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N-[1-(3-hydroxyadamantan-1-yl)ethyl]-1-(7-methoxy-4-methylquinazolin-2-yl)piperidine-4-carboxamide
1-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethan-1-one
N-{5-[3-(1H-pyrazol-3-yl)phenyl]pyridin-2-yl}methanesulfonamide
N-(2-methylpropyl)-1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
3-{1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-N-(3-chloro-4-fluorophenyl)propanamide
1-{1-[(3-methoxyphenyl)methyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
4-(4-{3-[1-(dimethylamino)ethyl]phenyl}-1H-1,2,3-triazol-1-yl)butan-1-ol
1-[2-(cyclohexylsulfanyl)ethyl]-3-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)urea
4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}-N-[2-(pyridin-3-yloxy)ethyl]benzamide
4-({1-[(4-fluorophenyl)methyl]-5-(oxan-4-yl)-1H-1,2,4-triazol-3-yl}methyl)-1-methylpiperidine
3-(ethylsulfanyl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}propanamide
3-{1-[2-(azepan-1-yl)acetyl]piperidin-3-yl}-N-(5-chloro-2-methoxyphenyl)propanamide
N,1-dimethyl-N-[(3-methylthiophen-2-yl)methyl]-6-oxo-1,6-dihydropyridazine-3-carboxamide
4-{[({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amino]methyl}benzene-1-sulfonamide
(furan-2-ylmethyl)({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})(prop-2-en-1-yl)amine
6-ethyl-N,1,5-trimethyl-2-oxo-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1,2-dihydropyridine-3-carboxamide
(1-{[5-(methoxymethyl)furan-2-yl]methyl}-4-(3-phenylpropyl)piperidin-4-yl)methanol
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-(1H-1,2,4-triazol-5-yl)benzamide
3-[4-hydroxy-4-(hydroxymethyl)azepane-1-carbonyl]-6-phenyl-1,2-dihydropyridin-2-one
4-[2-(2-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}phenoxy)ethyl]morpholine
3-{3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}-1-(pyrrolidin-1-yl)propan-1-one
N,N-dimethyl-2-[(1S,5R)-6-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-methyl-2-(2-{[(1-methylpiperidin-3-yl)methyl]amino}-4-(morpholin-4-yl)pyrimidin-5-yl)propanoic acid
2,3-dimethyl-6-[4-(1H-pyrazol-5-yl)phenyl]pyridine
N-cyclohexyl-3-(hydroxymethyl)-3-(2-methoxyethyl)piperidine-1-carboxamide
1-benzyl-5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)pyrrolidin-2-one
5-[benzyl(methyl)amino]-2-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-2,3-dihydropyridazin-3-one
4-{1-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-imidazol-2-yl}pyridine
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-3-ethyl-1-methyl-1H-pyrazole-5-carboxamide
(4aR,7aS)-1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(1,2-oxazol-3-ylmethyl)-3-(pyrrolidin-1-yl)piperidine
2-chloro-4-({[2-(1-methylpyrrolidin-2-yl)ethyl]carbamoyl}amino)benzamide
N-{2-[1-(furan-2-ylmethyl)piperidin-3-yl]ethyl}-3-hydroxybenzamide
1-ethyl-N,4,6-trimethyl-N-{[3-(methylsulfanyl)phenyl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
(1S,5R)-6-methyl-3-{[2-methyl-5-(1,2-oxazol-5-yl)thiophen-3-yl]sulfonyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-({imidazo[1,2-a]pyridin-3-ylmethyl}(methyl)amino)acetic acid
6-[(3-methoxypropyl)amino]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1,3-benzothiazole-6-carboxamide
5-ethyl-N-[(3-methyl-7-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1,2-oxazole-3-carboxamide
[3-({1-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl}methyl)phenyl]methanol
N-[(2S,4R,6S)-2-benzyl-6-(2-butyl-1H-imidazol-4-yl)oxan-4-yl]acetamide
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}propanamide
1-{[2-(cyclopentyloxy)phenyl]methyl}-3-(pyrrolidin-1-yl)piperidine
N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
(1S,5R)-3-methyl-6-{[5-(2-methylpropyl)thiophen-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
1-[2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)acetyl]piperidine-3-carbonitrile
6-{1-[1-(propan-2-yl)piperidine-4-carbonyl]piperidin-3-yl}pyrimidin-4-ol
N-(2-ethoxyethyl)-5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole-3-carboxamide
3-[2-(pyridin-2-yl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione