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{3-propyl-1-[5-(pyrrolidin-1-ylmethyl)pyridin-2-yl]piperidin-3-yl}methanol
4-(3-methylbutyl)-3-{2-oxo-2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]ethyl}piperazin-2-one
4-(1-{1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
4-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}-1,4-oxazepan-6-ol
4-(1-benzofuran-2-ylmethyl)-9-ethyl-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-ethyl-N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-3,5-dimethyl-1,2-oxazole-4-carboxamide
ethyl({[6-(4-fluorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl})[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
2-(2-methylpropyl)-8-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}-2,8-diazaspiro[4.5]decan-3-one
3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]piperidine
N-(3-chloro-4-methoxyphenyl)-4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carboxamide
7-(2-methoxyethyl)-2-(1-methyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-3,5,7-trimethyl-1H-indole-2-carboxamide
(3S,5R)-1-(6-oxo-1,6-dihydropyridine-3-carbonyl)-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
{5-[(3S)-3-(dimethylamino)azepane-1-carbonyl]-1H-1,3-benzodiazol-2-yl}methanol
4-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2,3-dihydro-1H-imidazol-2-one
N-[2-chloro-5-(pyrrolidine-1-carbonyl)phenyl]-1,1-dioxo-1λ6-thiomorpholine-4-carboxamide
1-[(2E)-3-phenylprop-2-en-1-yl]-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
7-(1-benzothiophen-3-yl)-4-(3-hydroxypropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperazine
1-cyclohexyl-N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]piperidine-4-carboxamide
4-(4-methoxy-3-methylphenyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
4-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-3-(3-fluorophenyl)piperazin-2-one
(cyclohex-3-en-1-ylmethyl)(methyl)(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amine
2-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-3,5,7-trimethyl-1H-indole
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]but-3-enamide
(3-methyl-1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methanol
8-(1H-indol-3-ylmethyl)-1-methyl-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(furan-3-ylmethyl)-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
3-(1-methyl-1H-imidazol-2-yl)-6-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]pyridazine
ethyl 4-[4-(cyclohexylmethyl)-3-oxo-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-11-yl]piperazine-1-carboxylate
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}pyrrolidine-1-sulfonamide
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-N,2,3,6-tetramethylquinoline-4-carboxamide
5-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}-3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-propylimidazolidine-2,4-dione
5-oxo-1-[4-(propan-2-yl)phenyl]-N-[2-(pyridin-3-yl)ethyl]pyrrolidine-3-carboxamide
2-[(3-{[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]carbamoyl}phenyl)amino]acetic acid
1-methyl-N-[2-(4-phenylpyrimidin-2-yl)ethyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-(3-ethyladamantan-1-yl)-3-(3-methyl-1,2,4-thiadiazol-5-yl)urea
6-(4-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl}piperazin-1-yl)pyridine-3-carbonitrile
N-({5-[(5-chlorothiophen-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
5-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl}-1-methyl-1H-1,2,3-benzotriazole
1-(2,2-dimethoxyethyl)-4-(3-methyl-1H-pyrazole-5-carbonyl)piperazine
2-[4-ethoxy-3-methoxy-5-(prop-2-en-1-yl)phenyl]-1H-imidazole
(1R,5S)-3-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-3,8-diazabicyclo[3.2.1]octane
2-(3,4-dichlorophenyl)pyridine-4-carboxamide
4-(3-methylphenoxy)-1-(1-methylpyrrolidine-3-carbonyl)piperidine-4-carboxylic acid
methyl 3-[(3S,4R)-3-acetamido-4-propylpyrrolidine-1-carbonyl]-5-methoxybenzoate
1-[5-(piperidin-1-ylmethyl)imidazo[2,1-b][1,3]thiazole-6-carbonyl]azocane
2-{4-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]piperidin-1-yl}acetamide
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
(2R)-2-amino-N-[(3-methoxyphenyl)methyl]-3-phenyl-N-(prop-2-en-1-yl)propanamide