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(3aS,7aR)-2-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-6-methyl-2-oxo-4-(pyridin-3-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
(1S,2S)-2-({6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)cyclohexan-1-ol
3-(2-phenoxyethyl)-8-(1,3-thiazol-4-ylmethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-({3-hydroxy-1-[(3-methoxyphenyl)methyl]-2-oxopiperidin-3-yl}methyl)piperazin-2-one
{1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}(1-methyl-1H-imidazol-2-yl)methanol
2-(2-hydroxyethyl)-9-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
(2E)-1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-3-phenylprop-2-en-1-one
N-methyl-N-(1,2-oxazol-3-ylmethyl)-2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
5-(2,2-dimethylpropanoyl)-N-[(4-methoxyphenyl)methyl]-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
7-(3,6-dimethylpyrazin-2-yl)-9-methoxy-4-(thiophen-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
7-chloro-N-ethyl-N-[(1R,2R)-2-hydroxycyclohexyl]-2-methylquinoline-4-carboxamide
(2S,4R)-1-benzyl-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}-N-(propan-2-yl)pyrrolidine-2-carboxamide
{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}(oxolan-2-ylmethyl)(pyridin-4-ylmethyl)amine
2-{2-ethyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-N-methylacetamide
2-[4-(2-propyl-1H-imidazol-1-yl)phenoxy]propanamide
3-oxo-N-[3-(pyridin-4-yl)propyl]-3,4-dihydroquinoxaline-2-carboxamide
(2S,4S)-N-ethyl-4-(4-{[(2E)-3-phenylprop-2-enamido]methyl}-1H-1,2,3-triazol-1-yl)pyrrolidine-2-carboxamide
2-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1H-indole
N-[(3S,4R)-4-(4-methoxyphenyl)-1-[2-(thiophen-2-yl)acetyl]pyrrolidin-3-yl]acetamide
(8R,9aS)-8-hydroxy-2-[2-(7-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
4-(3-hydroxy-3-methylbutyl)-N-[1-(thiophen-2-ylmethyl)piperidin-3-yl]benzamide
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}({[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl})amine
S-[2-(2,2-dimethylpropanoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-3-hydroxybutane-1-sulfonamido
7-(3-chlorophenyl)-4-[(dimethyl-1,2-oxazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-5,6,7,8-tetrahydroquinoline-3-carbonitrile
N-[2-(1H-imidazol-1-yl)propyl]-1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[(1S,2S)-2-[(4-fluorophenyl)methyl]cyclopentyl]-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-(pyrrolidin-3-yl)benzamide
1-(3-hydroxy-3-phenylpyrrolidin-1-yl)-2-(2,5,7-trimethyl-1H-indol-3-yl)ethan-1-one
ethyl 2-(1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)acetate
3-[2-(4-fluorophenyl)piperidin-1-yl]-1-(pyrrolidin-1-yl)propan-1-one
2-ethyl-8-(2-hydroxy-3-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
6-[({2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}amino)methyl]-1,4-oxazepan-6-ol
N3-cycloheptyl-1-cyclopropyl-4-oxo-N5-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-(4-fluorophenoxymethyl)-4-hydroxy-N-(1-phenylcyclopropyl)pyrimidine-5-carboxamide
methyl[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl](quinoxalin-5-ylmethyl)amine
(3aS,6aS)-2-[(3-fluorophenyl)methyl]-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-4-methylpyrimidine
N-[1-(4-fluorophenyl)-4-(2-oxo-1,3-oxazolidin-3-yl)-1H-indazol-3-yl]-2-(methylsulfanyl)acetamide
7-[(2,3-difluorophenyl)methyl]-2-[(2-ethylpyrimidin-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
4-(1H-imidazol-1-ylmethyl)-1-{[3-(5-methylfuran-2-yl)phenyl]methyl}piperidin-4-ol
3-(2,3-dimethylphenyl)-5-(2-ethoxyethyl)-1,2,4-oxadiazole
5-methoxy-9-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-1-oxa-9-azaspiro[5.5]undecane
(2-methoxyethyl)({2-phenyl-1-[1-(thiophen-2-ylmethyl)piperidin-4-yl]ethyl})(pyridin-2-ylmethyl)amine
1-[4-({4-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-one
N,2-dimethyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]pyrido[2,3-d]pyrimidin-4-amine
(3R)-3-[4-(4-fluorophenyl)-1,4-diazepane-1-carbonyl]-1,2,3,4-tetrahydroisoquinoline
(1S,5R)-6-benzyl-3-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[3-cyclopropyl-5-(methoxymethyl)-1H-1,2,4-triazol-1-yl]-2-methylpyridine