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methyl 4-({5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}carbamoyl)benzoate
2-[(2H-1,3-benzodioxol-4-ylmethyl)(methyl)amino]-1-(4-hydroxyphenyl)ethan-1-one
2-methoxy-1-{4-[4-(4-methyl-1,4-diazepane-1-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one
(1R,2R)-N-methyl-2-phenyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}cyclopropane-1-carboxamide
N-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-[3-(4-benzylpiperazin-1-yl)-3-oxopropyl]-N,N-dimethylpiperidine-1-carboxamide
3-tert-butyl-1-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]urea
2-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-1,3-thiazole-4-carboxamide
(4aS,7aR)-1-(6-aminopyridine-3-carbonyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2,2-dimethyl-1-(thiophen-2-yl)cyclopropane-1-carboxamide
4-{2-[1-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)piperidin-2-yl]ethyl}phenol
2-{1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]azetidin-3-yl}pyridine
1-methyl-3-(naphthalen-2-ylmethyl)-8-{[2-(trifluoromethyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(diphenylmethyl)-2-(1-methyl-1H-imidazol-2-yl)-1H-imidazole
2-[(3S,4R)-4-amino-1-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}pyrrolidin-3-yl]ethan-1-ol
2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(6-methylpyridin-2-yl)ethyl]acetamide
N-cyclobutyl-7-fluoro-2-methylquinoline-4-carboxamide
4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)-N-[1-(pyridin-3-yl)propan-2-yl]pyrimidine-5-carboxamide
2-(ethanesulfonyl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decane
1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-3-(naphthalene-2-carbonyl)piperidine
2-[3-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]pyridine
N-{[1-(3-carbamoylpropanoyl)piperidin-3-yl]methyl}naphthalene-1-carboxamide
7-[(5-chlorothiophen-2-yl)sulfonyl]-2-oxa-7-azaspiro[4.5]decane
7-[(2-fluorophenyl)methyl]-2-(4-methyl-1H-imidazole-2-carbonyl)-2,7-diazaspiro[4.5]decane
N-[1-(1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]acetamide
1-(2,2-diphenylethyl)-3-(1,3,4-thiadiazol-2-yl)urea
5-[5-(ethylsulfanyl)thiophene-2-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
(3aS,6aR)-5-(2-aminopyrimidin-4-yl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
methyl 6-[(2-fluoro-5-methoxyphenyl)methyl]-2-[methyl(2-methylpropyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
8-[(2-chloro-4-fluorophenyl)methyl]-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[(4-benzylpiperazin-1-yl)methyl]-N-(prop-2-en-1-yl)-1,3-oxazole-4-carboxamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(dimethylamino)ethyl]-N-{[8-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}propanamide
3,4-dimethyl-N-[(5-methylpyrazin-2-yl)methyl]-5-sulfamoylbenzamide
N-[2-(3-methylthiophen-2-yl)ethyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
1-(1'-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)ethan-1-one
(4aS,8aR)-6-[2-(2,3-dimethylphenoxy)ethyl]-1-(4-hydroxybutyl)-decahydro-1,6-naphthyridin-2-one
N-[2-(1H-imidazol-1-yl)propyl]-6-methoxy-3-methyl-1-benzofuran-2-carboxamide
4-{[2-(pyrrolidin-1-ylmethyl)piperidin-1-yl]methyl}-1H-indole
(3S,4R)-4-(3-methoxyphenyl)-1-(6-oxo-1,6-dihydropyridine-3-carbonyl)pyrrolidine-3-carboxylic acid
2-(5-{[(cyclopropylmethyl)sulfanyl]methyl}-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-1-yl)pyridine
5-{[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]methyl}-N-methyl-1,2,4-oxadiazole-3-carboxamide
N-methyl-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(thiophen-2-ylmethyl)butanamide
methyl 4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-5-methylthieno[2,3-d]pyrimidine-6-carboxylate
4-{2-[1-(3-chloro-4-fluorobenzoyl)piperidin-2-yl]ethyl}morpholine
7-[(2-fluorophenyl)methyl]-2-(1,3-thiazol-2-yl)-2,7-diazaspiro[4.5]decane
1-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
1-cyclopentyl-4-(5,6,7,8-tetrahydro-1,6-naphthyridine-6-carbonyl)pyrrolidin-2-one
2-methyl-8-(5-propyl-1,3,4-oxadiazol-2-yl)-2,8-diazaspiro[5.5]undecane
(3R,4S)-4-cyclopropyl-1-[2-(morpholin-4-yl)benzoyl]pyrrolidin-3-amine
1-{1-[(3-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-phenylpiperazine