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N,5,6-trimethyl-N-[(3-methyloxetan-3-yl)methyl]thieno[2,3-d]pyrimidin-4-amine
2-(2-fluoro-3-methoxyphenyl)-2-(thiomorpholin-4-yl)acetic acid
3-(morpholine-4-carbonyl)-1-propyl-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazol-3-yl)ethan-1-one
2-{4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
3-[4-(6-methoxypyridin-3-yl)-1H-1,2,3-triazol-1-yl]-2,3-dihydro-1λ6-thiophene-1,1-dione
[(5-{[(3-fluorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl](methyl)(pyridin-2-ylmethyl)amine
4-({2-[3-(4H-1,2,4-triazol-4-yl)phenyl]phenyl}methyl)morpholine
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-1,4-dithiepan-6-amine
2-{2-[(4-methyl-3-oxopiperazin-1-yl)methyl]-4-(pyrimidin-2-yl)phenoxy}acetic acid
2-[methyl({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]-1-phenylethan-1-ol
1-(1-methyl-1H-imidazole-2-carbonyl)-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
7-cyclopropanecarbonyl-N-[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-[4-(4-{methyl[2-(4-methylphenoxy)ethyl]amino}piperidin-1-yl)benzoyl]piperidin-3-ol
4-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-sulfonyl]-N-cyclopropylbenzamide
2-methoxy-5-[2-(1-phenylethyl)-1H-imidazol-1-yl]pyridine
[(2-cyclohexylpyrimidin-5-yl)methyl](methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
2-(4-acetylphenoxy)-1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidin-1-yl}-3-(1-methylpiperidin-2-yl)propan-1-one
7-(2-cyclohexylethyl)-2-(thiophene-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]butan-1-one
2-({3-[(3,4-difluorophenyl)amino]piperidin-1-yl}methyl)-6-ethoxyphenol
1-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]-2-(methylsulfanyl)ethan-1-one
2-butyl-1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-2,5-dihydro-1H-pyrrole
6-(4-{1-azabicyclo[2.2.2]octan-3-yl}piperazin-1-yl)-5-chloropyridine-3-carboxylic acid
N-(2-methyl-1-benzofuran-5-yl)-2-[2-(morpholin-4-yl)ethyl]piperidine-1-carboxamide
N-(2-methoxyethyl)-1-methyl-6-oxo-N-(pyridin-4-ylmethyl)-1,6-dihydropyridine-3-carboxamide
2-[2-({dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}amino)ethyl]-6-phenyl-2,3-dihydropyridazin-3-one
(3S,4S)-4-cyclopropyl-1-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]pyrrolidine-3-carboxylic acid
2-methoxy-N-[(1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)methyl]acetamide
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
3-(8-chloro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-1-(1,4-oxazepan-6-ylmethyl)urea
1-{2-[(4-methoxyphenyl)methyl]morpholin-4-yl}-3-(methylsulfanyl)propan-1-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-phenoxybutanamide
4-[1-(4-chloro-2-methoxy-5-methylphenyl)-1H-imidazol-2-yl]-2-methyl-1,3-oxazole
9-(3-methylfuran-2-carbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
2-[(4-chlorophenyl)methyl]-N-methyl-N-[2-(1,2,4-oxadiazol-3-yl)ethyl]-1,3-benzoxazole-5-carboxamide
5-(3-methoxyphenoxymethyl)-N-(oxolan-2-ylmethyl)-1H-pyrazole-3-carboxamide
2-[1-(3-methylbut-2-en-1-yl)-4-(3-phenylprop-2-yn-1-yl)piperazin-2-yl]ethan-1-ol
4-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-4-methylpiperidine
3-{1-[1-(3-fluorobenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(3-fluorophenyl)urea
2-{2-methyl-4-[(prop-2-en-1-yl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-1,3-thiazole-4-carboxamide
3-{[4-(3-hydroxyphenyl)piperidin-1-yl]methyl}-7-methoxy-1,2-dihydroquinolin-2-one
2-[1-butyl-5-(4-ethanesulfonamidophenyl)-1H-1,2,4-triazol-3-yl]acetamide
(propan-2-yl)({[5-(pyrimidin-2-ylsulfanyl)furan-2-yl]methyl})[(trimethyl-1H-pyrazol-4-yl)methyl]amine
5-methoxy-N-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}furan-2-carboxamide
(1S,2R)-2-({[2-(difluoromethoxy)phenyl]methyl}(methyl)amino)cyclohexan-1-ol
3-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
2-({[3-(hydroxymethyl)-2,4,6-trimethylphenyl]methyl}(thiophen-2-ylmethyl)amino)butan-1-ol
2-[2-(2-methoxy-4-methylphenoxymethyl)-1,3-oxazole-4-carbonyl]-1,2-oxazinane