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3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-{[5-(hydroxymethyl)furan-2-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[1-(5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carbonyl)pyrrolidin-2-yl]pyridine
2-(2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamido)-N-methylacetamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-[3-(thiophen-3-yl)propanoyl]piperidin-3-yl]propanoic acid
2-[(3S,4S)-3-[ethyl(methyl)amino]-4-hydroxypyrrolidin-1-yl]-2-oxo-S-(thiophen-2-yl)ethane-1-sulfonamido
1-{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidine-2-carboxamide
8-(4-carboxyquinolin-2-yl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(1-{[1-(4-methylpiperidine-4-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-amine
5-(2-chloro-4-fluorophenoxymethyl)-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
2-(4-methoxy-2,3-dimethylphenyl)-4-{[2-(2-methoxyphenyl)pyrrolidin-1-yl]methyl}-5-methyl-1,3-oxazole
1-[1-(2-ethoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carbonyl]piperidine-4-carboxamide
2-(3-chlorophenyl)-4-[4-(thiophen-3-ylmethyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
2-ethoxy-5-[2-({[4-(methylsulfanyl)phenyl]methyl}amino)pyrimidin-4-yl]benzoic acid
5-({8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)-1-methyl-1H-imidazole
N-[(3-chlorophenyl)methyl]-3-{1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl}propanamide
3-({2-[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-methyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}acetamide
2-(dimethylamino)-N-methyl-N-(1,2-oxazol-3-ylmethyl)benzamide
(4aS,7aR)-1-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{2-[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-5-methyl-1H-1,3-benzodiazole
N-(3-hydroxy-2,2-dimethylpropyl)-4-{[2-(1H-indol-3-yl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
3-ethyl-1-(2-phenylethyl)-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[3-(2-fluorophenoxymethyl)piperidine-1-carbonyl]benzonitrile
5-[2-(furan-2-yl)pyrrolidine-1-carbonyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
3-({[2-(benzylsulfanyl)ethyl]amino}methyl)piperidin-3-ol
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
4-(6-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl)thiomorpholine
N-(2,3-dihydro-1H-inden-2-yl)-N-methyl-4-(4-methylpiperazin-1-yl)benzamide
2-methyl-4-[(5-methyl-2-phenyl-1H-imidazol-4-yl)methyl]-1-(propan-2-yl)piperazine
4-[4-({[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl)amino}methyl)phenyl]-2-methylbut-3-yn-2-ol
3-(azepane-1-carbonyl)-1-ethyl-N-[3-(morpholin-4-yl)propyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-chloro-4-[(1-cycloheptylpiperidin-4-yl)oxy]-N-[2-(dimethylamino)ethyl]benzamide
3-(4-methoxyphenoxymethyl)-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperidine
ethyl 3-benzyl-1-{[4-(methylsulfanyl)phenyl]carbamoyl}piperidine-3-carboxylate
(1R,5R)-6-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
N-[(1R,2S)-2-phenylcyclopropyl]-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-(4-fluorophenyl)-4-(1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-yl)piperazine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-3,3-dimethylcyclohexan-1-amine
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-3-(5-methyl-1H-1,2,4-triazol-3-yl)propanamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-(1-propylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
(3S,9aR)-3-(1H-imidazol-4-ylmethyl)-8-(3-methoxybenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-5-(hydroxymethyl)furan-2-carboxamide
(1R,9S)-5-amino-3-(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
N-(2,1,3-benzoxadiazol-5-ylmethyl)-5-oxo-1-phenyl-2,5-dihydro-1H-pyrazole-3-carboxamide
2-(3-{2-[3-(dimethylamino)pyrrolidin-1-yl]ethyl}-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl)pyridine-3-carbonitrile
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
7-(3-chlorophenyl)-4-(1-methylpiperidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-methyl-2-oxo-N-{[1-(phenoxymethyl)cyclopropyl]methyl}-1,2-dihydroquinoline-4-carboxamide
1-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(methylamino)ethan-1-one