[methyl(9H-purin-6-yl)amino]methyl}pyrrolidin-2-one
1-(1H-imidazol-2-ylmethyl)-4-(3-methylphenoxy)piperidine
1-(2-{2-azaspiro[5.5]undecan-2-yl}-2-oxoethyl)-3-methoxy-1,2-dihydropyridin-2-one
8-[(3-methylphenyl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
3-chloro-4-{[methyl({[1-(propan-2-yl)piperidin-3-yl]methyl})amino]methyl}phenol
1-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-5-oxopyrrolidine-3-carboxylic acid
(3aS,6aS)-5-{[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]methyl}-1-oxo-2-propyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[5-(2-methoxyacetamido)-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carbonyl]piperidine-3-carboxamide
4-{4-[(4-chlorophenyl)methyl]piperazin-1-yl}-2-[(4-methoxyphenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
4-{3-methyl-5-[(methylamino)methyl]-1H-1,2,4-triazol-1-yl}benzene-1-sulfonamide
N-({1-[(2-aminopyrimidin-5-yl)methyl]piperidin-3-yl}methyl)cycloheptanecarboxamide
1-{5-[3-benzyl-3-(hydroxymethyl)piperidine-1-carbonyl]-2-methylphenyl}imidazolidin-2-one
1-{2-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-methyl-N-[(4-methylphenyl)methyl]piperidin-4-amine
9-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}-3-azaspiro[5.5]undecane
1-[2-({4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl}amino)ethyl]piperidine-3-carboxamide
1-(2,3-dihydro-1-benzofuran-7-carbonyl)-3-(1H-pyrazol-5-yl)piperidine
N-[2-(3-methoxyphenyl)phenyl]-1-(pyrazin-2-yl)piperidine-4-carboxamide
4-(6-ethyl-2-methylpyrimidin-4-yl)-2-(6-methoxynaphthalen-2-yl)morpholine
1-(azepan-1-yl)-3-{3-[(3,3,4-trimethylpiperazin-1-yl)methyl]phenoxy}propan-2-ol
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-2-(1-ethylpiperidin-4-yl)acetamide
{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(oxan-4-ylmethyl)amine