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N,N-dimethyl-5-[(4-{[1,2,4]triazolo[4,3-a]pyrimidin-5-yl}piperazin-1-yl)methyl]pyridin-2-amine
1-(2,6-dimethoxypyridin-3-yl)-3-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}urea
(pyridin-3-ylmethyl)(thiophen-3-ylmethyl){[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amine
N-[(4,6-dimethylpyridin-2-yl)methyl]-1-(2-methoxyethyl)-N-methylpiperidine-4-carboxamide
1-[(1R,5R)-6-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
(2S,4R)-4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
N,N-diethyl-5-{[methyl(2-phenylethyl)amino]methyl}-1,2-oxazole-3-carboxamide
2-[4-(pyridin-4-yl)piperidin-1-yl]quinoline
3-{2-[2-(2-cyclohexylpyrimidin-5-yl)-1H-imidazol-1-yl]ethyl}-1,3-oxazolidin-2-one
2-[5-(1H-indazol-1-ylmethyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl]acetic acid
1-(4-{[(dicyclopropylmethyl)amino]methyl}-2-methoxyphenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
3-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-1-[4-(propylsulfanyl)phenyl]urea
N-benzyl-N-ethyl-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
1-(2,3,6-trimethylquinoline-4-carbonyl)azetidin-3-ol
1-[3-(3-fluoro-4-phenylbenzoyl)piperidine-1-carbonyl]cyclopropane-1-carboxamide
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-3-(4H-1,2,4-triazol-4-yl)benzamide
N-(1-benzylpyrrolidin-3-yl)-3-[1-(1H-indol-3-ylmethyl)piperidin-4-yl]propanamide
1-(4-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperazin-1-yl)ethan-1-one
(3S,4R)-4-(3-methylthiophen-2-yl)-1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-3-ol
N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
N-(2-methoxyphenyl)-6-[(3-phenyl-1H-pyrazol-4-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl](1-phenoxypropan-2-yl)amine
4-(4-tert-butylbenzoyl)-1-methylpiperazine-2-carboxylic acid
(1S,5R)-6-[2-(1H-imidazol-2-yl)benzoyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-({5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}methyl)-3,5-dimethyl-1,4-dihydropyridin-4-one
N-[(2-chloropyridin-3-yl)methyl]-N-methyl-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
2-acetyl-8-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-[4-(trifluoromethyl)pyrimidin-2-yl]isoquinoline
ethyl 2-{[3-(6-methoxynaphthalene-2-carbonyl)piperidine-1-carbonyl]amino}acetate
6-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-benzyl-N-methyl-2-{4-[2-(2-oxopyrrolidin-1-yl)acetyl]morpholin-3-yl}acetamide
N-cyclopentyl-2-ethyl-N-[(5-methylthiophen-2-yl)methyl]pyrimidine-5-carboxamide
1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}cyclopropane-1-carboxamide
9-({1-[4-(propan-2-yl)phenyl]-1H-pyrazol-4-yl}methyl)-1,4,9-triazaspiro[5.5]undecan-5-one
1-(pyridin-3-ylmethyl)-4-(thiomorpholine-4-carbonyl)pyrrolidin-2-one
6-methoxy-3-({methyl[(3-methyloxetan-3-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
(1R,3S)-3-methoxy-3-methyl-7-[2-(methylsulfanyl)pyridine-3-carbonyl]-7-azaspiro[3.5]nonan-1-ol
2-{3-[4-(2-amino-6-methylpyrimidin-4-yl)piperazine-1-carbonyl]piperidin-1-yl}acetamide
3-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyridin-2-ol
N-methyl-N-(1H-pyrazol-5-ylmethyl)-2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
5-({1-tert-butyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-2-methyl-1,3-thiazole
2-({4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)pyridine
ethyl[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl][3-(methylsulfanyl)butyl]amine
1-(3-methoxyphenyl)-4-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperazin-2-one
4-{[2-(2,1,3-benzoxadiazol-4-yl)-1H-imidazol-1-yl]methyl}-1-ethylpyrrolidin-2-one
N-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
N-(oxan-4-yl)-3-(piperidin-3-yl)benzamide
4-{1-[2-chloro-5-(1H-pyrazol-1-yl)benzoyl]azetidin-3-yl}pyridine
2-[4-(1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)piperazin-1-yl]benzonitrile
(2S,4S)-4-amino-1-methyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}pyrrolidine-2-carboxamide