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N-{2-chloro-4-[2-(1H-1,2,3,4-tetrazol-1-yl)acetamido]phenyl}-2,2-dimethylpropanamide
(4aR,7aS)-4-(1-tert-butyl-1H-pyrrole-3-carbonyl)-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
4-[(2-methoxyphenyl)methyl]-3-[2-(4-methoxypiperidin-1-yl)-2-oxoethyl]piperazin-2-one
2-({1,9-dimethyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}sulfonyl)benzonitrile
1-[3-(2-ethoxyethoxy)benzoyl]-4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
2-(4-methoxy-3-methylphenyl)-2-[4-(piperidine-1-carbonyl)piperidin-1-yl]acetic acid
3,6,7-trimethyl-N-[2-(methylsulfanyl)ethyl]-1-benzofuran-2-carboxamide
4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)-1-[(3,4-dimethoxyphenyl)methyl]piperidine
[(3R,4R)-1-[(3-fluoro-2-methylphenyl)methyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
2-[1-(1-methylpiperidin-4-yl)-4-[3-(trifluoromethyl)pyridin-2-yl]piperazin-2-yl]ethan-1-ol
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(2,5-dioxoimidazolidin-4-yl)-N-methylpropanamide
methyl 2-(5-{1-[(2-aminopyridin-3-yl)methyl]piperidin-4-yl}-1H-pyrazol-3-yl)acetate
N-(2-oxo-2,3-dihydro-1H-indol-5-yl)thiophene-3-carboxamide
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-amine
3-(4-methyl-1,3-thiazol-5-yl)-1-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]propan-1-one
2-[4-({2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)phenyl]acetic acid
6-[(3,5-dimethoxyphenyl)methoxy]-4-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(propan-2-yl)-1,4-diazepan-2-one
N-(1,3-benzothiazol-2-ylmethyl)-1-(cyclohexylmethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
4-[(1-ethyl-5-{[1,2,3,4]tetrazolo[1,5-a]pyridin-7-yl}-1H-1,2,4-triazol-3-yl)methyl]-1-methylpiperidine
1-(2-chlorophenyl)-4-({7-hydroxy-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)piperazin-2-one
4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine
N-methyl-N-[1-(4-methylpyrimidine-5-carbonyl)pyrrolidin-3-yl]acetamide
2-({[3-(1H-imidazol-1-yl)propyl]amino}methyl)-6-methylquinolin-4-ol
(3S,4S)-1-[3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanoyl]-4-propylpyrrolidine-3-carboxylic acid
N-{[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2-(1-methyl-1H-pyrrol-3-yl)acetamide
2-methoxy-1-[(1R,5S,6R)-6-{[methyl(prop-2-yn-1-yl)amino]methyl}-3-azabicyclo[3.1.0]hexan-3-yl]ethan-1-one
N-(2-methoxyethyl)-2,5,7-trimethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]quinoline-4-carboxamide
N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
2-[8-(2-methylpropyl)-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
(2S)-1-{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}pyrrolidine-2-carboxamide
({3-[2-(1-cyclohexanecarbonylpiperidin-2-yl)ethoxy]phenyl}methyl)(methyl)(quinolin-8-ylmethyl)amine
N-(2-{1-[(3-methyl-1H-indol-2-yl)methyl]piperidin-3-yl}ethyl)methanesulfonamide
2-(5-oxo-5,6-dihydro-1,6-naphthyridin-6-yl)-N-(oxolan-2-ylmethyl)acetamide
N-cyclopropyl-3-[2-(4-fluorophenoxy)ethyl]benzamide
N-[(1-methylpiperidin-3-yl)methyl]-1,1-dioxo-N-(2-phenylethyl)-1λ6-thiane-4-carboxamide
3-(benzenesulfonyl)-1-[4-(1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
1-(2,1,3-benzoxadiazol-5-ylmethyl)-N-benzyl-N-methylpiperidin-3-amine
[3-(3-methoxypropyl)-1-[3-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl]methanol
6-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-indole
(5-{[({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)amino]methyl}furan-2-yl)methanol
3-(3,4-difluorophenyl)-N-(1,4-dioxan-2-ylmethyl)propanamide
4-({1-[(1-cyclopentyl-1H-imidazol-5-yl)methyl]piperidin-2-yl}methyl)morpholine
4-{4-[(3S,4S)-3,4-bis(hydroxymethyl)pyrrolidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
9-methoxy-4-(6-methylpyridazin-3-yl)-7-(quinolin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-(4-chlorophenyl)-1-{1-[4-(furan-2-yl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}piperidin-4-ol
2-(1-propylpiperidin-4-yl)-1-[2-(pyridin-2-yl)piperidin-1-yl]ethan-1-one
[(3S,5R)-1-[2-chloro-5-(1H-pyrazol-1-yl)benzoyl]-5-[(dimethylamino)methyl]piperidin-3-yl]methanol
1-(cyclohex-1-en-1-ylmethyl)-3-{1-[(2-methoxyphenyl)methyl]-1H-pyrazol-5-yl}urea
N-(1-benzothiophen-2-ylmethyl)-N,1-dimethyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-3-ethyl-5-methyl-1,2-oxazole-4-carboxamide