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1-(furan-3-ylmethyl)-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
3-[4-(3-fluorophenoxy)piperidine-1-carbonyl]-4-methylpyridine
5-[1-(1H-1,3-benzodiazole-5-carbonyl)pyrrolidin-2-yl]-N-ethyl-N-methylthiophene-2-carboxamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(pyrimidin-2-yl)pyrrolidin-3-yl]methanol
N-[(3R,4S)-1-acetyl-4-cyclopropylpyrrolidin-3-yl]-3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propanamide
6-methoxy-2-{1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-1,2,3,4-tetrahydroisoquinoline
6-(5-methylthiophen-2-yl)-2-{2-oxa-7-azaspiro[4.5]decan-7-yl}pyridine-3-carboxylic acid
2-(1H-indol-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
ethyl 3-(2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamido)propanoate
[(3R,4R)-1-(2,4-difluorobenzoyl)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
1-(2,3-dihydro-1H-inden-2-yl)-3-(oxolan-3-yl)-5-(1H-pyrrol-2-yl)-1H-1,2,4-triazole
4-{2-[(2-chlorophenyl)methyl]morpholine-4-carbonyl}pyridin-1-ium-1-olate
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(2,5-dimethoxyphenyl)acetamide
6-(2-aminoethyl)-N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]pyrimidin-4-amine
methyl[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl](pyridin-3-ylmethyl)amine
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
(3R,9aR)-3-benzyl-8-(4-phenylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-fluoro-N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]benzamide
3-(azepane-1-carbonyl)-1-(prop-2-en-1-yl)-5-[4-(propan-2-yl)piperazin-1-yl]-4,5,6,7-tetrahydro-1H-indazole
{3-[(3-chlorophenyl)methyl]-1-(2,5-dimethylpyrimidin-4-yl)piperidin-3-yl}methanol
N-({2-[3-(4-methoxybenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-4-methyl-1,3-oxazole-5-carboxamide
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-3-(piperidin-3-yl)benzamide
4-{6-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]pyridine-3-carbonyl}morpholine
2-{[3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazin-1-yl]methyl}-5-methoxyphenol
2-{[2-(furan-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}-1-(pyridin-3-yl)ethan-1-ol
methyl[(3-phenyl-1H-pyrazol-4-yl)methyl]{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}amine
ethyl 4-{2-ethyl-6-methyl-4-oxo-1-[2-(piperidin-1-yl)ethyl]-1,4-dihydropyridine-3-amido}piperidine-1-carboxylate
(3S,5R,9R)-11-[(3-fluorophenyl)methyl]-5-hydroxy-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
1-methyl-1'-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
2-(dimethyl-1,2-oxazol-4-yl)-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}acetamide
3-{2-[(3,5-difluorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}propanamide
2-amino-2-methyl-1-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
2-ethoxy-6-{[3-(2-hydroxyethyl)-4-[(2-methylphenyl)methyl]piperazin-1-yl]methyl}phenol
3-(2-methylpropyl)-5-[5-(propan-2-yl)-1,2-oxazol-3-yl]-1H-1,2,4-triazole
3-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}propan-1-ol
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(2-phenylpropyl)-1,2-oxazole-5-carboxamide
4-(benzyloxy)-1-[3-(1H-pyrazol-4-yl)benzoyl]piperidine
1-{3-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]phenyl}piperazine
4-ethyl-9-(1-ethyl-1H-1,2,4-triazol-5-yl)-2H,3H,4H,6H,7H,8H,9H-[1,4]oxazino[2,3-g]quinoline-3,7-dione
3-{[2-(2-chlorophenyl)-3-methyl-3H-imidazo[4,5-b]pyridin-6-yl]formamido}propanamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
4-{1-[6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonyl]piperidin-4-yl}morpholine
4-[1-(propan-2-yl)-2,3-dihydro-1H-indol-5-yl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N'-[(3R,4S)-1-cyclohexyl-4-propylpyrrolidin-3-yl]pentanediamide
3-methoxy-1-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-methyl-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
4-(2-phenylethyl)-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidine
3-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-N-(propan-2-yl)propanamide
4-methyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)piperidine-4-carboxamide
6-oxo-N-{[5-(pyridin-2-yl)thiophen-2-yl]methyl}piperazine-2-carboxamide