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4-methyl-2-{2-[(5-methyl-1-propyl-1H-pyrazol-4-yl)formamido]ethyl}-1,3-thiazole-5-carboxylic acid
(3aR,6aR)-2-benzyl-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
(2S,4R)-4-amino-N,N-diethyl-1-[(2E)-3-phenylprop-2-enoyl]pyrrolidine-2-carboxamide
(3aR,5R,6S,7aS)-2-[1-(4-methylphenyl)piperidin-4-yl]-octahydro-1H-isoindole-5,6-diol
6-ethyl-4-({methyl[1-(pyrimidin-4-yl)ethyl]amino}methyl)-2H-chromen-2-one
1-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-3-(methylsulfanyl)propan-1-one
6-[1-(3-chloro-4-fluorophenyl)-1H-1,2,4-triazol-5-yl]-2-methyl-2H,3H,5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-one
methyl 3-(2-methoxyacetamido)-5-[(quinolin-2-ylformamido)methyl]benzoate
(3R,4R)-4-(azepan-1-yl)-1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-ol
5-[(2-methoxyethyl)amino]-1-methyl-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-3-(4-benzylpiperazine-1-carbonyl)-6-methyl-2-propyl-1,4-dihydropyridin-4-one
2-{[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl}-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
2-{methyl[3-(pyrrolidin-1-yl)butyl]amino}acetic acid
3-phenoxy-N-[1-({[(4-phenyloxan-4-yl)methyl]carbamoyl}methyl)-1H-pyrazol-4-yl]propanamide
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]pyrrolidin-3-yl]methanol
2-methoxy-6-{[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]methyl}phenol
1-(oxolan-3-ylmethyl)-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
N3-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-N1,N1-dimethylpiperidine-1,3-dicarboxamide
N-(4-{[(3-phenylpropyl)carbamoyl]methyl}phenyl)butanamide
1-(diethylcarbamoyl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
3-[(furan-2-ylformamido)methyl]-N-(2-phenylphenyl)piperidine-1-carboxamide
5-{[(2-benzyl-1,3-thiazol-4-yl)formamido]methyl}thiophene-2-carboxylic acid
8-(3-hydroxypyridine-2-carbonyl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
5,6-dimethyl-1-(pyrimidin-5-yl)-1H-1,3-benzodiazole
2-chloro-N-[1-(1-{[4-(propan-2-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]benzamide
N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-3-propyl-1H-pyrazole-4-carboxamide
5-[({[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)methyl]-N-methylpyrimidin-2-amine
4-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methoxy}benzamide
1-[(1R,2R)-2-(benzyloxy)cyclopentyl]-3-(2-methyl-2H-1,2,3-benzotriazol-4-yl)urea
N-methyl-N-(1,2-oxazol-3-ylmethyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-[4-(5-oxo-1-phenyl-2,5-dihydro-1H-pyrazole-3-carbonyl)morpholin-3-yl]acetic acid
N-[(6-methylquinolin-5-yl)methyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
ethyl 5-{[(2-benzyl-1,3-benzoxazol-5-yl)formamido]methyl}furan-2-carboxylate
2-{5-[(2-benzylmorpholin-4-yl)methyl]furan-2-yl}benzonitrile
2-{1-[(2,3-difluoro-6-methoxyphenyl)methyl]piperidin-2-yl}pyridine
(4S)-1-[(2,5-dichlorophenyl)methyl]-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
6-methyl-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}pyridine-3-carboxamide
N,N-dimethyl-2-[(1S,5R)-3-(5-methylthiophene-2-carbonyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
2-[2-(hydroxymethyl)-1H-1,3-benzodiazol-5-yl]benzamide
2-methyl-6-(piperidin-3-yl)-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]pyrimidin-4-amine
1-{3-[5-(4-fluoro-2-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]propyl}-1H-1,2,4-triazole
2-(adamantan-1-yl)-N-[(2R)-1-hydroxy-3-phenylpropan-2-yl]acetamide
methyl 3-{2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamido}propanoate
5-(2-chlorophenyl)-N-(1,1-dioxo-1λ6-thian-4-yl)-N-methylfuran-2-carboxamide
6-({5H,6H,7H-cyclopenta[b]pyridin-7-yl}amino)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
1-[benzyl(methyl)amino]-3-{5-[(4-ethylpiperazin-1-yl)methyl]-2-methoxyphenoxy}propan-2-ol
3-(4-phenylbenzoyl)piperidine
N-[(3S,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-methoxybenzamide
5-methyl-1-propyl-N-[1-(pyridine-4-carbonyl)piperidin-4-yl]-1H-pyrazole-4-carboxamide