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1-[2-(1-methyl-1H-imidazol-2-yl)benzoyl]-2-(2-phenylethyl)piperidine
2-(propan-2-yl)-N-(2-propoxyethyl)pyrimidine-5-carboxamide
N-[(3,5-dimethoxyphenyl)methyl]-N-(1-methoxypropan-2-yl)thiophene-3-carboxamide
1-[3-(7-fluoro-1-methyl-1,2,3,4-tetrahydroisoquinolin-2-yl)-3-oxopropyl]-6-methyl-1,2-dihydropyridin-2-one
N-ethyl-4,5,6-trimethyl-2-oxo-N-[2-(phenylsulfanyl)ethyl]-1,2-dihydropyridine-3-carboxamide
3-(2-oxoimidazolidin-1-yl)-N-{2-[(trifluoromethyl)sulfanyl]ethyl}benzamide
5-chloro-2-hydroxy-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]benzamide
1,6-dimethyl-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{4-[(2-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}-1,3-thiazole-4-carboxamide
7-fluoro-1-(2-methylpropyl)-3-({[(2-phenyl-2H-1,2,3-triazol-4-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
2-chloro-N-[2-(morpholin-2-ylformamido)ethyl]benzamide
4-{2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetyl}-1-phenylpiperazin-2-one
(3S,5R)-N3-cyclopentyl-N5-(4-fluorophenyl)-1-(pyridin-4-ylmethyl)piperidine-3,5-dicarboxamide
9-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
4-[5-(methoxymethyl)furan-2-carbonyl]-1-(4-methoxyphenyl)-5-methylpiperazin-2-one
1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-3-(pyridin-3-yl)propan-1-one
N-{1-[4-(ethylamino)pyrimidin-2-yl]piperidin-4-yl}acetamide
4-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}morpholine
3-{[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}benzonitrile
2-methoxy-1-[1'-(1,2-oxazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
2-{[4-(3-methoxy-6-methylpyridin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}acetic acid
2,6-dimethyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)quinoline-4-carboxamide
(1R,5R)-6-(6-aminopyridine-3-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-(1-cyclopentyl-4-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperazin-2-yl)ethan-1-ol
2-[4-methyl-6-(pyrrolidine-1-carbonyl)-3,4-dihydro-2H-1,4-benzoxazin-2-yl]-1-(piperidin-1-yl)ethan-1-one
3-methyl-4-[5-(1-methyl-1H-1,3-benzodiazol-2-yl)furan-2-yl]-4H,5H,6H,7H-[1,2]oxazolo[5,4-b]pyridin-6-one
[(2-fluoro-4,5-dimethoxyphenyl)methyl](methyl){[1-(propan-2-yl)piperidin-3-yl]methyl}amine
N-cyclopropyl-2-{2-cyclopropyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}acetamide
(2S,4R)-1-(2,1,3-benzoxadiazol-4-ylmethyl)-N,N-diethyl-4-propanamidopyrrolidine-2-carboxamide
N,N-diethyl-5-methyl-4-{[2-(morpholin-4-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
1-[cyclohexyl(methyl)amino]-3-(2-methoxy-4-{[4-(2-methoxyethyl)piperazin-1-yl]methyl}phenoxy)propan-2-ol
2-methyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-[({[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amino)methyl]-1,2-dihydrophthalazin-1-one
3-({1,9-dimethyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}sulfonyl)benzonitrile
3-(1-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-1H-imidazol-2-yl)pyridine
{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}(methyl)(quinolin-8-ylmethyl)amine
1-[2-(2-butyl-2,5-dihydro-1H-pyrrol-1-yl)-2-oxoethyl]-1,2-dihydroquinoxalin-2-one
3-(adamantan-1-ylmethyl)-1-[3-(aminomethyl)phenyl]-3-(2-hydroxyethyl)urea
3-[cyclopropyl(1-methyl-1H-1,2,4-triazol-5-yl)methyl]-1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}urea
N-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-4-(2,4-dioxoimidazolidin-1-yl)benzamide
N-(2-{5,6-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-2-yl}ethyl)-3-(4-methyl-1,3-thiazol-5-yl)propanamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N,1-dimethyl-1H-pyrazole-5-carboxamide
N-(2-ethoxyethyl)-6-(4-methoxyphenyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-(oxolan-2-ylmethyl)-3-(propan-2-yl)-N-(pyridin-2-ylmethyl)-1H-pyrazole-5-carboxamide
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
1-(1-{1-[(2-chloro-6-fluoro-3-methylphenyl)methyl]piperidin-4-yl}ethyl)-4-methylpiperazine
1-(2-cyclohexylethyl)-3-hydroxy-3-{[methyl(thiophen-3-ylmethyl)amino]methyl}piperidin-2-one
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-(2-fluorobenzenesulfonyl)piperidine
1-(2-ethoxyethyl)-4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazine
[(6-chloroquinolin-2-yl)methyl](methyl)[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amine