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4,6-dimethyl-N-[3-methyl-1-(pyridin-3-yl)butyl]pyrimidin-2-amine
2-(2H-1,3-benzodioxol-5-yloxy)-1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]ethan-1-one
N-[(3S,4R)-4-hydroxyoxolan-3-yl]-N-methyl-2-(4-methylphenyl)quinoline-4-carboxamide
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-3-(pyridin-2-yl)-1H-pyrazole-5-carboxamide
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
1-[2-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidine-1-carbonyl)phenyl]ethan-1-one
2-{2-oxo-4-[3-(1H-pyrazol-1-yl)benzoyl]piperazin-1-yl}benzonitrile
2-(2,3-difluorophenyl)-1-[4-(hydroxymethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]ethan-1-one
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-(1H-indole-6-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(3R,9aR)-8-benzyl-3-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)-1,8-naphthyridine-2-carboxamide
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
1-[1-(2-ethoxyethyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-methyl-N-(oxan-2-ylmethyl)-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
N,N-dimethyl-2-[4-(5-{[(2-methylphenyl)carbamoyl]amino}-1H-pyrazol-1-yl)piperidin-1-yl]acetamide
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
2-methoxy-3-[4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]pyrazine
N-(2,4-dimethoxyphenyl)-3-[(3,4-dimethylphenyl)amino]piperidine-1-carboxamide
2-[({1-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}oxy)methyl]pyridine
4-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
1'-(2-chloro-5-fluorobenzoyl)-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
6-ethoxy-3-{[methyl(1H-pyrazol-3-ylmethyl)amino]methyl}-1,2-dihydroquinolin-2-one
1-(6-hydroxy-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1,4-diazepan-1-yl)-2-(2H-1,2,3,4-tetrazol-2-yl)ethan-1-one
[(4-fluorophenyl)methyl]({[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl})amine
2-({4-oxo-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}sulfonyl)benzonitrile
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazol-5-yl]-1H-1,2,4-triazole
N'-(3-chloro-4-fluorophenyl)-N-[2-(1-methylpyrrolidin-2-yl)ethyl]propanediamide
N-[1-(4-methoxyphenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]pyridazine-3-carboxamide
4-[4-(3-methoxyphenyl)benzoyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
3-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-3-methyl-1-[4-(1H-1,2,4-triazol-1-yl)phenyl]urea
N-methyl-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-{[3-(trifluoromethyl)phenyl]methyl}acetamide
9-(cyclopropylmethyl)-1-methyl-4-(pyrrolidine-1-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(dimethylamino)-N-(1H-indol-4-ylmethyl)-2-(3-methylphenyl)acetamide
5-{[(3S)-3-ethylmorpholin-4-yl]sulfonyl}-3-methyl-2,3-dihydro-1,3-benzoxazol-2-one
1-(2H-1,3-benzodioxol-5-yl)-3-methyl-5-[1-(1H-pyrrol-1-yl)ethyl]-1H-1,2,4-triazole
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(2,3-dimethylphenoxy)-2-methylpropanamide
N-ethyl-3-(4-methoxyphenyl)-3-phenylpropanamide
N-[2-(dimethylamino)-2-(thiophen-2-yl)ethyl]-5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(4-methylpiperidine-4-carbonyl)piperidin-3-amine
1-{4-[methyl({[1-(piperidin-1-yl)cyclohexyl]methyl})amino]piperidin-1-yl}ethan-1-one
6-methyl-N-[2-(4-phenylpyrimidin-2-yl)ethyl]imidazo[1,2-a]pyridine-2-carboxamide
1-phenyl-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}cyclohexane-1-carboxamide
2-(2-fluoro-3-methoxyphenyl)-1,3-thiazole
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
N-(oxolan-2-ylmethyl)-2-(pyridin-4-yl)-N-(thiophen-3-ylmethyl)acetamide
1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-3-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}urea
2-(3-phenylpropyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-{4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1,4-diazepan-1-yl}-N,N-dimethylacetamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]acetamide
N-({1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]pyrrolidin-3-yl}methyl)-6-methylpyridine-2-carboxamide