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methyl 3-(cyclobutylmethoxy)-5-(2-methyl-3-oxopiperazine-1-carbonyl)benzoate
3-(4-methoxyphenyl)-1-[2-(morpholine-4-carbonyl)piperazin-1-yl]propan-1-one
1-(1-methyl-1H-pyrrol-2-yl)-2-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}ethane-1,2-dione
4-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-7-methyl-3,4-dihydro-2H-1,4-benzothiazin-3-one
6-[2-(furan-2-yl)pyrrolidine-1-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
4-[(3,5-dimethoxyphenyl)methyl]-3-[2-(1,2-oxazinan-2-yl)-2-oxoethyl]piperazin-2-one
2-(piperazin-1-yl)-N-{[1-(propan-2-yl)piperidin-4-yl]methyl}acetamide
1-[(4-ethylphenyl)methyl]-3-(2-methoxyethyl)-5-(4H-1,2,4-triazol-4-ylmethyl)-1H-1,2,4-triazole
1-[3-chloro-4-(1H-imidazol-1-yl)phenyl]-3-[2-(dimethylamino)ethyl]-3-methylurea
ethyl 5-(morpholin-4-ylmethyl)-1-(pyridin-2-yl)-1H-pyrazole-4-carboxylate
1-[(2-methoxyphenyl)methyl]-6-oxo-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidine-3-carboxamide
4-(4-fluoro-3-methylbenzoyl)-1-(3-methoxyphenyl)piperazin-2-one
1-ethyl-8-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-4-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}-1,3-thiazol-2-amine
N,1,3-trimethyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazole-4-carboxamide
4-oxo-N-[2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-4H-chromene-2-carboxamide
2-[(1-butyl-1H-1,2,4-triazol-5-yl)methyl]-5,6-dimethyl-2,3-dihydropyridazin-3-one
7-[2-(4-methylphenoxymethyl)furan-3-carbonyl]-2-oxa-7-azaspiro[4.5]decane
N-(2,3-dihydro-1H-inden-2-yl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-methyl-1,2-dihydroquinoxalin-2-one
N-methyl-N-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1,2,3,4-tetrahydronaphthalen-1-amine
2-(2-chloro-4-{[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]methyl}phenoxy)propanoic acid
3-{[(3-cyano-4-methylphenyl)carbamoyl]amino}-N-cyclohexylpropanamide
4-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-2-(pyridin-3-yl)morpholine
N-(2-ethylphenyl)-2-[4-(morpholin-4-yl)pentanamido]benzamide
(3S,4R)-1-[2-(dimethylamino)acetyl]-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
4-cyclobutyl-N-[2-(4-ethylpiperazin-1-yl)-2-methylpropyl]-6-methylpyrimidin-2-amine
2-[7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-6-methylpyridine-3-carbonitrile
3-[(1-methyl-1H-imidazol-2-yl)methyl]-1-[2-(propan-2-ylsulfanyl)phenyl]-3-propylurea
methyl 3-[(3S,4R)-4-(dimethylamino)-1-(2,2-diphenylethyl)piperidin-3-yl]propanoate
(4S,4aS,8aS)-4-phenyl-1-(thiophen-2-ylmethyl)-decahydroquinolin-4-ol
3-(3-methoxyphenoxymethyl)-1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidine
3-(1H-1,3-benzodiazol-2-yl)-1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]propan-1-one
N-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
5-[2-(1H-indol-3-yl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]-1-(pyrimidin-2-yl)piperidin-4-amine
1-{4-[1-(3-chlorophenyl)piperidin-4-yl]-6-hydroxy-1,4-diazepan-1-yl}ethan-1-one
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-4-(1H-pyrazol-1-yl)butan-1-one
2-ethoxy-1-[6-hydroxy-4-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-1,4-diazepan-1-yl]ethan-1-one
5-[2-(4-chlorophenyl)acetyl]-N-[(1-ethylpyrrolidin-2-yl)methyl]-1-(2-methoxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-ethyl-5-[methyl({[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl})amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carboxamide
5-[benzyl(methyl)amino]-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-methyl-5-(2-{pyrazolo[1,5-a]pyridin-7-yl}phenyl)-1,3,4-thiadiazole
3-{[(4,6-dimethylpyridin-2-yl)methyl](methyl)carbamoyl}-5-methoxybenzoic acid
3-[1-(furan-2-ylmethyl)-1H-pyrazol-5-yl]-1-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]urea
2-[4-(3,5-dimethyl-1-benzofuran-2-yl)-3-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-1-yl]acetic acid
1-ethyl-4-(5-propyl-1,2-oxazole-3-carbonyl)piperazin-2-one
1-(5-methoxyfuran-2-carbonyl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-2-(pyridin-3-yl)pyridine