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N-(1,4-dimethyl-1H-pyrazol-5-yl)-4-({methyl[1-(pyridin-2-yl)ethyl]amino}methyl)benzamide
(2S)-1-(3,5-dichloro-4-methylbenzoyl)pyrrolidine-2-carboxamide
1-ethyl-N-methyl-3-(piperidine-1-carbonyl)-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[1-(1-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]propan-2-ol
(2S)-2-{[3-(1H-pyrazol-1-yl)phenyl]formamido}-3-(pyridin-4-yl)propanoic acid
8-[4-(1H-imidazol-1-yl)butanoyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-2-(pyrrolidin-1-yl)benzamide
5-tert-butyl-2-{5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-1,3-benzodiazole
3-fluoro-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)benzamide
N-[1-(cyclohex-1-en-1-yl)ethyl]-3-(1-methyl-1H-pyrazol-5-yl)propanamide
2,2-dimethyl-1-[6-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]butan-1-one
1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
6-{3-oxo-3-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]propyl}-2,3-dihydropyridazin-3-one
1-methyl-N-[1-(methylcarbamoyl)cyclohexyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
3-(2-phenylethyl)-1-(1,3-thiazol-2-yl)piperidine
9-(5-propyl-1,3,4-thiadiazol-2-yl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(dimethyl-1,2-oxazol-4-yl)-N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)propanamide
(butan-2-yl)({[4-(1H-pyrazol-1-yl)phenyl]methyl})(pyridin-4-ylmethyl)amine
(2E)-N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(pyridin-2-yl)prop-2-enamide
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-2-(3-methylphenyl)acetamide
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-N-(2-hydroxyethyl)oxolane-2-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-2-one
ethyl 4-{[(2-propyl-1,3-thiazol-4-yl)methyl]amino}piperidine-1-carboxylate
5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)furan-2-carboxamide
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
5-[4-(1,2-benzothiazol-3-yl)piperazine-1-carbonyl]-1-ethylpiperidin-2-one
1-(4-{2-oxo-2-[3-(pyridin-3-yl)azetidin-1-yl]ethyl}phenyl)imidazolidin-2-one
1-[(4-fluorophenyl)methyl]-5-(4-methoxy-3,5-dimethylbenzoyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole
(1R,5S,6S)-6-{[4-(naphthalen-2-yl)piperazin-1-yl]methyl}-3-azabicyclo[3.1.0]hexane
6-{[(2R)-1-ethylpyrrolidin-2-yl]methyl}-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
4-{[5-(3-methoxypyrazin-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}thiomorpholine
2-(dimethylamino)-7-[1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-{3,9-diazaspiro[5.6]dodecane-9-carbonyl}pyridin-2-ol
1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-5-[2-({[3-(trifluoromethyl)phenyl]methyl}amino)ethyl]pyrrolidin-2-one
3-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)pyridin-2-ol
2-cyclopropyl-8-[(4-methoxypyridin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
methyl 2-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]pyridine-4-carboxylate
2-(4-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-diazepan-1-yl)-N,N-dimethylacetamide
N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-2,2-diphenylacetamide
methyl 4-[7-(5-chloropyridin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-4-oxobutanoate
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-(2-methoxyethyl)-N-(propan-2-yl)acetamide
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(3-fluoro-4-methylbenzoyl)piperidine
6-chloro-2-{[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]methyl}-1,4-dihydroquinolin-4-one
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-4-(1H-1,2,4-triazol-3-yl)benzamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[(1r,4r)-4-hydroxycyclohexyl]piperidin-2-one
N-[(2R,3R)-2-(2-methoxyethoxy)-1'-(1,3-thiazol-2-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
1-[(2-methylphenyl)methyl]-4-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperazine
3-{2-[3-(2-fluorophenoxy)azetidin-1-yl]-2-oxoethyl}-5,5-dimethyl-1,3-oxazolidine-2,4-dione
methyl 1-[2-(1H-indol-3-yl)ethyl]-3-(2-methoxyacetamido)-5-[(1-methoxypropan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-(2-hydroxyethyl)-N-methyl-4-{octahydropyrrolo[1,2-a]piperazine-2-sulfonyl}benzamide