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N-(1-{1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
8-(7-chloroquinolin-4-yl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
6-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)pyridine-2-carbonitrile
N-(1-benzoylpiperidin-3-yl)-4-(4-chlorophenyl)butanamide
1-[2-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-2-oxoethyl]azepan-2-one
3-[2-(2-hydroxyphenyl)ethyl]-4-(thiophen-2-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[2-(pyridin-2-yl)pyrrolidin-1-yl]-2-(thiophen-2-yl)ethan-1-one
(1S,5R)-6-(cyclopropylmethyl)-3-(5-phenylpentanoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(2H-1,3-benzodioxol-4-ylmethyl)[(2-ethoxyphenyl)methyl]ethylamine
1-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1H-pyrrol-1-yl)propan-1-one
1,6-dimethyl-N-[1-(4-methylpyridin-2-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(2-{[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
5-methyl-5-(4-methylpent-3-en-1-yl)-1-[2-(1,3-thiazol-4-yl)ethyl]piperidin-2-one
4-benzoyl-1-(3-methoxyphenyl)-6-methylpiperazin-2-one
ethyl 1-{1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}piperidine-3-carboxylate
2-(1H-indazol-3-yl)-1-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]ethan-1-one
3-cyclopentyl-5-[2-(3,4-dimethoxyphenyl)ethyl]-1-methyl-1H-1,2,4-triazole
N-methyl-2-(4-methyl-1H-pyrazol-1-yl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]propanamide
5-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-(2-{[methyl(propyl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)propan-1-one
N-{[7-fluoro-5-(3-fluoro-4-methylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,2-dimethyloxane-4-carboxamide
N-{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-9H-fluoren-9-amine
2-(2,6-dichlorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-1-yl]ethan-1-one
2-(dimethylamino)-2-(3-methylphenyl)-N-[(5-methylpyrazin-2-yl)methyl]acetamide
N-[4-({4-[(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)phenyl]acetamide
N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-1,3-thiazole-4-carboxamide
5-(1-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}pyrrolidin-2-yl)-3-methyl-1,2-oxazole
N-[(4-fluorophenyl)methyl]-N-methyl-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
2,3-dimethyl-6-[2-(1H-pyrazol-1-yl)butanoyl]-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
N-[(4-hydroxy-1-methylpiperidin-4-yl)methyl]-1-[(3-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
N-[3-(ethylcarbamoyl)-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-1H-1,2,4-triazole-5-carboxamide
2-(1-{1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]piperidin-3-yl}-N-methylformamido)-N-methylacetamide
2-cyclopentyl-N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)acetamide
N-[(3R,4S)-1-[(2-aminopyrimidin-5-yl)methyl]-4-cyclopropylpyrrolidin-3-yl]-1-(methoxymethyl)cyclobutane-1-carboxamide
(3R,4R)-4-ethyl-1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3,4-diol
methyl (2S,4R)-4-[2-(dimethyl-1,3-thiazol-5-yl)acetamido]-1-methylpyrrolidine-2-carboxylate
1-(3-methoxyphenyl)-6-methyl-4-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperazin-2-one
2-{[4-(2,4-dimethoxy-3-methylphenyl)-1H-1,2,3-triazol-1-yl]methyl}-3,4-dihydroquinazolin-4-one
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5-oxo-1-phenyl-2,5-dihydro-1H-pyrazole-3-carboxamide
2-(6-methoxypyridin-3-yl)-5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridine
3-{2-oxo-2-[3-(4-phenylbenzoyl)piperidin-1-yl]ethyl}-1,3-thiazolidine-2,4-dione
[1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-3-yl]methanamine
N-(2,3-dihydro-1H-inden-2-yl)-2-{4-[(2-methylphenyl)methyl]morpholin-3-yl}acetamide
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-6-methyl-2-(piperidin-1-yl)pyrimidin-4-amine
8-(3-oxo-1,2,3,4-tetrahydroquinoxaline-6-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-(4-{[4-(cyclohexylmethyl)-5-oxo-1,4-diazepan-1-yl]methyl}phenyl)acetamide
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-2-(methylamino)-1,3-thiazole-4-carboxamide
3-{2-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-3,4-dihydroquinazolin-4-one
N-[3-(furan-2-yl)-3-phenylpropyl]-2-[1-(2-methoxyethyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]acetamide
N-[(3-methyl-1-benzofuran-2-yl)methyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide