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N-[(2R,3R)-1'-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-2-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopropyl-4-(1H-pyrazol-3-yl)benzamide
3-(oxolan-3-yl)-5-[3-(thiophen-3-yl)-1H-pyrazol-5-yl]-1,2,4-oxadiazole
7-[4-methyl-3-(1H-pyrrol-1-yl)benzoyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
N-(2-hydroxy-3-methoxypropyl)-2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
{1-ethyl-5-[(6-methoxy-2H-chromen-3-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(4,4,4-trifluorobutyl)-2,7-diazaspiro[4.5]decan-6-one
N-cyclopropyl-N-{[7-fluoro-2-(morpholin-4-yl)quinolin-3-yl]methyl}-2-(thiophen-3-yl)acetamide
4-methoxy-N-{[1-(oxane-4-carbonyl)piperidin-3-yl]methyl}benzene-1-sulfonamide
1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
8-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]benzamide
N-[2-(4-fluorophenyl)ethyl]-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
N-(furan-2-ylmethyl)-3-hydroxy-N-(1-hydroxybutan-2-yl)pyridine-2-carboxamide
4-(5-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}furan-2-carbonyl)morpholine
2-[4-(3-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]pyridin-4-amine
3-[2-({2-methylthieno[2,3-d]pyrimidin-4-yl}amino)ethyl]-1,3-oxazinan-2-one
2-({[2-amino-6-(cyclopropylamino)pyrimidin-4-yl](methyl)amino}methyl)-3H,4H-thieno[3,2-d]pyrimidin-4-one
3-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}pyrrolidin-2-yl)-5-(propan-2-yl)-1,2-oxazole
1-[3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propyl]-5-oxopyrrolidine-3-carboxylic acid
N-{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}-N-methyloxan-4-amine
1'-(morpholine-4-sulfonyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
1-{5-[(3,3-difluoropiperidin-1-yl)methyl]imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-methyl-1,4-diazepane
4-hydroxy-N-(3-methyl-1,2,4-thiadiazol-5-yl)-4-[3-(trifluoromethyl)phenyl]piperidine-1-carboxamide
3-[(3-aminopyrrolidin-1-yl)sulfonyl]-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]benzamide
(3R,5S)-1-benzyl-N3-(4-fluorophenyl)-N5-(naphthalen-1-ylmethyl)piperidine-3,5-dicarboxamide
1,3-dimethyl-6-[4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1-{[(1-benzylpyrrolidin-3-yl)amino]methyl}cyclopentyl)methanol
methyl 5-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-[1-(azepan-1-yl)-2-methylpropan-2-yl]-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
1-[4-(propan-2-yl)piperazin-1-yl]-3-{[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}propan-1-one
4-[(1S,5R)-7-oxo-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]oxane-4-carbonitrile
3-[methyl({[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl})amino]propane-1,2-diol
N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
1-[3-(pyridin-3-yl)propanoyl]-4-(pyrimidin-2-yl)piperazine-2-carboxylic acid
(3S,9aR)-8-(3-chlorobenzoyl)-3-(1H-imidazol-4-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[2-(3-{[4-(3-chlorophenyl)piperazin-1-yl]methyl}phenoxy)propyl]-2-methyl-1,3-thiazole-4-carboxamide
1-cyclobutyl-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
2-hydroxy-N-{2-[4-(1-methylpiperidin-4-yl)morpholin-2-yl]ethyl}benzamide
N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyrazolo[1,5-a]pyridine-7-carboxamide
1-[(2-methoxyphenyl)methyl]-3-[3-(4-methylpiperidine-1-carbonyl)phenyl]urea
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N,1-dimethyl-1H-pyrazole-5-carboxamide
1-(6-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}pyridin-3-yl)ethan-1-one
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
1-(3-cyano-4-ethoxyphenyl)-3-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
N-[(3S,4R)-1-(5-ethyl-1,3,4-thiadiazol-2-yl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
(2-{2-[(2-chlorophenyl)methyl]morpholin-4-yl}-2-oxoethyl)urea
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({[(4-methyl-1,3-thiazol-2-yl)methyl]amino}methyl)piperidin-2-one
{1-[4-methyl-2-(pyridin-3-yl)pyrimidine-5-carbonyl]-3-propylpiperidin-3-yl}methanol