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4-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]-6-[(3-methoxyphenyl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one
4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]piperidine
2-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-N-(2-methylpropyl)-2-oxoacetamide
3-{3-[3-(4-methoxy-2-methylbenzoyl)piperidin-1-yl]propyl}pyridine
N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-N-(pyridin-4-ylmethyl)furan-2-carboxamide
3-(4-chloro-1H-pyrazol-1-yl)-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]propan-1-one
[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl][(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amine
1-(2,5-dimethylfuran-3-carbonyl)-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
5-butyl-1-(3-phenylphenyl)-4-(1,3-thiazole-4-carbonyl)piperazin-2-one
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(morpholin-2-yl)ethan-1-one
[(3R,4R)-1-(5-fluoro-2-methylbenzoyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
(3aR,7aS)-2-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
2-methoxyethyl (1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxylate
1-[(3-ethyl-1,2-oxazol-5-yl)methyl]-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
methyl 4-chloro-1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1H-pyrazole-3-carboxylate
1-(4-ethylpiperazin-1-yl)-3-[1-(2-methoxyacetyl)piperidin-4-yl]propan-1-one
3-methoxy-2-methyl-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]benzamide
2-{1-cyclopentyl-4-[(2,6-dimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-{4-[(4,4-difluoropiperidin-1-yl)methyl]phenoxy}propanoic acid
3-{2-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
3-({[2-(azepan-1-yl)ethyl](ethyl)amino}methyl)-N-methylpyridin-2-amine
N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-1-phenyl-1H-1,2,3-triazole-5-carboxamide
1-{3-fluoro-6-methylimidazo[1,2-a]pyridine-2-carbonyl}-2-(4-fluorophenyl)piperidine
1-[(2-chlorophenyl)methyl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
4-{1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidin-4-yl}thiomorpholine
propyl 7-(1,2,3,4-tetrahydroquinoline-1-sulfonyl)-1,2,3,4-tetrahydroisoquinoline-2-carboxylate
N3-cyclohexyl-1-(2-methylpropyl)-4-oxo-N5-(pyridin-3-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
1-(2-{1-tert-butyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}-2-oxoethyl)-1,2,3,6-tetrahydropyridazine-3,6-dione
N-[2-(2-methoxynaphthalen-1-yl)ethyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
3-[(3R,4S)-1-[(4-ethylphenyl)carbamoyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
1-[4-(4-chlorophenyl)-4-hydroxypiperidin-1-yl]-2-[2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)-4-(thiophen-2-yl)phenoxy]ethan-1-one
N-[(1-methylpiperidin-3-yl)methyl]-2-propanoyl-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
N-[(2-aminopyrimidin-5-yl)methyl]-5-(3-fluorophenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
2-ethyl-1-{4-[4-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]piperidin-1-yl}butan-1-one
1-[(2,3-difluoro-6-methoxyphenyl)methyl]-N,N-dimethylazepan-4-amine
2-(6-methoxynaphthalen-2-yl)-4-(3-methoxypyridine-2-carbonyl)morpholine
3-(4-methoxyphenyl)-1-(4-methoxypiperidin-1-yl)-3-phenylpropan-1-one
4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-6-(pyrrolidin-1-yl)pyrimidin-2-amine
2-(dimethylamino)-7-[(2S)-2-(dimethylamino)-3-phenylpropanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-4-(oxolan-3-yl)-1H-1,2,3-triazole
2-{[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]methyl}-5-fluoro-3-methyl-1H-indole
(1S,5R)-1,3,3-trimethyl-6-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-6-azabicyclo[3.2.1]octane
4-[2-methyl-4-(2-methylpropyl)-3-oxopiperazine-1-carbonyl]benzene-1-sulfonamide
8-[3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanoyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-4-(1H-pyrazol-3-yl)benzamide
4-({5-[1-(5-ethyl-1,2,4-oxadiazol-3-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
N-[(5-ethylpyridin-2-yl)methyl]-3-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]propanamide
(4-{[methyl({[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl})amino]methyl}oxan-4-yl)methanol
4-(hydroxymethyl)-1-[1-methyl-3-(trifluoromethyl)-1H-thieno[2,3-c]pyrazole-5-carbonyl]piperidin-4-ol
N-[2-(dimethylamino)ethyl]-4-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}morpholine-2-carboxamide