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1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(3-hydroxyphenyl)ethan-1-one
(4aR,8aS)-1-(cyclohexylmethyl)-6-[(4-methoxy-3-methylphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
5-(4,4-difluoropiperidine-1-carbonyl)-2-(pyrrolidin-1-yl)pyrimidine
methyl (1R,3S,3aR,6aS)-1-butyl-5-ethyl-3-(1-methyl-1H-imidazol-5-yl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
1-[4-(aminomethyl)piperidin-1-yl]-4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]butan-1-one
2-[1-(2-hydroxyethyl)piperidin-3-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-hydroxy-1-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-methylbutan-1-one
2-[methyl(oxan-4-ylmethyl)amino]-2-(2-methylphenyl)acetic acid
(3S,9aR)-3-[(1R)-1-(benzyloxy)ethyl]-8-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-benzyl-1-[(2S)-2-methylbutyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-1-(2-methoxyacetyl)-N-methylpiperidine-3-carboxamide
(1R,3R)-N1-[6-(methoxymethyl)pyrimidin-4-yl]cyclopentane-1,3-diamine
4-[2-(1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidin-2-yl)ethyl]phenol
1-{2-[(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-3,3-dimethylurea
(3aR,6aS)-5-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
{2-[2-benzyl-4-(4-methylphenyl)-5-oxopiperazin-1-yl]-2-oxoethyl}urea
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-ethylacetamide
N'1-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]cyclopropane-1,1-dicarboxamide
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
4-benzyl-3-[1-(5-fluoropyrimidin-2-yl)piperidin-4-yl]-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{3-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-oxopropyl}pyrrolidin-2-one
2-(2-methoxy-4-methylphenoxymethyl)-N-[(5-methylpyrazin-2-yl)methyl]-1,3-oxazole-4-carboxamide
N-(2,3-dihydro-1H-inden-1-yl)-3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
methyl 2-[(5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-1H-pyrazol-4-yl)formamido]-4-(methylsulfanyl)butanoate
3-[(1-acetylpiperidin-4-yl)oxy]-4-methoxy-N-[(4-methylphenyl)methyl]benzamide
(4aR,7aS)-1-{2-[(2-hydroxyethyl)(methyl)amino]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-butyl-8-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-1-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperidin-4-amine
N-[2-(5-methoxy-1H-indol-3-yl)ethyl]-2-methylpyrido[2,3-d]pyrimidin-4-amine
2-(2-aminoethyl)-N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methylquinazolin-4-amine
N-(1-hydroxybutan-2-yl)-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
N-{1-[1-(2,6-dimethylhept-5-en-1-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-2,2-dimethylpropanamide
(4aS,8aR)-1-(3-hydroxypropyl)-6-(1H-indole-5-carbonyl)-decahydro-1,6-naphthyridin-2-one
(4aS,7aR)-1-(3-cyclopropyl-1,2-oxazole-5-carbonyl)-4-(2-methoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]-1H-indole-2-carboxamide
methyl 4-[(3-{[2-(2-methoxyphenoxy)acetamido]methyl}piperidin-1-yl)methyl]benzoate
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-3-(2-ethyl-5-oxopyrrolidin-2-yl)propanamide
3-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]pyridin-2-ol
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
1-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
N-[(3R,5S)-1-butanoyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]-3,5-difluoropyridine-2-carboxamide
1-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
N-[(5-methylfuran-2-yl)methyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-2-(morpholin-4-yl)pyridine-3-carboxamide
N-benzyl-N-ethyl-3-[3-(1H-imidazol-1-yl)pyrrolidin-1-yl]propanamide
ethyl 1-cyclobutanecarbonyl-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylate
5-ethyl-2-(1-{2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-imidazol-2-yl)pyridine
3-(1H-1,3-benzodiazol-1-yl)-N-[1-(pyridin-3-yl)propan-2-yl]propanamide
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-(6-methoxynaphthalene-2-carbonyl)piperidine