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N-[2-(4-fluorophenyl)ethyl]-2-[(3S,4S)-3-hydroxy-4-(propan-2-yloxy)pyrrolidin-1-yl]acetamide
3-(2-methoxyethyl)-8-(2-methylpropyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-chloro-5-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-1,2-dihydropyridin-2-one
9-[(2,2-dimethyloxan-4-yl)methyl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-cyclopropyl-N-[1-(2-fluorophenyl)piperidin-4-yl]-6-oxopiperidine-3-carboxamide
N-[2-(2-ethoxyphenyl)ethyl]-5-ethyl-1,3,4-oxadiazol-2-amine
4-[1-(morpholin-2-ylmethyl)-1H-1,2,3-triazol-4-yl]quinoline
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-methylthiophene-2-sulfonamide
2-{5-[1-(2-chloropyridine-4-carbonyl)piperidin-2-yl]-1,2,3,6-tetrahydropyridin-1-yl}ethan-1-ol
(3S,4S)-4-cyclopropyl-1-[(1-ethyl-1H-pyrazol-3-yl)methyl]pyrrolidine-3-carboxylic acid
(3S,4R)-4-(3-fluorophenyl)-1-[1-(furan-2-ylmethyl)piperidin-4-yl]pyrrolidine-3-carboxylic acid
2-cyclopropyl-N-{1-[(cyclopropylcarbamoyl)methyl]piperidin-4-yl}-6-oxo-1,6-dihydropyrimidine-5-carboxamide
8-[3-(pyridin-4-yl)propanoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-methoxy-6-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridine
4-(9H-purin-6-yl)-N-(pyridin-4-ylmethyl)piperazine-2-carboxamide
ethyl 2-[1-(5-methoxyfuran-2-carbonyl)piperidin-2-yl]acetate
(2S)-N-[3-(1H-indol-2-yl)phenyl]-1-(pyridin-2-ylmethyl)pyrrolidine-2-carboxamide
methyl 2-[4-({[(1-phenylcyclopentyl)methyl]carbamoyl}amino)phenoxy]acetate
7-fluoro-3-methyl-N-[3-(1H-pyrazol-1-yl)propyl]-1-benzofuran-2-carboxamide
5-(2-{[(2S)-2,3-dihydroxypropyl]amino}pyrimidin-4-yl)-2-ethoxybenzoic acid
(2R,3R,6R)-5-[(2-ethoxyphenyl)methyl]-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(3R,4R)-1-[(4-fluoro-3-methoxyphenyl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol
N,N-dimethyl-6-(1-methyl-1H-indol-2-yl)pyridine-2-carboxamide
4-{2-[1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)piperidin-2-yl]ethyl}phenol
4-{1-benzyl-5-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}morpholine
N-ethyl-2-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)pyridine-3-carboxamide
N-(furan-3-ylmethyl)-N-methyl-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
N-[2-({4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}methyl)quinolin-6-yl]acetamide
3-(2-oxopiperidin-1-yl)-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)propanamide
4-benzyl-3-{1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
7-(cyclobutylmethyl)-2-(2,4-dimethyl-6-oxo-1,6-dihydropyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-acetyl-N-[3-(3-phenylpropoxy)phenyl]piperazine-1-carboxamide
2-[6-(1-hydroxyethyl)pyridin-2-yl]benzamide
5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1H-pyrazole-3-carboxamide
2-[(3,4-difluorophenyl)methyl]-8-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
7-(2-oxo-1,3-oxazolidin-3-yl)-4-(1,3-thiazol-2-yl)-1,2,3,4-tetrahydroquinolin-2-one
1-(4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
N-[3-(4-methoxyphenyl)propyl]-6-(methylamino)pyridine-3-carboxamide
3-chloro-N-(2-hydroxyethyl)-5-methoxy-N-[(2E)-3-phenylprop-2-en-1-yl]benzamide
N-methyl-2-(4-methylphenoxymethyl)-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}furan-3-carboxamide
6-cyclopentyl-1-methyl-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-3-methyl-1H-pyrazole-5-carboxamide
6-(2H-1,3-benzodioxol-5-ylmethyl)-3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
5-ethyl-N4-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-6-methylpyrimidine-2,4-diamine
5-(4-fluorophenyl)-N-methyl-N-(oxan-2-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
2-{[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}benzonitrile
2,5-dimethyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-(4-cyano-2-ethylphenyl)-4-(1H-pyrrole-2-carbonyl)piperazine-1-carboxamide
6-(difluoromethyl)-2-(4-{[4-(2-methoxyethyl)piperazin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
1-[(2S)-2-amino-2-benzylpropanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one