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1-[2-(furan-2-yl)ethyl]-2-[4-(1H-pyrazol-1-yl)phenyl]-1H-imidazole
1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-(2-ethyl-4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazole
3-(2-fluorophenyl)-1-(2-methoxyethyl)-3-[2-(4-methyl-3-phenylpiperazin-1-yl)-2-oxoethyl]pyrrolidine-2,5-dione
3-[(3R,4S)-4-(dimethylamino)-1-[(naphthalen-1-yl)carbamoyl]piperidin-3-yl]propanoic acid
(4S)-1-[(2-fluorophenyl)methyl]-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})amine
2-[4-(benzenesulfonyl)morpholin-3-yl]-N-(pyridin-2-ylmethyl)acetamide
1-[(1-{2-amino-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-4-yl)methyl]pyrrolidin-2-one
(1S,5R)-6-benzyl-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(2,5-dimethoxyphenyl)-N-(furan-2-ylmethyl)-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}acetamide
2-(dimethylamino)-N-(2-hydroxyethyl)-4-methyl-N-(1,3-thiazol-2-ylmethyl)pyrimidine-5-carboxamide
1-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
1-[5-(azepan-1-ylmethyl)-2-methoxyphenoxy]-3-[benzyl(methyl)amino]propan-2-ol
1-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-3-methyl-3-phenylpiperidine
1-(4-methylpiperazin-1-yl)-3-[5-(1,3-thiazol-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propan-1-one
methyl N-[(1-cyclohexylpiperidin-3-yl)methyl]-N-(pyridin-3-ylmethyl)carbamate
ethyl 3-benzyl-1-[(4-hydroxyphenyl)methyl]piperidine-3-carboxylate
2-({2-[1-(4-methoxyphenyl)-1H-imidazol-2-yl]-1H-imidazol-1-yl}methyl)pyridine
1-[(4-methylphenyl)methyl]-4-(2-propoxypropanoyl)piperazin-2-one
2-ethyl-8-(1-oxo-1,2,3,4-tetrahydroisoquinoline-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
[1-(5-chlorofuran-2-carbonyl)-3-(3-methoxypropyl)piperidin-3-yl]methanol
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine-2-carboxamide
1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-(2-methoxyethoxy)-N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}acetamide
2-[4-(1-methanesulfonylpyrrolidin-3-yl)piperidin-1-yl]pyrimidine
7-chloro-3-[2-(1-ethylpiperidin-4-yl)ethyl]-3,4-dihydroquinazolin-4-one
(2S,4R)-4-[4-(4-cyanobenzenesulfonamidomethyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine
5-(methoxymethyl)-N-[(3-methoxyphenyl)methyl]-N-methylfuran-2-carboxamide
5-methyl-1'-(3-phenyl-1,2-oxazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(2R,3R)-1'-[(3-fluorophenyl)methyl]-3-(pyrrolidin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-[(2,4-difluorophenyl)methyl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
1-[2-(dimethylamino)ethyl]-4-(5-methyl-4-phenyl-1H-imidazol-2-yl)pyrrolidin-2-one
N-(2,4-difluorophenyl)spiro[azepane-4,2'-chromene]-1-carboxamide
(1R,3S,4S)-3-hydroxy-N,4,7,7-tetramethyl-N-[3-(1H-pyrazol-1-yl)propyl]bicyclo[2.2.1]heptane-1-carboxamide
(4aS,8aR)-6-[(3E)-hex-3-enoyl]-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one
4-(2-methoxyethyl)-1-{[4-(2-methylphenyl)phenyl]methyl}-1,4-diazepan-5-one
1-(2,3-dimethylphenyl)-N-[3-(oxolan-3-yl)propyl]piperidin-4-amine
1-(cyclohexylmethyl)-N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-6-oxopiperidine-3-carboxamide
(1R,3R,5S)-8-(dimethyl-1,3-thiazole-5-carbonyl)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octane
4-(4-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-1-yl)-6-methylpyrimidin-2-amine
1-[2-(1H-imidazol-2-yl)benzoyl]-4-(1,3-thiazol-2-yl)piperazine
{4-[(6-methoxynaphthalen-2-yl)methyl]morpholin-3-yl}methanol
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-1,3-benzothiazole-6-carboxamide
1-(4-cyclopropanecarbonyl-1,4-diazepan-1-yl)-2-(dimethylamino)-2-(3-methylphenyl)ethan-1-one
1'-(6,8-dimethylquinolin-4-yl)-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
7-chloro-1-{3-methyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-9H-fluoren-9-one
N1,N1-dimethyl-N3-[3-(phenylsulfanyl)propyl]piperidine-1,3-dicarboxamide
3-[(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)methyl]pyridin-2-amine
1-[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]-2-(oxolan-2-yl)-1H-1,3-benzodiazole