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2-({[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}amino)-N-methylpyridine-3-carboxamide
3-(azocan-1-yl)-1-{4-[(pyrimidin-2-yl)amino]piperidin-1-yl}propan-1-one
ethyl 1-[3-(4-methoxyphenyl)-3-phenylpropanoyl]piperidine-4-carboxylate
(1R,3S)-3-(2-hydroxyethoxy)-7-{[3-(trifluoromethyl)phenyl]methyl}-7-azaspiro[3.5]nonan-1-ol
1-(4-fluoro-3-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)ethan-1-one
N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-1H-indole-5-carboxamide
4-(1-tert-butyl-1H-pyrazol-4-yl)-1-(2-phenylethyl)-1,2,3,6-tetrahydropyridine
1-[2-(furan-2-yl)azepan-1-yl]-2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
4-{1-[(2-chlorophenyl)methyl]-1H-imidazol-2-yl}-2,6-dimethoxyphenol
(3S)-1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-N,N-dimethylazepan-3-amine
1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine
1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-3-(1H-imidazol-2-yl)piperidine
4-(2,2-dimethylpropanoyl)-6-[(3-fluorophenyl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-1,5-dimethyl-1H-pyrazole-3-carboxamide
(1R,2S,6R,7S)-4-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-4-azatricyclo[5.2.2.02,6]undecane
(3R,4R)-1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
N-ethyl-N-[(2E)-3-phenylprop-2-en-1-yl]-2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]acetamide
1-{3-[5-(1-ethyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]propyl}piperidine-4-carboxamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1H-pyrazole-4-carboxamide
7-[3-(2-chlorophenyl)-5-methyl-1,2-oxazole-4-carbonyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-amino-4-(3,5-dimethoxyphenyl)-6-(5-methylfuran-2-yl)pyridine-3-carbonitrile
(2S)-4-methanesulfonyl-2-[(3,5,7-trimethyl-1H-indol-2-yl)formamido]butanoic acid
(3-phenylprop-2-yn-1-yl)(prop-2-en-1-yl){[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
1-{1-[3-cyclopropyl-1-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-4-methylpiperazine
1-[4-({3-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)phenyl]ethan-1-one
3-chloro-N-(2-methoxyethyl)-4-{[1-(piperidin-4-yl)piperidin-4-yl]oxy}benzamide
4-{furo[3,2-c]pyridin-4-yl}-1H-pyrrolo[2,3-b]pyridin-6-amine
N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)but-2-ynamide
3-[(4-cyanopiperidin-1-yl)sulfonyl]-N-(pyrrolidin-3-yl)benzamide
(1S,6R)-9-(2,3-difluoro-6-methoxybenzoyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
2-(1-{[1-(2,3-dimethylbenzoyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-amine
5-[(1-methyl-1H-imidazol-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
5-{[3-(2-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
3-[3-(3-aminoazetidin-1-yl)-3-oxopropyl]-3-benzyl-1-methyl-2,3-dihydro-1H-indol-2-one
1-benzyl-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]pyrrolidin-3-amine
N-ethyl-N-[2-(4-methylbenzenesulfonyl)ethyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
3,3-dimethyl-1-({5-[(3-methyl-1-benzofuran-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)urea
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidine
5-{[4-(4-methoxybenzoyl)piperazin-1-yl]methyl}-2-(methoxymethyl)pyrimidine
7-(3-chlorophenyl)-4-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-cyclopropanecarbonyl-8-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
N3-[2-(4-ethoxyphenyl)propan-2-yl]-N1,N1-dimethylpiperidine-1,3-dicarboxamide
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl][(2-methylphenyl)(pyridin-4-yl)methyl]amine
1-{5-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1H-pyrazol-3-yl}ethan-1-one
2-(3-{[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)amino]methyl}phenoxy)ethan-1-ol
2-(2-{1-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperidin-2-yl}ethyl)pyridine
8-(dimethyl-1,3-thiazole-5-carbonyl)-3-(2-ethylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)[(2E)-3-phenylprop-2-en-1-yl]amine